Assay Detail
Functional
CHEMBL1964068
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PubChem BioAssay. Dose response for HTS for Beta-2AR agonists via FAP method from Powderset3. (Class of assay: confirmatory)
22
Total Activities
22
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 22 | 7.09 | 8.81 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1419122 | — | — | 1 | 8.81 |
| CHEMBL1373386 | — | — | 1 | 8.26 |
| CHEMBL1478198 | — | — | 1 | 8.19 |
| CHEMBL1346316 | — | — | 1 | 8.16 |
| CHEMBL1570111 | — | — | 1 | 8.13 |
| CHEMBL1452334 | — | — | 1 | 8.01 |
| CHEMBL1472233 | — | — | 1 | 7.84 |
| CHEMBL1541608 | — | — | 1 | 7.84 |
| CHEMBL1457704 | — | — | 1 | 7.62 |
| CHEMBL1318405 | — | — | 1 | 7.44 |
| CHEMBL1327806 | — | — | 1 | 7.26 |
| CHEMBL1375364 | — | — | 1 | 7.21 |
| CHEMBL1376574 | — | — | 1 | 7.05 |
| CHEMBL531401 | — | — | 1 | 6.69 |
| CHEMBL1723653 | — | — | 1 | 6.14 |
| CHEMBL1325250 | — | — | 1 | 5.94 |
| CHEMBL1505690 | — | — | 1 | 5.82 |
| CHEMBL1570251 | — | — | 1 | 5.82 |
| CHEMBL1387056 | — | — | 1 | 5.77 |
| CHEMBL1326167 | — | — | 1 | 5.74 |
| CHEMBL1483555 | — | — | 1 | 5.09 |
| CHEMBL1728558 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1419122 | — | EC50 | = | 1.53 | nM | 8.81 |
| CHEMBL1373386 | — | EC50 | = | 5.48 | nM | 8.26 |
| CHEMBL1478198 | — | EC50 | = | 6.43 | nM | 8.19 |
| CHEMBL1346316 | — | EC50 | = | 6.9 | nM | 8.16 |
| CHEMBL1570111 | — | EC50 | = | 7.4 | nM | 8.13 |
| CHEMBL1452334 | — | EC50 | = | 9.77 | nM | 8.01 |
| CHEMBL1472233 | — | EC50 | = | 14.3 | nM | 7.84 |
| CHEMBL1541608 | — | EC50 | = | 14.3 | nM | 7.84 |
| CHEMBL1457704 | — | EC50 | = | 23.8 | nM | 7.62 |
| CHEMBL1318405 | — | EC50 | = | 36.6 | nM | 7.44 |
| CHEMBL1327806 | — | EC50 | = | 55.5 | nM | 7.26 |
| CHEMBL1375364 | — | EC50 | = | 60.9 | nM | 7.21 |
| CHEMBL1376574 | — | EC50 | = | 88.3 | nM | 7.05 |
| CHEMBL531401 | — | EC50 | = | 204.0 | nM | 6.69 |
| CHEMBL1723653 | — | EC50 | = | 731.0 | nM | 6.14 |
| CHEMBL1325250 | — | EC50 | = | 1140.0 | nM | 5.94 |
| CHEMBL1505690 | — | EC50 | = | 1510.0 | nM | 5.82 |
| CHEMBL1570251 | — | EC50 | = | 1510.0 | nM | 5.82 |
| CHEMBL1387056 | — | EC50 | = | 1710.0 | nM | 5.77 |
| CHEMBL1326167 | — | EC50 | = | 1810.0 | nM | 5.74 |
| CHEMBL1483555 | — | EC50 | = | 8090.0 | nM | 5.09 |
| CHEMBL1728558 | — | EC50 | = | 607500.0 | nM | - |