Assay Detail
Functional
CHEMBL3562027
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PubChem BioAssay. HCT116 viability from Cell TiterGlo-IC50. (Class of assay: confirmatory)
232
Total Activities
232
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 232 | 6.40 | 9.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL917 | FLOXURIDINE | 4.0 | 1 | 9.00 |
| CHEMBL42442 | OXFENDAZOLE | 2.0 | 1 | 9.00 |
| CHEMBL37161 | FENBENDAZOLE | 2.0 | 1 | 9.00 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 9.00 |
| CHEMBL290106 | BITHIONOL | 4.0 | 1 | 9.00 |
| CHEMBL378544 | VINBLASTINE SULFATE | 4.0 | 1 | 9.00 |
| CHEMBL1750 | CLOFARABINE | 4.0 | 1 | 9.00 |
| CHEMBL34259 | METHOTREXATE | 4.0 | 1 | 9.00 |
| CHEMBL1448 | NICLOSAMIDE | 4.0 | 1 | 8.84 |
| CHEMBL105442 | CI-1040 | 2.0 | 1 | 8.75 |
| CHEMBL24944 | TRIBROMSALAN | 4.0 | 1 | 8.52 |
| CHEMBL1981438 | CLOFLUCARBAN | 2.0 | 1 | 8.52 |
| CHEMBL232201 | BENZIODARONE | 4.0 | 1 | 8.52 |
| CHEMBL3559830 | — | — | 1 | 8.44 |
| CHEMBL140144 | — | — | 1 | 8.37 |
| CHEMBL451887 | CARFILZOMIB | 4.0 | 1 | 8.25 |
| CHEMBL81782 | — | — | 1 | 8.02 |
| CHEMBL287542 | RAFOXANIDE | 2.0 | 1 | 7.77 |
| CHEMBL1545634 | — | — | 1 | 7.75 |
| CHEMBL2358886 | — | — | 1 | 7.64 |
| CHEMBL2361697 | — | — | 1 | 7.62 |
| CHEMBL448290 | THIOINOSINE | -1.0 | 1 | 7.54 |
| CHEMBL496 | HEXACHLOROPHENE | 4.0 | 1 | 7.51 |
| CHEMBL1607 | TOPOTECAN HYDROCHLORIDE | 4.0 | 1 | 7.47 |
| CHEMBL86754 | IODOQUINOL | 2.0 | 1 | 7.39 |
| CHEMBL1200596 | CHLOROXINE | 4.0 | 1 | 7.32 |
| CHEMBL178 | DAUNORUBICIN | 4.0 | 1 | 7.29 |
| CHEMBL50588 | EMETINE | 4.0 | 1 | 7.21 |
| CHEMBL1456 | MYCOPHENOLATE MOFETIL | 4.0 | 1 | 7.17 |
| CHEMBL1320139 | HELIOMYCIN | 2.0 | 1 | 7.11 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL42442 | OXFENDAZOLE | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL37161 | FENBENDAZOLE | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL378544 | VINBLASTINE SULFATE | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL290106 | BITHIONOL | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL1750 | CLOFARABINE | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL917 | FLOXURIDINE | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL1448 | NICLOSAMIDE | IC50 | = | 1.44 | nM | 8.84 |
| CHEMBL105442 | CI-1040 | IC50 | = | 1.79 | nM | 8.75 |
| CHEMBL1981438 | CLOFLUCARBAN | IC50 | = | 3.0 | nM | 8.52 |
| CHEMBL24944 | TRIBROMSALAN | IC50 | = | 3.0 | nM | 8.52 |
| CHEMBL232201 | BENZIODARONE | IC50 | = | 3.0 | nM | 8.52 |
| CHEMBL3559830 | — | IC50 | = | 3.65 | nM | 8.44 |
| CHEMBL140144 | — | IC50 | = | 4.24 | nM | 8.37 |
| CHEMBL451887 | CARFILZOMIB | IC50 | = | 5.58 | nM | 8.25 |
| CHEMBL81782 | — | IC50 | = | 9.57 | nM | 8.02 |
| CHEMBL287542 | RAFOXANIDE | IC50 | = | 16.95 | nM | 7.77 |
| CHEMBL1545634 | — | IC50 | = | 17.87 | nM | 7.75 |
| CHEMBL2358886 | — | IC50 | = | 23.09 | nM | 7.64 |
| CHEMBL2361697 | — | IC50 | = | 24.06 | nM | 7.62 |
| CHEMBL448290 | THIOINOSINE | IC50 | = | 28.58 | nM | 7.54 |
| CHEMBL496 | HEXACHLOROPHENE | IC50 | = | 31.21 | nM | 7.51 |
| CHEMBL1607 | TOPOTECAN HYDROCHLORIDE | IC50 | = | 34.08 | nM | 7.47 |
| CHEMBL86754 | IODOQUINOL | IC50 | = | 40.97 | nM | 7.39 |
| CHEMBL1200596 | CHLOROXINE | IC50 | = | 47.46 | nM | 7.32 |
| CHEMBL178 | DAUNORUBICIN | IC50 | = | 50.86 | nM | 7.29 |
| CHEMBL50588 | EMETINE | IC50 | = | 61.47 | nM | 7.21 |
| CHEMBL1456 | MYCOPHENOLATE MOFETIL | IC50 | = | 67.2 | nM | 7.17 |
| CHEMBL1320139 | HELIOMYCIN | IC50 | = | 77.47 | nM | 7.11 |
| CHEMBL12131 | CLOSANTEL | IC50 | = | 97.75 | nM | 7.01 |
| CHEMBL1483 | ALBENDAZOLE | IC50 | = | 111.8 | nM | 6.95 |
| CHEMBL2360738 | — | IC50 | = | 135.7 | nM | 6.87 |
| CHEMBL1450 | ATOVAQUONE | IC50 | = | 138.4 | nM | 6.86 |
| CHEMBL727 | THIOGUANINE | IC50 | = | 138.55 | nM | 6.86 |
| CHEMBL1788401 | CYCLOBENDAZOLE | IC50 | = | 173.5 | nM | 6.76 |
| CHEMBL473535 | FENTICLOR | IC50 | = | 182.8 | nM | 6.74 |
| CHEMBL223448 | BROXYQUINOLINE | IC50 | = | 192.72 | nM | 6.71 |
| CHEMBL1542 | AZATHIOPRINE | IC50 | = | 207.39 | nM | 6.68 |
| CHEMBL1076347 | TRICLOCARBAN | IC50 | = | 227.9 | nM | 6.64 |
| CHEMBL292009 | BUPARVAQUONE | IC50 | = | 226.8 | nM | 6.64 |
| CHEMBL1200563 | CERIVASTATIN SODIUM | IC50 | = | 240.31 | nM | 6.62 |
| CHEMBL1425 | MERCAPTOPURINE ANHYDROUS | IC50 | = | 259.1 | nM | 6.59 |
| CHEMBL3185933 | IODOPHTHALEIN SODIUM | IC50 | = | 384.3 | nM | 6.42 |
| CHEMBL2355158 | — | IC50 | = | 394.0 | nM | 6.41 |
| CHEMBL497 | CLIOQUINOL | IC50 | = | 391.7 | nM | 6.41 |
| CHEMBL264373 | METOPRINE | IC50 | = | 413.42 | nM | 6.38 |
| CHEMBL550348 | DEFERASIROX | IC50 | = | 437.57 | nM | 6.36 |
| CHEMBL3188653 | — | IC50 | = | 485.48 | nM | 6.31 |
| CHEMBL64894 | GENTIAN VIOLET | IC50 | = | 513.7 | nM | 6.29 |