Assay Detail
Functional
CHEMBL1738089
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: SAR VHR1 Fluorescent Assay for In Vitro dose response studies. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID1654, AID1661, AID1878, AID1992, AID2004, AID2070, AID2085]
76
Total Activities
75
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Dual specificity protein phosphatase 3 (CHEMBL2635) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 76 | 5.24 | 7.19 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1460470 | — | — | 1 | 7.19 |
| CHEMBL1608642 | — | — | 2 | 6.44 |
| CHEMBL1445488 | — | — | 1 | 6.42 |
| CHEMBL1536896 | — | — | 1 | 6.32 |
| CHEMBL1501132 | — | — | 1 | 6.31 |
| CHEMBL1526088 | — | — | 1 | 6.06 |
| CHEMBL1407368 | — | — | 1 | 5.93 |
| CHEMBL1603381 | — | — | 1 | 5.91 |
| CHEMBL1371869 | — | — | 1 | 5.90 |
| CHEMBL1424189 | — | — | 1 | 5.50 |
| CHEMBL1393151 | — | — | 1 | 5.44 |
| CHEMBL1702303 | — | — | 1 | 5.32 |
| CHEMBL1608654 | — | — | 1 | 5.24 |
| CHEMBL1489230 | — | — | 1 | 5.24 |
| CHEMBL1722185 | — | — | 1 | 5.18 |
| CHEMBL1449836 | — | — | 1 | 5.15 |
| CHEMBL1530080 | — | — | 1 | 5.13 |
| CHEMBL1609429 | — | — | 1 | 5.11 |
| CHEMBL1452974 | — | — | 1 | 5.05 |
| CHEMBL1526669 | — | — | 1 | 4.92 |
| CHEMBL1414679 | — | — | 1 | 4.91 |
| CHEMBL1372387 | — | — | 1 | 4.87 |
| CHEMBL1709810 | — | — | 1 | 4.87 |
| CHEMBL1705741 | — | — | 1 | 4.85 |
| CHEMBL1304974 | — | — | 1 | 4.84 |
| CHEMBL1730460 | — | — | 1 | 4.83 |
| CHEMBL1724547 | — | — | 1 | 4.82 |
| CHEMBL1727475 | — | — | 1 | 4.74 |
| CHEMBL1371777 | — | — | 1 | 4.71 |
| CHEMBL1484942 | — | — | 1 | 4.65 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1460470 | — | IC50 | = | 65.0 | nM | 7.19 |
| CHEMBL1608642 | — | IC50 | = | 366.0 | nM | 6.44 |
| CHEMBL1445488 | — | IC50 | = | 382.0 | nM | 6.42 |
| CHEMBL1536896 | — | IC50 | = | 480.0 | nM | 6.32 |
| CHEMBL1501132 | — | IC50 | = | 492.0 | nM | 6.31 |
| CHEMBL1526088 | — | IC50 | = | 878.0 | nM | 6.06 |
| CHEMBL1407368 | — | IC50 | = | 1180.0 | nM | 5.93 |
| CHEMBL1603381 | — | IC50 | = | 1230.0 | nM | 5.91 |
| CHEMBL1371869 | — | IC50 | = | 1250.0 | nM | 5.90 |
| CHEMBL1424189 | — | IC50 | = | 3200.0 | nM | 5.50 |
| CHEMBL1393151 | — | IC50 | = | 3630.0 | nM | 5.44 |
| CHEMBL1702303 | — | IC50 | = | 4840.0 | nM | 5.32 |
| CHEMBL1608654 | — | IC50 | = | 5820.0 | nM | 5.24 |
| CHEMBL1489230 | — | IC50 | = | 5710.0 | nM | 5.24 |
| CHEMBL1722185 | — | IC50 | = | 6610.0 | nM | 5.18 |
| CHEMBL1449836 | — | IC50 | = | 7060.0 | nM | 5.15 |
| CHEMBL1530080 | — | IC50 | = | 7490.0 | nM | 5.13 |
| CHEMBL1609429 | — | IC50 | = | 7700.0 | nM | 5.11 |
| CHEMBL1452974 | — | IC50 | = | 8810.0 | nM | 5.05 |
| CHEMBL1526669 | — | IC50 | = | 12100.0 | nM | 4.92 |
| CHEMBL1414679 | — | IC50 | = | 12300.0 | nM | 4.91 |
| CHEMBL1709810 | — | IC50 | = | 13400.0 | nM | 4.87 |
| CHEMBL1372387 | — | IC50 | = | 13500.0 | nM | 4.87 |
| CHEMBL1705741 | — | IC50 | = | 14000.0 | nM | 4.85 |
| CHEMBL1304974 | — | IC50 | = | 14600.0 | nM | 4.84 |
| CHEMBL1730460 | — | IC50 | = | 14700.0 | nM | 4.83 |
| CHEMBL1724547 | — | IC50 | = | 15100.0 | nM | 4.82 |
| CHEMBL1727475 | — | IC50 | = | 18300.0 | nM | 4.74 |
| CHEMBL1371777 | — | IC50 | = | 19700.0 | nM | 4.71 |
| CHEMBL1484942 | — | IC50 | = | 22500.0 | nM | 4.65 |
| CHEMBL1714877 | — | IC50 | = | 26400.0 | nM | 4.58 |
| CHEMBL1451516 | — | IC50 | = | 27900.0 | nM | 4.55 |
| CHEMBL1449334 | — | IC50 | = | 29500.0 | nM | 4.53 |
| CHEMBL1441524 | — | IC50 | = | 30400.0 | nM | 4.52 |
| CHEMBL1483335 | — | IC50 | = | 33500.0 | nM | 4.47 |
| CHEMBL1489619 | — | IC50 | = | 86300.0 | nM | 4.06 |
| CHEMBL1715760 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1725341 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1608642 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1734920 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1715328 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1736022 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1735040 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1578067 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1536551 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1733670 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1727280 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1530046 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1607593 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1385949 | — | IC50 | > | 99000.0 | nM | - |