Assay Detail
Functional
CHEMBL1738080
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Dose Response confirmation of uHTS hits from a small molecule inhibitors of LYP via a fluorescence intensity assay using pCAP substrate. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID1779, AID1784, AID2135]
140
Total Activities
140
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Tyrosine-protein phosphatase non-receptor type 22 (CHEMBL2889) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 140 | 5.04 | 5.87 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL578512 | — | — | 1 | 5.87 |
| CHEMBL1325945 | — | — | 1 | 5.75 |
| CHEMBL570345 | — | — | 1 | 5.62 |
| CHEMBL1424694 | — | — | 1 | 5.61 |
| CHEMBL1443268 | — | — | 1 | 5.58 |
| CHEMBL1438889 | — | — | 1 | 5.43 |
| CHEMBL1320181 | — | — | 1 | 5.42 |
| CHEMBL1439815 | — | — | 1 | 5.34 |
| CHEMBL1492305 | — | — | 1 | 5.32 |
| CHEMBL1426096 | — | — | 1 | 5.24 |
| CHEMBL1533230 | — | — | 1 | 5.22 |
| CHEMBL1580263 | — | — | 1 | 5.21 |
| CHEMBL2000167 | — | — | 1 | 5.18 |
| CHEMBL1527520 | — | — | 1 | 5.17 |
| CHEMBL1371816 | — | — | 1 | 5.16 |
| CHEMBL1536896 | — | — | 1 | 5.14 |
| CHEMBL3190951 | — | — | 1 | 5.12 |
| CHEMBL1471865 | — | — | 1 | 5.07 |
| CHEMBL1488035 | — | — | 1 | 4.88 |
| CHEMBL599924 | — | — | 1 | 4.88 |
| CHEMBL1464805 | — | — | 1 | 4.80 |
| CHEMBL1981200 | — | — | 1 | 4.80 |
| CHEMBL1417070 | — | — | 1 | 4.71 |
| CHEMBL1529554 | — | — | 1 | 4.67 |
| CHEMBL1576746 | — | — | 1 | 4.50 |
| CHEMBL1976414 | — | — | 1 | 4.19 |
| CHEMBL1309430 | — | — | 1 | 4.16 |
| CHEMBL1429070 | — | — | 1 | 4.12 |
| CHEMBL1586851 | — | — | 1 | 4.12 |
| CHEMBL3208812 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL578512 | — | IC50 | = | 1350.0 | nM | 5.87 |
| CHEMBL1325945 | — | IC50 | = | 1784.0 | nM | 5.75 |
| CHEMBL570345 | — | IC50 | = | 2393.0 | nM | 5.62 |
| CHEMBL1424694 | — | IC50 | = | 2443.0 | nM | 5.61 |
| CHEMBL1443268 | — | IC50 | = | 2612.0 | nM | 5.58 |
| CHEMBL1438889 | — | IC50 | = | 3741.0 | nM | 5.43 |
| CHEMBL1320181 | — | IC50 | = | 3779.0 | nM | 5.42 |
| CHEMBL1439815 | — | IC50 | = | 4575.0 | nM | 5.34 |
| CHEMBL1492305 | — | IC50 | = | 4759.0 | nM | 5.32 |
| CHEMBL1426096 | — | IC50 | = | 5757.0 | nM | 5.24 |
| CHEMBL1533230 | — | IC50 | = | 5967.0 | nM | 5.22 |
| CHEMBL1580263 | — | IC50 | = | 6114.0 | nM | 5.21 |
| CHEMBL2000167 | — | IC50 | = | 6628.0 | nM | 5.18 |
| CHEMBL1527520 | — | IC50 | = | 6844.0 | nM | 5.17 |
| CHEMBL1371816 | — | IC50 | = | 6862.0 | nM | 5.16 |
| CHEMBL1536896 | — | IC50 | = | 7259.0 | nM | 5.14 |
| CHEMBL3190951 | — | IC50 | = | 7654.0 | nM | 5.12 |
| CHEMBL1471865 | — | IC50 | = | 8582.0 | nM | 5.07 |
| CHEMBL1488035 | — | IC50 | = | 13194.0 | nM | 4.88 |
| CHEMBL599924 | — | IC50 | = | 13021.0 | nM | 4.88 |
| CHEMBL1464805 | — | IC50 | = | 15958.0 | nM | 4.80 |
| CHEMBL1981200 | — | IC50 | = | 15696.0 | nM | 4.80 |
| CHEMBL1417070 | — | IC50 | = | 19619.0 | nM | 4.71 |
| CHEMBL1529554 | — | IC50 | = | 21589.0 | nM | 4.67 |
| CHEMBL1576746 | — | IC50 | = | 31981.0 | nM | 4.50 |
| CHEMBL1976414 | — | IC50 | = | 64741.0 | nM | 4.19 |
| CHEMBL1309430 | — | IC50 | = | 68933.0 | nM | 4.16 |
| CHEMBL1429070 | — | IC50 | = | 76324.0 | nM | 4.12 |
| CHEMBL1586851 | — | IC50 | = | 75261.0 | nM | 4.12 |
| CHEMBL1467425 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1549636 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1606761 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1535241 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1338178 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1360572 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1600686 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL3212510 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1499300 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1993612 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1335318 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1414751 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1493152 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1337760 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1301248 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1490435 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1371394 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1431216 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1344691 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1373137 | — | IC50 | > | 79400.0 | nM | - |
| CHEMBL1505659 | — | IC50 | > | 79400.0 | nM | - |