Assay Detail
Functional
CHEMBL1964023
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Counterscreen for inhibitors of the Steroid Receptor Coactivator 1 (SRC1; NCOA1): Luminescence-based cell-based high throughput dose response assay to identify inhibitors of the Herpes Virus Virion Protein 16 (VP16). (Class of assay: confirmatory)
240
Total Activities
240
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
Tegument protein VP16 (CHEMBL4218) ↗| Type | SINGLE PROTEIN |
| Organism | Herpes simplex virus (type 1 / strain 17) |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 240 | 4.91 | 5.50 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1399772 | — | — | 1 | 5.50 |
| CHEMBL1413178 | — | — | 1 | 5.46 |
| CHEMBL1383315 | — | — | 1 | 5.40 |
| CHEMBL1893675 | — | — | 1 | 5.39 |
| CHEMBL1965376 | — | — | 1 | 5.33 |
| CHEMBL1373969 | — | — | 1 | 5.33 |
| CHEMBL479368 | — | — | 1 | 5.32 |
| CHEMBL1985479 | — | — | 1 | 5.31 |
| CHEMBL2005690 | — | — | 1 | 5.31 |
| CHEMBL2007313 | — | — | 1 | 5.30 |
| CHEMBL1387923 | — | — | 1 | 5.29 |
| CHEMBL1996281 | — | — | 1 | 5.28 |
| CHEMBL485636 | — | — | 1 | 5.27 |
| CHEMBL1469670 | — | — | 1 | 5.27 |
| CHEMBL1461035 | — | — | 1 | 5.26 |
| CHEMBL1585209 | — | — | 1 | 5.25 |
| CHEMBL1318140 | — | — | 1 | 5.24 |
| CHEMBL356169 | — | — | 1 | 5.23 |
| CHEMBL1329069 | — | — | 1 | 5.22 |
| CHEMBL494325 | — | — | 1 | 5.22 |
| CHEMBL1440409 | — | — | 1 | 5.20 |
| CHEMBL1736199 | — | — | 1 | 5.19 |
| CHEMBL1398705 | — | — | 1 | 5.18 |
| CHEMBL1307972 | — | — | 1 | 5.17 |
| CHEMBL1735689 | — | — | 1 | 5.17 |
| CHEMBL1412433 | — | — | 1 | 5.16 |
| CHEMBL1974053 | — | — | 1 | 5.16 |
| CHEMBL1544409 | — | — | 1 | 5.16 |
| CHEMBL2004809 | — | — | 1 | 5.12 |
| CHEMBL1564670 | — | — | 1 | 5.11 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1399772 | — | IC50 | = | 3197.0 | nM | 5.50 |
| CHEMBL1413178 | — | IC50 | = | 3503.0 | nM | 5.46 |
| CHEMBL1383315 | — | IC50 | = | 3976.0 | nM | 5.40 |
| CHEMBL1893675 | — | IC50 | = | 4102.0 | nM | 5.39 |
| CHEMBL1965376 | — | IC50 | = | 4648.0 | nM | 5.33 |
| CHEMBL1373969 | — | IC50 | = | 4713.0 | nM | 5.33 |
| CHEMBL479368 | — | IC50 | = | 4771.0 | nM | 5.32 |
| CHEMBL2005690 | — | IC50 | = | 4874.0 | nM | 5.31 |
| CHEMBL1985479 | — | IC50 | = | 4899.0 | nM | 5.31 |
| CHEMBL2007313 | — | IC50 | = | 5004.0 | nM | 5.30 |
| CHEMBL1387923 | — | IC50 | = | 5144.0 | nM | 5.29 |
| CHEMBL1996281 | — | IC50 | = | 5286.0 | nM | 5.28 |
| CHEMBL485636 | — | IC50 | = | 5390.0 | nM | 5.27 |
| CHEMBL1469670 | — | IC50 | = | 5373.0 | nM | 5.27 |
| CHEMBL1461035 | — | IC50 | = | 5545.0 | nM | 5.26 |
| CHEMBL1585209 | — | IC50 | = | 5596.0 | nM | 5.25 |
| CHEMBL1318140 | — | IC50 | = | 5786.0 | nM | 5.24 |
| CHEMBL356169 | — | IC50 | = | 5946.0 | nM | 5.23 |
| CHEMBL494325 | — | IC50 | = | 5958.0 | nM | 5.22 |
| CHEMBL1329069 | — | IC50 | = | 5961.0 | nM | 5.22 |
| CHEMBL1440409 | — | IC50 | = | 6341.0 | nM | 5.20 |
| CHEMBL1736199 | — | IC50 | = | 6476.0 | nM | 5.19 |
| CHEMBL1398705 | — | IC50 | = | 6663.0 | nM | 5.18 |
| CHEMBL1735689 | — | IC50 | = | 6824.0 | nM | 5.17 |
| CHEMBL1307972 | — | IC50 | = | 6687.0 | nM | 5.17 |
| CHEMBL1544409 | — | IC50 | = | 6956.0 | nM | 5.16 |
| CHEMBL1412433 | — | IC50 | = | 6968.0 | nM | 5.16 |
| CHEMBL1974053 | — | IC50 | = | 6893.0 | nM | 5.16 |
| CHEMBL2004809 | — | IC50 | = | 7516.0 | nM | 5.12 |
| CHEMBL1421781 | — | IC50 | = | 7857.0 | nM | 5.11 |
| CHEMBL1471916 | — | IC50 | = | 7851.0 | nM | 5.11 |
| CHEMBL1564670 | — | IC50 | = | 7748.0 | nM | 5.11 |
| CHEMBL1444434 | — | IC50 | = | 7945.0 | nM | 5.10 |
| CHEMBL1600535 | — | IC50 | = | 7866.0 | nM | 5.10 |
| CHEMBL1882211 | — | IC50 | = | 7887.0 | nM | 5.10 |
| CHEMBL1896348 | — | IC50 | = | 7873.0 | nM | 5.10 |
| CHEMBL2373711 | — | IC50 | = | 8052.0 | nM | 5.09 |
| CHEMBL1996902 | — | IC50 | = | 8117.0 | nM | 5.09 |
| CHEMBL1572233 | — | IC50 | = | 8064.0 | nM | 5.09 |
| CHEMBL1412284 | — | IC50 | = | 8326.0 | nM | 5.08 |
| CHEMBL1605666 | — | IC50 | = | 8403.0 | nM | 5.08 |
| CHEMBL1323722 | — | IC50 | = | 8239.0 | nM | 5.08 |
| CHEMBL1528507 | — | IC50 | = | 8403.0 | nM | 5.08 |
| CHEMBL1494091 | — | IC50 | = | 8313.0 | nM | 5.08 |
| CHEMBL1983418 | — | IC50 | = | 8610.0 | nM | 5.07 |
| CHEMBL1516127 | — | IC50 | = | 8588.0 | nM | 5.07 |
| CHEMBL1975006 | — | IC50 | = | 8437.0 | nM | 5.07 |
| CHEMBL1385327 | — | IC50 | = | 8466.0 | nM | 5.07 |
| CHEMBL1380143 | — | IC50 | = | 8465.0 | nM | 5.07 |
| CHEMBL1331226 | — | IC50 | = | 8731.0 | nM | 5.06 |