Assay Detail
Functional
CHEMBL3562021
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PubChem BioAssay. RKO viability from Cell TiterGlo-IC50. (Class of assay: confirmatory)
234
Total Activities
233
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 234 | 6.44 | 9.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3182961 | — | — | 1 | 9.00 |
| CHEMBL1448 | NICLOSAMIDE | 4.0 | 1 | 9.00 |
| CHEMBL917 | FLOXURIDINE | 4.0 | 1 | 9.00 |
| CHEMBL42442 | OXFENDAZOLE | 2.0 | 1 | 9.00 |
| CHEMBL37161 | FENBENDAZOLE | 2.0 | 1 | 9.00 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 9.00 |
| CHEMBL378544 | VINBLASTINE SULFATE | 4.0 | 2 | 9.00 |
| CHEMBL290106 | BITHIONOL | 4.0 | 1 | 9.00 |
| CHEMBL1750 | CLOFARABINE | 4.0 | 1 | 9.00 |
| CHEMBL34259 | METHOTREXATE | 4.0 | 1 | 9.00 |
| CHEMBL2358886 | — | — | 1 | 8.56 |
| CHEMBL140144 | — | — | 1 | 8.54 |
| CHEMBL24944 | TRIBROMSALAN | 4.0 | 1 | 8.52 |
| CHEMBL1981438 | CLOFLUCARBAN | 2.0 | 1 | 8.52 |
| CHEMBL232201 | BENZIODARONE | 4.0 | 1 | 8.52 |
| CHEMBL105442 | CI-1040 | 2.0 | 1 | 8.50 |
| CHEMBL451887 | CARFILZOMIB | 4.0 | 1 | 8.40 |
| CHEMBL3559830 | — | — | 1 | 8.09 |
| CHEMBL50588 | EMETINE | 4.0 | 1 | 8.08 |
| CHEMBL81782 | — | — | 1 | 8.05 |
| CHEMBL2361697 | — | — | 1 | 7.89 |
| CHEMBL2360738 | — | — | 1 | 7.89 |
| CHEMBL448290 | THIOINOSINE | -1.0 | 1 | 7.84 |
| CHEMBL86754 | IODOQUINOL | 2.0 | 1 | 7.64 |
| CHEMBL287542 | RAFOXANIDE | 2.0 | 1 | 7.52 |
| CHEMBL2359490 | — | — | 1 | 7.48 |
| CHEMBL1607 | TOPOTECAN HYDROCHLORIDE | 4.0 | 1 | 7.47 |
| CHEMBL3185933 | IODOPHTHALEIN SODIUM | 2.0 | 1 | 7.43 |
| CHEMBL1200596 | CHLOROXINE | 4.0 | 1 | 7.20 |
| CHEMBL1320139 | HELIOMYCIN | 2.0 | 1 | 7.12 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL378544 | VINBLASTINE SULFATE | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL1750 | CLOFARABINE | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL3182961 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL1448 | NICLOSAMIDE | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL917 | FLOXURIDINE | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL37161 | FENBENDAZOLE | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL378544 | VINBLASTINE SULFATE | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL290106 | BITHIONOL | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL42442 | OXFENDAZOLE | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL2358886 | — | IC50 | = | 2.72 | nM | 8.56 |
| CHEMBL140144 | — | IC50 | = | 2.88 | nM | 8.54 |
| CHEMBL232201 | BENZIODARONE | IC50 | = | 3.0 | nM | 8.52 |
| CHEMBL1981438 | CLOFLUCARBAN | IC50 | = | 3.0 | nM | 8.52 |
| CHEMBL24944 | TRIBROMSALAN | IC50 | = | 3.0 | nM | 8.52 |
| CHEMBL105442 | CI-1040 | IC50 | = | 3.19 | nM | 8.50 |
| CHEMBL451887 | CARFILZOMIB | IC50 | = | 3.94 | nM | 8.40 |
| CHEMBL3559830 | — | IC50 | = | 8.1 | nM | 8.09 |
| CHEMBL50588 | EMETINE | IC50 | = | 8.31 | nM | 8.08 |
| CHEMBL81782 | — | IC50 | = | 8.98 | nM | 8.05 |
| CHEMBL2360738 | — | IC50 | = | 12.8 | nM | 7.89 |
| CHEMBL2361697 | — | IC50 | = | 12.81 | nM | 7.89 |
| CHEMBL448290 | THIOINOSINE | IC50 | = | 14.37 | nM | 7.84 |
| CHEMBL86754 | IODOQUINOL | IC50 | = | 22.7 | nM | 7.64 |
| CHEMBL287542 | RAFOXANIDE | IC50 | = | 30.3 | nM | 7.52 |
| CHEMBL2359490 | — | IC50 | = | 33.16 | nM | 7.48 |
| CHEMBL1607 | TOPOTECAN HYDROCHLORIDE | IC50 | = | 34.16 | nM | 7.47 |
| CHEMBL3185933 | IODOPHTHALEIN SODIUM | IC50 | = | 37.27 | nM | 7.43 |
| CHEMBL1200596 | CHLOROXINE | IC50 | = | 62.74 | nM | 7.20 |
| CHEMBL1320139 | HELIOMYCIN | IC50 | = | 75.4 | nM | 7.12 |
| CHEMBL550348 | DEFERASIROX | IC50 | = | 100.1 | nM | 7.00 |
| CHEMBL496 | HEXACHLOROPHENE | IC50 | = | 108.5 | nM | 6.96 |
| CHEMBL543876 | — | IC50 | = | 113.0 | nM | 6.95 |
| CHEMBL1450 | ATOVAQUONE | IC50 | = | 114.2 | nM | 6.94 |
| CHEMBL264373 | METOPRINE | IC50 | = | 117.05 | nM | 6.93 |
| CHEMBL1545634 | — | IC50 | = | 118.29 | nM | 6.93 |
| CHEMBL178 | DAUNORUBICIN | IC50 | = | 118.15 | nM | 6.93 |
| CHEMBL473535 | FENTICLOR | IC50 | = | 116.4 | nM | 6.93 |
| CHEMBL292009 | BUPARVAQUONE | IC50 | = | 132.9 | nM | 6.88 |
| CHEMBL388590 | BENZBROMARONE | IC50 | = | 131.2 | nM | 6.88 |
| CHEMBL127516 | BUTAMBEN | IC50 | = | 136.8 | nM | 6.86 |
| CHEMBL1325297 | — | IC50 | = | 142.4 | nM | 6.85 |
| CHEMBL5219790 | CETRIMIDE | IC50 | = | 147.3 | nM | 6.83 |
| CHEMBL1788401 | CYCLOBENDAZOLE | IC50 | = | 162.2 | nM | 6.79 |
| CHEMBL223448 | BROXYQUINOLINE | IC50 | = | 163.13 | nM | 6.79 |
| CHEMBL1456 | MYCOPHENOLATE MOFETIL | IC50 | = | 164.8 | nM | 6.78 |
| CHEMBL1483 | ALBENDAZOLE | IC50 | = | 165.33 | nM | 6.78 |
| CHEMBL329522 | EXIFONE | IC50 | = | 192.37 | nM | 6.72 |
| CHEMBL12131 | CLOSANTEL | IC50 | = | 197.1 | nM | 6.71 |