Assay Detail
Functional
CHEMBL3368953
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiviral activity against Reovirus type-1 infected in BHK21 cells assessed as inhibition of virus-induced cytopathogenicity after 3 to 4 days by MTT assay
86
Total Activities
86
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Reovirus sp. |
| Cell Type | BHK-21 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Antiviral activity of benzimidazole derivatives. III. Novel anti-CVB-5, anti-RSV and anti-Sb-1 agents.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 86 | 4.90 | 5.62 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL418899 | 2'-B-METHYL-GUANOSINE | — | 1 | 5.62 |
| CHEMBL3325678 | — | — | 1 | 4.57 |
| CHEMBL3325677 | — | — | 1 | 4.50 |
| CHEMBL573352 | TAS-106 | 2.0 | 1 | - |
| CHEMBL1643 | RIBAVIRIN | 4.0 | 1 | - |
| CHEMBL564201 | 6-AZAURIDINE | — | 1 | - |
| CHEMBL866 | MYCOPHENOLIC ACID | 4.0 | 1 | - |
| CHEMBL184 | ACYCLOVIR | 4.0 | 1 | - |
| CHEMBL3325956 | — | — | 1 | - |
| CHEMBL3325835 | — | — | 1 | - |
| CHEMBL3325836 | — | — | 1 | - |
| CHEMBL3325837 | — | — | 1 | - |
| CHEMBL3325838 | — | — | 1 | - |
| CHEMBL3325839 | — | — | 1 | - |
| CHEMBL3325840 | — | — | 1 | - |
| CHEMBL3325935 | — | — | 1 | - |
| CHEMBL3325936 | — | — | 1 | - |
| CHEMBL3325937 | — | — | 1 | - |
| CHEMBL3325938 | — | — | 1 | - |
| CHEMBL3325950 | — | — | 1 | - |
| CHEMBL3325940 | — | — | 1 | - |
| CHEMBL3325941 | — | — | 1 | - |
| CHEMBL3325942 | — | — | 1 | - |
| CHEMBL3325943 | — | — | 1 | - |
| CHEMBL3325944 | — | — | 1 | - |
| CHEMBL3325945 | — | — | 1 | - |
| CHEMBL3325946 | — | — | 1 | - |
| CHEMBL3325947 | — | — | 1 | - |
| CHEMBL3325948 | — | — | 1 | - |
| CHEMBL3325939 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL418899 | 2'-B-METHYL-GUANOSINE | EC50 | = | 2400.0 | nM | 5.62 |
| CHEMBL3325678 | — | EC50 | = | 27000.0 | nM | 4.57 |
| CHEMBL3325677 | — | EC50 | = | 32000.0 | nM | 4.50 |
| CHEMBL564201 | 6-AZAURIDINE | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325682 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL1643 | RIBAVIRIN | EC50 | > | 100000.0 | nM | - |
| CHEMBL573352 | TAS-106 | EC50 | > | 100000.0 | nM | - |
| CHEMBL1969873 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL1996660 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL2005128 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL2009615 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325949 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325955 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL1989039 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325954 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325953 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325952 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL351569 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL1995839 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325951 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325833 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325674 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325685 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325684 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325683 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL1922082 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325938 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325939 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325948 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325947 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325946 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325945 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325944 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325943 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325942 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325941 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325940 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325950 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL866 | MYCOPHENOLIC ACID | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325937 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325936 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325935 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325840 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325839 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325838 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325837 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325836 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325835 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3325956 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL184 | ACYCLOVIR | EC50 | > | 100000.0 | nM | - |