Assay Detail
Functional
CHEMBL1614318
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Luminescence-based dose response cell-based high throughput screening assay for cytotoxic compounds using the IEC-6 intestinal epithelial cell line. (Class of assay: confirmatory) [Related pubchem assays: 1858 (Summary AID.), 1825 (Counterscreen.), 1907 (Confirmation screen.)]
122
Total Activities
122
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Cell Type | Epithelial cell |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 122 | 6.21 | 8.03 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL11417 | STREPTONIGRIN | 2.0 | 1 | 8.03 |
| CHEMBL513000 | — | — | 1 | 7.46 |
| CHEMBL61 | PODOFILOX | 4.0 | 1 | 7.33 |
| CHEMBL1455468 | — | — | 1 | 7.33 |
| CHEMBL1504768 | — | — | 1 | 7.27 |
| CHEMBL1329221 | — | — | 1 | 7.27 |
| CHEMBL1405453 | — | — | 1 | 7.25 |
| CHEMBL1479301 | — | — | 1 | 7.21 |
| CHEMBL107 | COLCHICINE | 4.0 | 1 | 7.20 |
| CHEMBL304291 | — | — | 1 | 7.14 |
| CHEMBL1998521 | — | — | 1 | 7.12 |
| CHEMBL1357620 | — | — | 1 | 7.10 |
| CHEMBL1536981 | — | — | 1 | 7.05 |
| CHEMBL1610049 | — | — | 1 | 7.02 |
| CHEMBL1473676 | — | — | 1 | 7.00 |
| CHEMBL1540099 | — | — | 1 | 7.00 |
| CHEMBL3189873 | — | — | 1 | 6.99 |
| CHEMBL1461711 | — | — | 1 | 6.95 |
| CHEMBL323668 | — | — | 1 | 6.92 |
| CHEMBL1524921 | — | — | 1 | 6.87 |
| CHEMBL1595169 | — | — | 1 | 6.85 |
| CHEMBL460601 | — | — | 1 | 6.84 |
| CHEMBL579318 | — | — | 1 | 6.80 |
| CHEMBL1560237 | — | — | 1 | 6.80 |
| CHEMBL1580075 | — | — | 1 | 6.75 |
| CHEMBL3191874 | — | — | 1 | 6.74 |
| CHEMBL1523841 | — | — | 1 | 6.72 |
| CHEMBL1452795 | — | — | 1 | 6.65 |
| CHEMBL1367034 | — | — | 1 | 6.64 |
| CHEMBL3197177 | — | — | 1 | 6.61 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL11417 | STREPTONIGRIN | IC50 | = | 9.4 | nM | 8.03 |
| CHEMBL513000 | — | IC50 | = | 34.57 | nM | 7.46 |
| CHEMBL61 | PODOFILOX | IC50 | = | 46.82 | nM | 7.33 |
| CHEMBL1455468 | — | IC50 | = | 47.11 | nM | 7.33 |
| CHEMBL1329221 | — | IC50 | = | 53.3 | nM | 7.27 |
| CHEMBL1504768 | — | IC50 | = | 53.95 | nM | 7.27 |
| CHEMBL1405453 | — | IC50 | = | 55.81 | nM | 7.25 |
| CHEMBL1479301 | — | IC50 | = | 61.84 | nM | 7.21 |
| CHEMBL107 | COLCHICINE | IC50 | = | 62.79 | nM | 7.20 |
| CHEMBL304291 | — | IC50 | = | 71.94 | nM | 7.14 |
| CHEMBL1998521 | — | IC50 | = | 76.23 | nM | 7.12 |
| CHEMBL1357620 | — | IC50 | = | 79.45 | nM | 7.10 |
| CHEMBL1536981 | — | IC50 | = | 89.48 | nM | 7.05 |
| CHEMBL1610049 | — | IC50 | = | 96.0 | nM | 7.02 |
| CHEMBL1540099 | — | IC50 | = | 100.56 | nM | 7.00 |
| CHEMBL1473676 | — | IC50 | = | 100.7 | nM | 7.00 |
| CHEMBL3189873 | — | IC50 | = | 103.09 | nM | 6.99 |
| CHEMBL1461711 | — | IC50 | = | 112.2 | nM | 6.95 |
| CHEMBL323668 | — | IC50 | = | 120.86 | nM | 6.92 |
| CHEMBL1524921 | — | IC50 | = | 135.67 | nM | 6.87 |
| CHEMBL1595169 | — | IC50 | = | 139.92 | nM | 6.85 |
| CHEMBL460601 | — | IC50 | = | 145.75 | nM | 6.84 |
| CHEMBL579318 | — | IC50 | = | 157.68 | nM | 6.80 |
| CHEMBL1560237 | — | IC50 | = | 157.02 | nM | 6.80 |
| CHEMBL1580075 | — | IC50 | = | 177.15 | nM | 6.75 |
| CHEMBL3191874 | — | IC50 | = | 183.1 | nM | 6.74 |
| CHEMBL1523841 | — | IC50 | = | 188.7 | nM | 6.72 |
| CHEMBL1452795 | — | IC50 | = | 223.24 | nM | 6.65 |
| CHEMBL1367034 | — | IC50 | = | 226.31 | nM | 6.64 |
| CHEMBL1475884 | — | IC50 | = | 243.8 | nM | 6.61 |
| CHEMBL3197177 | — | IC50 | = | 244.39 | nM | 6.61 |
| CHEMBL2359072 | — | IC50 | = | 295.93 | nM | 6.53 |
| CHEMBL3196518 | — | IC50 | = | 320.11 | nM | 6.50 |
| CHEMBL599924 | — | IC50 | = | 335.17 | nM | 6.47 |
| CHEMBL1987060 | — | IC50 | = | 353.29 | nM | 6.45 |
| CHEMBL1489294 | — | IC50 | = | 373.47 | nM | 6.43 |
| CHEMBL1584985 | — | IC50 | = | 389.23 | nM | 6.41 |
| CHEMBL600778 | — | IC50 | = | 386.27 | nM | 6.41 |
| CHEMBL1354927 | — | IC50 | = | 396.19 | nM | 6.40 |
| CHEMBL1384253 | — | IC50 | = | 421.07 | nM | 6.38 |
| CHEMBL2000517 | — | IC50 | = | 427.89 | nM | 6.37 |
| CHEMBL1572157 | — | IC50 | = | 425.37 | nM | 6.37 |
| CHEMBL411729 | CYTOCHALASIN B | IC50 | = | 423.96 | nM | 6.37 |
| CHEMBL3192995 | — | IC50 | = | 445.52 | nM | 6.35 |
| CHEMBL3193468 | — | IC50 | = | 481.59 | nM | 6.32 |
| CHEMBL89445 | TERPYRIDINE | IC50 | = | 483.18 | nM | 6.32 |
| CHEMBL1400375 | — | IC50 | = | 511.77 | nM | 6.29 |
| CHEMBL1486214 | — | IC50 | = | 513.97 | nM | 6.29 |
| CHEMBL1372082 | — | IC50 | = | 520.77 | nM | 6.28 |
| CHEMBL3197070 | — | IC50 | = | 540.27 | nM | 6.27 |