Assay Detail
Binding
CHEMBL1613985
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: HTS discovery of chemical inhibitors of anti-apoptotic protein Bfl-1. (Class of assay: confirmatory) [Related pubchem assays: 621 ]
44
Total Activities
44
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Mus musculus |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 44 | 5.14 | 6.19 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1271764 | — | — | 1 | 6.19 |
| CHEMBL1351212 | — | — | 1 | 5.54 |
| CHEMBL1381644 | — | — | 1 | 5.46 |
| CHEMBL1449204 | — | — | 1 | 5.43 |
| CHEMBL1417970 | — | — | 1 | 5.42 |
| CHEMBL1548175 | — | — | 1 | 5.32 |
| CHEMBL1526405 | — | — | 1 | 5.26 |
| CHEMBL1346587 | — | — | 1 | 5.24 |
| CHEMBL1399711 | — | — | 1 | 5.21 |
| CHEMBL1312063 | — | — | 1 | 5.05 |
| CHEMBL1331084 | — | — | 1 | 4.95 |
| CHEMBL1503307 | — | — | 1 | 4.85 |
| CHEMBL1305391 | — | — | 1 | 4.84 |
| CHEMBL1550296 | — | — | 1 | 4.74 |
| CHEMBL1516834 | — | — | 1 | 4.65 |
| CHEMBL1353989 | — | — | 1 | 4.61 |
| CHEMBL1371774 | — | — | 1 | 4.59 |
| CHEMBL1406829 | — | — | 1 | - |
| CHEMBL1310494 | — | — | 1 | - |
| CHEMBL1507695 | — | — | 1 | - |
| CHEMBL3392041 | — | — | 1 | - |
| CHEMBL1393593 | — | — | 1 | - |
| CHEMBL1365898 | — | — | 1 | - |
| CHEMBL1505982 | — | — | 1 | - |
| CHEMBL1610465 | — | — | 1 | - |
| CHEMBL1612321 | — | — | 1 | - |
| CHEMBL1373720 | — | — | 1 | - |
| CHEMBL1501864 | — | — | 1 | - |
| CHEMBL1487918 | — | — | 1 | - |
| CHEMBL1438721 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1271764 | — | IC50 | = | 650.0 | nM | 6.19 |
| CHEMBL1351212 | — | IC50 | = | 2850.0 | nM | 5.54 |
| CHEMBL1381644 | — | IC50 | = | 3491.2 | nM | 5.46 |
| CHEMBL1449204 | — | IC50 | = | 3720.0 | nM | 5.43 |
| CHEMBL1417970 | — | IC50 | = | 3780.0 | nM | 5.42 |
| CHEMBL1548175 | — | IC50 | = | 4790.0 | nM | 5.32 |
| CHEMBL1526405 | — | IC50 | = | 5440.0 | nM | 5.26 |
| CHEMBL1346587 | — | IC50 | = | 5820.0 | nM | 5.24 |
| CHEMBL1399711 | — | IC50 | = | 6150.0 | nM | 5.21 |
| CHEMBL1312063 | — | IC50 | = | 8880.0 | nM | 5.05 |
| CHEMBL1331084 | — | IC50 | = | 11200.0 | nM | 4.95 |
| CHEMBL1503307 | — | IC50 | = | 14100.0 | nM | 4.85 |
| CHEMBL1305391 | — | IC50 | = | 14459.0 | nM | 4.84 |
| CHEMBL1550296 | — | IC50 | = | 18100.0 | nM | 4.74 |
| CHEMBL1516834 | — | IC50 | = | 22400.0 | nM | 4.65 |
| CHEMBL1353989 | — | IC50 | = | 24600.0 | nM | 4.61 |
| CHEMBL1371774 | — | IC50 | = | 25400.0 | nM | 4.59 |
| CHEMBL1534131 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1385840 | ERGOCORNINE | IC50 | > | 100000.0 | nM | - |
| CHEMBL1379677 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1532568 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1402456 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL166209 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1449293 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL503 | LOVASTATIN | IC50 | > | 100000.0 | nM | - |
| CHEMBL1068 | OXCARBAZEPINE | IC50 | > | 100000.0 | nM | - |
| CHEMBL1568497 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1369154 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1498529 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1478187 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1399595 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1438721 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1487918 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1501864 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1373720 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1612321 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1610465 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1505982 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1365898 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1393593 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL3392041 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1507695 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1310494 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1406829 | — | IC50 | > | 100000.0 | nM | - |