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Assay Detail

CHEMBL1614164

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
PUBCHEM_BIOASSAY: Fluorescence Cell-Based Retest of Candida albicans Growth in the Presence of Fluconazole. (Class of assay: confirmatory) [Related pubchem assays: 2007 (Project Summary), 1979 (Primary HTS)]
1721
Total Activities
1718
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Category confirmatory
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

PubChem BioAssay data set

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1721 5.93 7.48

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1401052 1 7.48
CHEMBL1242180 1 7.46
CHEMBL1518873 1 7.46
CHEMBL3212594 1 7.44
CHEMBL1309091 1 7.43
CHEMBL1500188 1 7.41
CHEMBL1412223 1 7.40
CHEMBL1609759 1 7.39
CHEMBL1519955 1 7.36
CHEMBL1315921 1 7.34
CHEMBL1318350 1 7.34
CHEMBL1587683 1 7.34
CHEMBL1322948 1 7.34
CHEMBL1425546 1 7.34
CHEMBL453974 1 7.31
CHEMBL1789993 1 7.30
CHEMBL466853 1 7.29
CHEMBL1497897 1 7.28
CHEMBL1587806 1 7.27
CHEMBL584458 1 7.27
CHEMBL1562664 1 7.26
CHEMBL1789998 1 7.26
CHEMBL140425 1 7.26
CHEMBL388590 BENZBROMARONE 4.0 1 7.23
CHEMBL1384718 1 7.19
CHEMBL1964793 1 7.17
CHEMBL1388738 1 7.16
CHEMBL1524829 1 7.15
CHEMBL1419164 1 7.09
CHEMBL1452795 1 7.08

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1401052 EC50 = 33.0 nM 7.48
CHEMBL1518873 EC50 = 35.0 nM 7.46
CHEMBL1242180 EC50 = 35.0 nM 7.46
CHEMBL3212594 EC50 = 36.0 nM 7.44
CHEMBL1309091 EC50 = 37.0 nM 7.43
CHEMBL1500188 EC50 = 39.0 nM 7.41
CHEMBL1412223 EC50 = 40.0 nM 7.40
CHEMBL1609759 EC50 = 41.0 nM 7.39
CHEMBL1519955 EC50 = 44.0 nM 7.36
CHEMBL1315921 EC50 = 46.0 nM 7.34
CHEMBL1425546 EC50 = 46.0 nM 7.34
CHEMBL1318350 EC50 = 46.0 nM 7.34
CHEMBL1587683 EC50 = 46.0 nM 7.34
CHEMBL1322948 EC50 = 46.0 nM 7.34
CHEMBL453974 EC50 = 49.0 nM 7.31
CHEMBL1789993 EC50 = 50.0 nM 7.30
CHEMBL466853 EC50 = 51.0 nM 7.29
CHEMBL1497897 EC50 = 52.0 nM 7.28
CHEMBL1587806 EC50 = 54.0 nM 7.27
CHEMBL584458 EC50 = 54.0 nM 7.27
CHEMBL140425 EC50 = 55.0 nM 7.26
CHEMBL1562664 EC50 = 55.0 nM 7.26
CHEMBL1789998 EC50 = 55.0 nM 7.26
CHEMBL388590 BENZBROMARONE EC50 = 59.0 nM 7.23
CHEMBL1384718 EC50 = 65.0 nM 7.19
CHEMBL1964793 EC50 = 68.0 nM 7.17
CHEMBL1388738 EC50 = 69.0 nM 7.16
CHEMBL1524829 EC50 = 71.0 nM 7.15
CHEMBL1419164 EC50 = 82.0 nM 7.09
CHEMBL334707 EC50 = 84.0 nM 7.08
CHEMBL1452795 EC50 = 83.0 nM 7.08
CHEMBL1464485 EC50 = 92.0 nM 7.04
CHEMBL1488279 EC50 = 95.0 nM 7.02
CHEMBL1528425 EC50 = 98.0 nM 7.01
CHEMBL1364999 EC50 = 97.0 nM 7.01
CHEMBL1392455 EC50 = 101.0 nM 7.00
CHEMBL1464391 EC50 = 101.0 nM 7.00
CHEMBL1578482 EC50 = 100.0 nM 7.00
CHEMBL1580315 EC50 = 102.0 nM 6.99
CHEMBL1790008 EC50 = 111.0 nM 6.96
CHEMBL1477033 EC50 = 110.0 nM 6.96
CHEMBL3189966 EC50 = 114.0 nM 6.94
CHEMBL1484777 EC50 = 117.0 nM 6.93
CHEMBL1308432 EC50 = 119.0 nM 6.92
CHEMBL1580272 EC50 = 119.0 nM 6.92
CHEMBL1472773 EC50 = 121.0 nM 6.92
CHEMBL1342833 EC50 = 123.0 nM 6.91
CHEMBL1606685 EC50 = 122.0 nM 6.91
CHEMBL1346822 EC50 = 126.0 nM 6.90
CHEMBL1340114 EC50 = 130.0 nM 6.89