Assay Detail
Functional
CHEMBL1794570
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Counterscreen for IDE activators: Fluorescence polarization-based biochemical high throughput dose response assay to identify fluorescent artifacts and/or optically active compounds. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID493087, AID493124, AID588681]
231
Total Activities
231
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HEK293 |
| Category | confirmatory |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 231 | 5.17 | 7.35 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1553368 | — | — | 1 | 7.35 |
| CHEMBL354349 | EUFLAVINE | -1.0 | 1 | 6.24 |
| CHEMBL1568474 | — | — | 1 | 6.18 |
| CHEMBL1705738 | — | — | 1 | 5.96 |
| CHEMBL1332522 | — | — | 1 | 5.81 |
| CHEMBL857 | BIOTIN | 4.0 | 1 | 5.69 |
| CHEMBL1486690 | PYRONIN Y | — | 1 | 5.68 |
| CHEMBL1312403 | — | — | 1 | 5.61 |
| CHEMBL1378294 | — | — | 1 | 5.34 |
| CHEMBL1412077 | — | — | 1 | 5.31 |
| CHEMBL1409608 | — | — | 1 | 5.27 |
| CHEMBL1578670 | — | — | 1 | 5.26 |
| CHEMBL1387366 | — | — | 1 | 5.18 |
| CHEMBL1522563 | — | — | 1 | 5.16 |
| CHEMBL1574420 | — | — | 1 | 5.16 |
| CHEMBL1232381 | — | — | 1 | 4.92 |
| CHEMBL1472131 | — | — | 1 | 4.92 |
| CHEMBL3193419 | — | — | 1 | 4.91 |
| CHEMBL1725771 | — | — | 1 | 4.88 |
| CHEMBL1510317 | — | — | 1 | 4.77 |
| CHEMBL1527972 | — | — | 1 | 4.69 |
| CHEMBL1732485 | — | — | 1 | 4.67 |
| CHEMBL1403262 | — | — | 1 | 4.65 |
| CHEMBL1591898 | — | — | 1 | 4.62 |
| CHEMBL1458111 | — | — | 1 | 4.51 |
| CHEMBL1575701 | — | — | 1 | 4.49 |
| CHEMBL1442125 | — | — | 1 | 4.30 |
| CHEMBL1370456 | — | — | 1 | 4.27 |
| CHEMBL1393633 | — | — | 1 | 4.23 |
| CHEMBL1418754 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1553368 | — | EC50 | = | 45.0 | nM | 7.35 |
| CHEMBL354349 | EUFLAVINE | EC50 | = | 575.83 | nM | 6.24 |
| CHEMBL1568474 | — | EC50 | = | 658.59 | nM | 6.18 |
| CHEMBL1705738 | — | EC50 | = | 1089.0 | nM | 5.96 |
| CHEMBL1332522 | — | EC50 | = | 1554.0 | nM | 5.81 |
| CHEMBL857 | BIOTIN | EC50 | = | 2057.0 | nM | 5.69 |
| CHEMBL1486690 | PYRONIN Y | EC50 | = | 2085.0 | nM | 5.68 |
| CHEMBL1312403 | — | EC50 | = | 2444.0 | nM | 5.61 |
| CHEMBL1378294 | — | EC50 | = | 4602.0 | nM | 5.34 |
| CHEMBL1412077 | — | EC50 | = | 4946.0 | nM | 5.31 |
| CHEMBL1409608 | — | EC50 | = | 5377.0 | nM | 5.27 |
| CHEMBL1578670 | — | EC50 | = | 5525.0 | nM | 5.26 |
| CHEMBL1387366 | — | EC50 | = | 6566.0 | nM | 5.18 |
| CHEMBL1574420 | — | EC50 | = | 6885.0 | nM | 5.16 |
| CHEMBL1522563 | — | EC50 | = | 6890.0 | nM | 5.16 |
| CHEMBL1472131 | — | EC50 | = | 12111.0 | nM | 4.92 |
| CHEMBL1232381 | — | EC50 | = | 11887.0 | nM | 4.92 |
| CHEMBL3193419 | — | EC50 | = | 12393.0 | nM | 4.91 |
| CHEMBL1725771 | — | EC50 | = | 13193.0 | nM | 4.88 |
| CHEMBL1510317 | — | EC50 | = | 17046.0 | nM | 4.77 |
| CHEMBL1527972 | — | EC50 | = | 20412.0 | nM | 4.69 |
| CHEMBL1732485 | — | EC50 | = | 21215.0 | nM | 4.67 |
| CHEMBL1403262 | — | EC50 | = | 22554.0 | nM | 4.65 |
| CHEMBL1591898 | — | EC50 | = | 24011.0 | nM | 4.62 |
| CHEMBL1458111 | — | EC50 | = | 30871.0 | nM | 4.51 |
| CHEMBL1575701 | — | EC50 | = | 32143.0 | nM | 4.49 |
| CHEMBL1442125 | — | EC50 | = | 50253.0 | nM | 4.30 |
| CHEMBL1370456 | — | EC50 | = | 53645.0 | nM | 4.27 |
| CHEMBL1393633 | — | EC50 | = | 58665.0 | nM | 4.23 |
| CHEMBL250711 | OLEOYL DOPAMINE | EC50 | > | 54705.0 | nM | - |
| CHEMBL3391764 | — | EC50 | > | 54676.0 | nM | - |
| CHEMBL1578991 | — | EC50 | > | 54748.0 | nM | - |
| CHEMBL1979800 | — | EC50 | > | 54699.0 | nM | - |
| CHEMBL589245 | — | EC50 | > | 55935.0 | nM | - |
| CHEMBL1586096 | — | EC50 | > | 55941.0 | nM | - |
| CHEMBL3189224 | — | EC50 | > | 55958.0 | nM | - |
| CHEMBL1602206 | — | EC50 | > | 54710.0 | nM | - |
| CHEMBL532160 | — | EC50 | > | 54699.0 | nM | - |
| CHEMBL1390912 | — | EC50 | > | 55933.0 | nM | - |
| CHEMBL1491750 | — | EC50 | > | 54699.0 | nM | - |
| CHEMBL1558968 | — | EC50 | > | 54705.0 | nM | - |
| CHEMBL1547938 | — | EC50 | > | 54732.0 | nM | - |
| CHEMBL1982108 | — | EC50 | > | 54705.0 | nM | - |
| CHEMBL1731264 | — | EC50 | > | 55986.0 | nM | - |
| CHEMBL1462480 | — | EC50 | > | 54699.0 | nM | - |
| CHEMBL1452296 | — | EC50 | > | 55935.0 | nM | - |
| CHEMBL1485551 | — | EC50 | > | 55947.0 | nM | - |
| CHEMBL1587031 | — | EC50 | > | 55963.0 | nM | - |
| CHEMBL1986183 | — | EC50 | > | 54688.0 | nM | - |
| CHEMBL1511114 | — | EC50 | > | 54686.0 | nM | - |