Assay Detail
Functional
CHEMBL3561978
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PubChem BioAssay. nuclear beta catenin stimulation in WNT3A conditioned C2C12 cells-IC50. (Class of assay: confirmatory)
98
Total Activities
97
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Cell Type | C2C12 |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 98 | 6.45 | 8.48 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2358886 | — | — | 1 | 8.48 |
| CHEMBL378544 | VINBLASTINE SULFATE | 4.0 | 2 | 8.46 |
| CHEMBL90555 | VINCRISTINE | 4.0 | 1 | 8.40 |
| CHEMBL538943 | VINORELBINE TARTRATE | 4.0 | 1 | 8.05 |
| CHEMBL140144 | — | — | 1 | 7.90 |
| CHEMBL61 | PODOFILOX | 4.0 | 1 | 7.88 |
| CHEMBL3182961 | — | — | 1 | 7.87 |
| CHEMBL3559830 | — | — | 1 | 7.74 |
| CHEMBL107 | COLCHICINE | 4.0 | 1 | 7.73 |
| CHEMBL34259 | METHOTREXATE | 4.0 | 1 | 7.58 |
| CHEMBL451887 | CARFILZOMIB | 4.0 | 1 | 7.54 |
| CHEMBL1417019 | MITOXANTRONE HYDROCHLORIDE | 4.0 | 1 | 7.52 |
| CHEMBL528271 | PARBENDAZOLE | 2.0 | 1 | 7.47 |
| CHEMBL1554 | DACTINOMYCIN | 4.0 | 1 | 7.43 |
| CHEMBL264373 | METOPRINE | -1.0 | 1 | 7.30 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 7.19 |
| CHEMBL1200976 | IDARUBICIN HYDROCHLORIDE | 4.0 | 1 | 7.00 |
| CHEMBL5416410 | DASATINIB | 4.0 | 1 | 6.98 |
| CHEMBL1607 | TOPOTECAN HYDROCHLORIDE | 4.0 | 1 | 6.87 |
| CHEMBL2105698 | ALVOCIDIB HYDROCHLORIDE | 2.0 | 1 | 6.72 |
| CHEMBL9514 | NOCODAZOLE | 2.0 | 1 | 6.63 |
| CHEMBL3184300 | — | — | 1 | 6.51 |
| CHEMBL1788401 | CYCLOBENDAZOLE | 2.0 | 1 | 6.46 |
| CHEMBL1087630 | OXIBENDAZOLE | 2.0 | 1 | 6.44 |
| CHEMBL1569226 | — | — | 1 | 6.43 |
| CHEMBL178 | DAUNORUBICIN | 4.0 | 1 | 6.43 |
| CHEMBL42442 | OXFENDAZOLE | 2.0 | 1 | 6.33 |
| CHEMBL1473700 | PIROCTONE | 2.0 | 1 | 6.23 |
| CHEMBL2356692 | — | — | 1 | 6.15 |
| CHEMBL922 | ADEFOVIR DIPIVOXIL | 4.0 | 1 | 6.15 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2358886 | — | IC50 | = | 3.3 | nM | 8.48 |
| CHEMBL378544 | VINBLASTINE SULFATE | IC50 | = | 3.5 | nM | 8.46 |
| CHEMBL90555 | VINCRISTINE | IC50 | = | 4.0 | nM | 8.40 |
| CHEMBL378544 | VINBLASTINE SULFATE | IC50 | = | 5.8 | nM | 8.24 |
| CHEMBL538943 | VINORELBINE TARTRATE | IC50 | = | 8.9 | nM | 8.05 |
| CHEMBL140144 | — | IC50 | = | 12.7 | nM | 7.90 |
| CHEMBL61 | PODOFILOX | IC50 | = | 13.1 | nM | 7.88 |
| CHEMBL3182961 | — | IC50 | = | 13.5 | nM | 7.87 |
| CHEMBL3559830 | — | IC50 | = | 18.3 | nM | 7.74 |
| CHEMBL107 | COLCHICINE | IC50 | = | 18.5 | nM | 7.73 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 26.5 | nM | 7.58 |
| CHEMBL451887 | CARFILZOMIB | IC50 | = | 29.2 | nM | 7.54 |
| CHEMBL1417019 | MITOXANTRONE HYDROCHLORIDE | IC50 | = | 30.3 | nM | 7.52 |
| CHEMBL528271 | PARBENDAZOLE | IC50 | = | 33.6 | nM | 7.47 |
| CHEMBL1554 | DACTINOMYCIN | IC50 | = | 37.0 | nM | 7.43 |
| CHEMBL264373 | METOPRINE | IC50 | = | 50.4 | nM | 7.30 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 65.2 | nM | 7.19 |
| CHEMBL1200976 | IDARUBICIN HYDROCHLORIDE | IC50 | = | 100.1 | nM | 7.00 |
| CHEMBL5416410 | DASATINIB | IC50 | = | 104.4 | nM | 6.98 |
| CHEMBL1607 | TOPOTECAN HYDROCHLORIDE | IC50 | = | 133.7 | nM | 6.87 |
| CHEMBL2105698 | ALVOCIDIB HYDROCHLORIDE | IC50 | = | 190.5 | nM | 6.72 |
| CHEMBL9514 | NOCODAZOLE | IC50 | = | 235.1 | nM | 6.63 |
| CHEMBL3184300 | — | IC50 | = | 308.5 | nM | 6.51 |
| CHEMBL1788401 | CYCLOBENDAZOLE | IC50 | = | 348.6 | nM | 6.46 |
| CHEMBL1087630 | OXIBENDAZOLE | IC50 | = | 365.3 | nM | 6.44 |
| CHEMBL1569226 | — | IC50 | = | 372.8 | nM | 6.43 |
| CHEMBL178 | DAUNORUBICIN | IC50 | = | 369.1 | nM | 6.43 |
| CHEMBL42442 | OXFENDAZOLE | IC50 | = | 468.3 | nM | 6.33 |
| CHEMBL1473700 | PIROCTONE | IC50 | = | 591.3 | nM | 6.23 |
| CHEMBL922 | ADEFOVIR DIPIVOXIL | IC50 | = | 704.3 | nM | 6.15 |
| CHEMBL2356692 | — | IC50 | = | 709.9 | nM | 6.15 |
| CHEMBL36 | PYRIMETHAMINE | IC50 | = | 860.0 | nM | 6.07 |
| CHEMBL31965 | CANERTINIB | IC50 | = | 1001.7 | nM | 6.00 |
| CHEMBL549473 | DIPYRITHIONE | IC50 | = | 991.4 | nM | 6.00 |
| CHEMBL1320139 | HELIOMYCIN | IC50 | = | 1071.5 | nM | 5.97 |
| CHEMBL113051 | GIMATECAN | IC50 | = | 1157.1 | nM | 5.94 |
| CHEMBL1483 | ALBENDAZOLE | IC50 | = | 1276.4 | nM | 5.89 |
| CHEMBL3184339 | — | IC50 | = | 1513.3 | nM | 5.82 |
| CHEMBL1448 | NICLOSAMIDE | IC50 | = | 1570.8 | nM | 5.80 |
| CHEMBL685 | MEBENDAZOLE | IC50 | = | 1738.7 | nM | 5.76 |
| CHEMBL429023 | ROTENONE | IC50 | = | 2987.5 | nM | 5.53 |
| CHEMBL51483 | GOSSYPOL | IC50 | = | 3485.9 | nM | 5.46 |
| CHEMBL1405447 | VITAMIN K3H2 | IC50 | = | 4394.6 | nM | 5.36 |
| CHEMBL2355051 | CLOMIPHENE | IC50 | = | 4351.6 | nM | 5.36 |
| CHEMBL420762 | MOZAVAPTAN | IC50 | = | 4559.3 | nM | 5.34 |
| CHEMBL37161 | FENBENDAZOLE | IC50 | = | 4841.3 | nM | 5.32 |
| CHEMBL460499 | CARMOFUR | IC50 | = | 4982.9 | nM | 5.30 |
| CHEMBL17205 | CYCLOVALONE | IC50 | = | 5045.0 | nM | 5.30 |
| CHEMBL221872 | — | IC50 | = | 5292.3 | nM | 5.28 |
| CHEMBL449782 | CEPHARANTHINE | IC50 | = | 5630.1 | nM | 5.25 |