Assay Detail
Functional
CHEMBL1614035
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Dose Response confirmation of HTS hits from an HePTP Fluorescent Assay using OMFP substrate - Set 2. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID1059, AID1077, AID1784, AID2068, AID2085, AID2134, AID521]
140
Total Activities
140
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Tyrosine-protein phosphatase non-receptor type 7 (CHEMBL2219) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 140 | 4.96 | 5.78 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1536896 | — | — | 1 | 5.78 |
| CHEMBL1320181 | — | — | 1 | 5.62 |
| CHEMBL2001743 | — | — | 1 | 5.60 |
| CHEMBL1438889 | — | — | 1 | 5.42 |
| CHEMBL2000167 | — | — | 1 | 5.41 |
| CHEMBL1426096 | — | — | 1 | 5.38 |
| CHEMBL570345 | — | — | 1 | 5.35 |
| CHEMBL1424694 | — | — | 1 | 5.31 |
| CHEMBL1471865 | — | — | 1 | 5.21 |
| CHEMBL1580263 | — | — | 1 | 5.17 |
| CHEMBL3190951 | — | — | 1 | 5.13 |
| CHEMBL1488035 | — | — | 1 | 5.05 |
| CHEMBL599924 | — | — | 1 | 4.99 |
| CHEMBL1529554 | — | — | 1 | 4.96 |
| CHEMBL1527520 | — | — | 1 | 4.95 |
| CHEMBL1492305 | — | — | 1 | 4.94 |
| CHEMBL1439815 | — | — | 1 | 4.91 |
| CHEMBL1371816 | — | — | 1 | 4.84 |
| CHEMBL1443268 | — | — | 1 | 4.83 |
| CHEMBL1981200 | — | — | 1 | 4.83 |
| CHEMBL1533230 | — | — | 1 | 4.75 |
| CHEMBL1464805 | — | — | 1 | 4.31 |
| CHEMBL1976414 | — | — | 1 | 4.31 |
| CHEMBL1417070 | — | — | 1 | 4.30 |
| CHEMBL1576746 | — | — | 1 | 4.24 |
| CHEMBL1309430 | — | — | 1 | 4.16 |
| CHEMBL1583199 | — | — | 1 | 4.13 |
| CHEMBL3208812 | — | — | 1 | - |
| CHEMBL1412887 | — | — | 1 | - |
| CHEMBL1323857 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1536896 | — | IC50 | = | 1678.0 | nM | 5.78 |
| CHEMBL1320181 | — | IC50 | = | 2414.0 | nM | 5.62 |
| CHEMBL2001743 | — | IC50 | = | 2519.0 | nM | 5.60 |
| CHEMBL1438889 | — | IC50 | = | 3780.0 | nM | 5.42 |
| CHEMBL2000167 | — | IC50 | = | 3928.0 | nM | 5.41 |
| CHEMBL1426096 | — | IC50 | = | 4198.0 | nM | 5.38 |
| CHEMBL570345 | — | IC50 | = | 4500.0 | nM | 5.35 |
| CHEMBL1424694 | — | IC50 | = | 4892.0 | nM | 5.31 |
| CHEMBL1471865 | — | IC50 | = | 6178.0 | nM | 5.21 |
| CHEMBL1580263 | — | IC50 | = | 6845.0 | nM | 5.17 |
| CHEMBL3190951 | — | IC50 | = | 7331.0 | nM | 5.13 |
| CHEMBL1488035 | — | IC50 | = | 8913.0 | nM | 5.05 |
| CHEMBL599924 | — | IC50 | = | 10295.0 | nM | 4.99 |
| CHEMBL1529554 | — | IC50 | = | 10923.0 | nM | 4.96 |
| CHEMBL1527520 | — | IC50 | = | 11211.0 | nM | 4.95 |
| CHEMBL1492305 | — | IC50 | = | 11523.0 | nM | 4.94 |
| CHEMBL1439815 | — | IC50 | = | 12190.0 | nM | 4.91 |
| CHEMBL1371816 | — | IC50 | = | 14604.0 | nM | 4.84 |
| CHEMBL1981200 | — | IC50 | = | 14931.0 | nM | 4.83 |
| CHEMBL1443268 | — | IC50 | = | 14611.0 | nM | 4.83 |
| CHEMBL1533230 | — | IC50 | = | 17939.0 | nM | 4.75 |
| CHEMBL1464805 | — | IC50 | = | 48744.0 | nM | 4.31 |
| CHEMBL1976414 | — | IC50 | = | 49146.0 | nM | 4.31 |
| CHEMBL1417070 | — | IC50 | = | 49831.0 | nM | 4.30 |
| CHEMBL1576746 | — | IC50 | = | 58190.0 | nM | 4.24 |
| CHEMBL1309430 | — | IC50 | = | 69263.0 | nM | 4.16 |
| CHEMBL1583199 | — | IC50 | = | 74275.0 | nM | 4.13 |
| CHEMBL1335318 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1467425 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1326115 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1549636 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1606761 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1535241 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1338178 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1360572 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1600686 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL3212510 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1499300 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1993612 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1414751 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1493152 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1337760 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1301248 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1490435 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1371394 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1431216 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1344691 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1505659 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1534728 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1444510 | — | IC50 | > | 79400.0 | nM | - |