Assay Detail
Functional
CHEMBL1614484
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Luminescence Cell-Based Dose Confirmation to Identify Activators of 5'UTR Stem-Loop Driven Alpha-Synuclein mRNA Translation in H4 Neuroglioblastoma Cells. (Class of assay: confirmatory) [Related pubchem assays: 1829 (Project Summary), 1814 (Primary HTS)]
235
Total Activities
235
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 235 | 6.32 | 7.16 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1588285 | — | — | 1 | 7.16 |
| CHEMBL41384 | — | — | 1 | 6.98 |
| CHEMBL1363615 | — | — | 1 | 6.94 |
| CHEMBL3191871 | — | — | 1 | 6.92 |
| CHEMBL1427062 | — | — | 1 | 6.86 |
| CHEMBL1460534 | — | — | 1 | 6.85 |
| CHEMBL1328527 | — | — | 1 | 6.79 |
| CHEMBL1350043 | — | — | 1 | 6.76 |
| CHEMBL1575402 | — | — | 1 | 6.70 |
| CHEMBL1428673 | — | — | 1 | 6.70 |
| CHEMBL1462008 | — | — | 1 | 6.69 |
| CHEMBL1324123 | — | — | 1 | 6.68 |
| CHEMBL1311920 | — | — | 1 | 6.68 |
| CHEMBL1403922 | — | — | 1 | 6.67 |
| CHEMBL1479595 | — | — | 1 | 6.66 |
| CHEMBL1309378 | — | — | 1 | 6.66 |
| CHEMBL1565691 | — | — | 1 | 6.66 |
| CHEMBL1341119 | — | — | 1 | 6.64 |
| CHEMBL1499934 | — | — | 1 | 6.64 |
| CHEMBL1490429 | — | — | 1 | 6.64 |
| CHEMBL1977589 | — | — | 1 | 6.64 |
| CHEMBL1987798 | — | — | 1 | 6.64 |
| CHEMBL1323422 | — | — | 1 | 6.64 |
| CHEMBL1518032 | — | — | 1 | 6.63 |
| CHEMBL1501185 | — | — | 1 | 6.63 |
| CHEMBL1587805 | — | — | 1 | 6.63 |
| CHEMBL3211154 | — | — | 1 | 6.63 |
| CHEMBL1448605 | — | — | 1 | 6.62 |
| CHEMBL1495474 | — | — | 1 | 6.62 |
| CHEMBL1524533 | — | — | 1 | 6.62 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1588285 | — | EC50 | = | 69.0 | nM | 7.16 |
| CHEMBL41384 | — | EC50 | = | 104.0 | nM | 6.98 |
| CHEMBL1363615 | — | EC50 | = | 114.0 | nM | 6.94 |
| CHEMBL3191871 | — | EC50 | = | 121.0 | nM | 6.92 |
| CHEMBL1427062 | — | EC50 | = | 138.0 | nM | 6.86 |
| CHEMBL1460534 | — | EC50 | = | 141.0 | nM | 6.85 |
| CHEMBL1328527 | — | EC50 | = | 161.0 | nM | 6.79 |
| CHEMBL1350043 | — | EC50 | = | 174.0 | nM | 6.76 |
| CHEMBL1575402 | — | EC50 | = | 200.0 | nM | 6.70 |
| CHEMBL1428673 | — | EC50 | = | 198.0 | nM | 6.70 |
| CHEMBL1462008 | — | EC50 | = | 206.0 | nM | 6.69 |
| CHEMBL1324123 | — | EC50 | = | 210.0 | nM | 6.68 |
| CHEMBL1311920 | — | EC50 | = | 208.0 | nM | 6.68 |
| CHEMBL1403922 | — | EC50 | = | 216.0 | nM | 6.67 |
| CHEMBL1479595 | — | EC50 | = | 217.0 | nM | 6.66 |
| CHEMBL1309378 | — | EC50 | = | 219.0 | nM | 6.66 |
| CHEMBL1565691 | — | EC50 | = | 218.0 | nM | 6.66 |
| CHEMBL1323422 | — | EC50 | = | 230.0 | nM | 6.64 |
| CHEMBL1987798 | — | EC50 | = | 228.0 | nM | 6.64 |
| CHEMBL1977589 | — | EC50 | = | 227.0 | nM | 6.64 |
| CHEMBL1341119 | — | EC50 | = | 228.0 | nM | 6.64 |
| CHEMBL1490429 | — | EC50 | = | 231.0 | nM | 6.64 |
| CHEMBL1499934 | — | EC50 | = | 229.0 | nM | 6.64 |
| CHEMBL1518032 | — | EC50 | = | 232.0 | nM | 6.63 |
| CHEMBL1587805 | — | EC50 | = | 232.0 | nM | 6.63 |
| CHEMBL3211154 | — | EC50 | = | 236.0 | nM | 6.63 |
| CHEMBL1501185 | — | EC50 | = | 236.0 | nM | 6.63 |
| CHEMBL1588860 | — | EC50 | = | 240.0 | nM | 6.62 |
| CHEMBL1448605 | — | EC50 | = | 238.0 | nM | 6.62 |
| CHEMBL1495474 | — | EC50 | = | 240.0 | nM | 6.62 |
| CHEMBL1564261 | — | EC50 | = | 239.0 | nM | 6.62 |
| CHEMBL1524533 | — | EC50 | = | 237.0 | nM | 6.62 |
| CHEMBL1536507 | — | EC50 | = | 247.0 | nM | 6.61 |
| CHEMBL1501255 | — | EC50 | = | 247.0 | nM | 6.61 |
| CHEMBL1608267 | — | EC50 | = | 244.0 | nM | 6.61 |
| CHEMBL1477375 | — | EC50 | = | 244.0 | nM | 6.61 |
| CHEMBL1300939 | — | EC50 | = | 249.0 | nM | 6.60 |
| CHEMBL1595774 | — | EC50 | = | 251.0 | nM | 6.60 |
| CHEMBL1424373 | — | EC50 | = | 250.0 | nM | 6.60 |
| CHEMBL1584476 | — | EC50 | = | 251.0 | nM | 6.60 |
| CHEMBL1510913 | — | EC50 | = | 252.0 | nM | 6.60 |
| CHEMBL1323133 | — | EC50 | = | 256.0 | nM | 6.59 |
| CHEMBL3213101 | — | EC50 | = | 256.0 | nM | 6.59 |
| CHEMBL1543054 | — | EC50 | = | 261.0 | nM | 6.58 |
| CHEMBL1507676 | — | EC50 | = | 262.0 | nM | 6.58 |
| CHEMBL1441858 | — | EC50 | = | 272.0 | nM | 6.57 |
| CHEMBL1991055 | — | EC50 | = | 278.0 | nM | 6.56 |
| CHEMBL1533107 | — | EC50 | = | 277.0 | nM | 6.56 |
| CHEMBL1581941 | — | EC50 | = | 282.0 | nM | 6.55 |
| CHEMBL1471700 | — | EC50 | = | 280.0 | nM | 6.55 |