Assay Detail
Functional
CHEMBL1963832
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: NTRK2
937
Total Activities
920
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | other |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 937 | 6.31 | 9.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1980995 | — | — | 1 | 9.10 |
| CHEMBL2007421 | — | — | 1 | 9.00 |
| CHEMBL1983268 | ENTRECTINIB | 4.0 | 1 | 8.60 |
| CHEMBL411903 | — | — | 1 | 8.40 |
| CHEMBL1972220 | — | — | 1 | 8.40 |
| CHEMBL1980407 | — | — | 1 | 8.30 |
| CHEMBL1971947 | — | — | 1 | 8.30 |
| CHEMBL1982476 | — | — | 1 | 8.20 |
| CHEMBL260092 | — | — | 1 | 8.20 |
| CHEMBL2005631 | — | — | 1 | 8.20 |
| CHEMBL1980297 | ILORASERTIB | 2.0 | 1 | 8.00 |
| CHEMBL1970083 | — | — | 1 | 8.00 |
| CHEMBL1997892 | — | — | 1 | 8.00 |
| CHEMBL2004716 | — | — | 1 | 8.00 |
| CHEMBL1970142 | — | — | 1 | 8.00 |
| CHEMBL1965170 | — | — | 1 | 8.00 |
| CHEMBL1998585 | — | — | 1 | 7.90 |
| CHEMBL1967116 | — | — | 1 | 7.90 |
| CHEMBL1977134 | — | — | 1 | 7.90 |
| CHEMBL2005886 | — | — | 1 | 7.80 |
| CHEMBL482767 | SNS-314 | 1.0 | 1 | 7.80 |
| CHEMBL1988387 | — | — | 1 | 7.70 |
| CHEMBL1993661 | — | — | 1 | 7.70 |
| CHEMBL1977148 | — | — | 1 | 7.60 |
| CHEMBL1964692 | — | — | 1 | 7.60 |
| CHEMBL1988717 | — | — | 1 | 7.60 |
| CHEMBL1969102 | — | — | 1 | 7.60 |
| CHEMBL1982466 | — | — | 1 | 7.60 |
| CHEMBL1994321 | — | — | 1 | 7.50 |
| CHEMBL1983111 | — | — | 1 | 7.50 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1980995 | — | Ki | = | 0.7943 | nM | 9.10 |
| CHEMBL2007421 | — | Ki | = | 1.0 | nM | 9.00 |
| CHEMBL1983268 | ENTRECTINIB | Ki | = | 2.512 | nM | 8.60 |
| CHEMBL411903 | — | Ki | = | 3.981 | nM | 8.40 |
| CHEMBL1972220 | — | Ki | = | 3.981 | nM | 8.40 |
| CHEMBL1980407 | — | Ki | = | 5.012 | nM | 8.30 |
| CHEMBL1971947 | — | Ki | = | 5.012 | nM | 8.30 |
| CHEMBL1982476 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL2005631 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL260092 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL1970142 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL1997892 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL1965170 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL1970083 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL2004716 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL1980297 | ILORASERTIB | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL1967116 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL1998585 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL1977134 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL482767 | SNS-314 | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL2005886 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1988387 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1993661 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1982466 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1969102 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1964692 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1988717 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1977148 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1994321 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL1983111 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL1084546 | PF-00562271 | Ki | = | 39.81 | nM | 7.40 |
| CHEMBL1989708 | — | Ki | = | 39.81 | nM | 7.40 |
| CHEMBL2006765 | — | Ki | = | 39.81 | nM | 7.40 |
| CHEMBL1997623 | — | Ki | = | 39.81 | nM | 7.40 |
| CHEMBL1999414 | — | Ki | = | 50.12 | nM | 7.30 |
| CHEMBL1983640 | — | Ki | = | 50.12 | nM | 7.30 |
| CHEMBL1968406 | — | Ki | = | 50.12 | nM | 7.30 |
| CHEMBL1970317 | — | Ki | = | 50.12 | nM | 7.30 |
| CHEMBL196363 | — | Ki | = | 63.1 | nM | 7.20 |
| CHEMBL1996646 | — | Ki | = | 63.1 | nM | 7.20 |
| CHEMBL2004290 | — | Ki | = | 63.1 | nM | 7.20 |
| CHEMBL1965988 | — | Ki | = | 79.43 | nM | 7.10 |
| CHEMBL1973540 | — | Ki | = | 79.43 | nM | 7.10 |
| CHEMBL2001485 | — | Ki | = | 79.43 | nM | 7.10 |
| CHEMBL1980391 | RG-1530 | Ki | = | 100.0 | nM | 7.00 |
| CHEMBL2005478 | — | Ki | = | 100.0 | nM | 7.00 |
| CHEMBL2004311 | — | Ki | = | 100.0 | nM | 7.00 |
| CHEMBL2002165 | — | Ki | = | 100.0 | nM | 7.00 |
| CHEMBL1984162 | — | Ki | = | 100.0 | nM | 7.00 |
| CHEMBL1964441 | — | Ki | = | 100.0 | nM | 7.00 |