Assay Detail
ADMET
CHEMBL3880353
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Antiproliferative activity against mouse BA/F3 cells in presence of mouse IL3 after 72 hrs by Alamar blue assay
30
Total Activities
30
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | ADMET |
| Organism | Mus musculus |
| Cell Type | BaF3 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Pyrazolyl quinoxaline kinase inhibitors
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 30 | 5.72 | 6.35 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3961923 | — | — | 1 | 6.35 |
| CHEMBL3951316 | — | — | 1 | 6.31 |
| CHEMBL3934596 | — | — | 1 | 6.23 |
| CHEMBL3971277 | — | — | 1 | 6.21 |
| CHEMBL3927947 | — | — | 1 | 6.21 |
| CHEMBL3981706 | — | — | 1 | 6.08 |
| CHEMBL3919730 | — | — | 1 | 5.96 |
| CHEMBL3967645 | — | — | 1 | 5.96 |
| CHEMBL3954671 | — | — | 1 | 5.80 |
| CHEMBL3898322 | — | — | 1 | 5.80 |
| CHEMBL3956164 | — | — | 1 | 5.77 |
| CHEMBL3956571 | — | — | 1 | 5.72 |
| CHEMBL3931381 | — | — | 1 | 5.72 |
| CHEMBL3984039 | — | — | 1 | 5.72 |
| CHEMBL3922586 | — | — | 1 | 5.72 |
| CHEMBL3958312 | — | — | 1 | 5.72 |
| CHEMBL3985332 | — | — | 1 | 5.72 |
| CHEMBL3962736 | — | — | 1 | 5.72 |
| CHEMBL3931421 | — | — | 1 | 5.64 |
| CHEMBL3955800 | — | — | 1 | 5.64 |
| CHEMBL3932112 | — | — | 1 | 5.60 |
| CHEMBL3978453 | — | — | 1 | 5.60 |
| CHEMBL3922418 | — | — | 1 | 5.55 |
| CHEMBL3942763 | — | — | 1 | 5.46 |
| CHEMBL3890126 | — | — | 1 | 5.44 |
| CHEMBL3939439 | — | — | 1 | 5.28 |
| CHEMBL3910393 | — | — | 1 | 5.24 |
| CHEMBL3925286 | — | — | 1 | 5.13 |
| CHEMBL3959345 | — | — | 1 | 5.13 |
| CHEMBL3922285 | — | — | 1 | 5.04 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3961923 | — | IC50 | = | 446.68 | nM | 6.35 |
| CHEMBL3951316 | — | IC50 | = | 489.78 | nM | 6.31 |
| CHEMBL3934596 | — | IC50 | = | 588.84 | nM | 6.23 |
| CHEMBL3971277 | — | IC50 | = | 616.6 | nM | 6.21 |
| CHEMBL3927947 | — | IC50 | = | 616.6 | nM | 6.21 |
| CHEMBL3981706 | — | IC50 | = | 831.76 | nM | 6.08 |
| CHEMBL3919730 | — | IC50 | = | 1096.48 | nM | 5.96 |
| CHEMBL3967645 | — | IC50 | = | 1096.48 | nM | 5.96 |
| CHEMBL3954671 | — | IC50 | = | 1584.89 | nM | 5.80 |
| CHEMBL3898322 | — | IC50 | = | 1584.89 | nM | 5.80 |
| CHEMBL3956164 | — | IC50 | = | 1698.24 | nM | 5.77 |
| CHEMBL3956571 | — | IC50 | = | 1905.46 | nM | 5.72 |
| CHEMBL3931381 | — | IC50 | = | 1905.46 | nM | 5.72 |
| CHEMBL3984039 | — | IC50 | = | 1905.46 | nM | 5.72 |
| CHEMBL3922586 | — | IC50 | = | 1905.46 | nM | 5.72 |
| CHEMBL3958312 | — | IC50 | = | 1905.46 | nM | 5.72 |
| CHEMBL3985332 | — | IC50 | = | 1905.46 | nM | 5.72 |
| CHEMBL3962736 | — | IC50 | = | 1905.46 | nM | 5.72 |
| CHEMBL3931421 | — | IC50 | = | 2290.87 | nM | 5.64 |
| CHEMBL3955800 | — | IC50 | = | 2290.87 | nM | 5.64 |
| CHEMBL3932112 | — | IC50 | = | 2511.89 | nM | 5.60 |
| CHEMBL3978453 | — | IC50 | = | 2511.89 | nM | 5.60 |
| CHEMBL3922418 | — | IC50 | = | 2818.38 | nM | 5.55 |
| CHEMBL3942763 | — | IC50 | = | 3467.37 | nM | 5.46 |
| CHEMBL3890126 | — | IC50 | = | 3630.78 | nM | 5.44 |
| CHEMBL3939439 | — | IC50 | = | 5248.07 | nM | 5.28 |
| CHEMBL3910393 | — | IC50 | = | 5754.4 | nM | 5.24 |
| CHEMBL3925286 | — | IC50 | = | 7413.1 | nM | 5.13 |
| CHEMBL3959345 | — | IC50 | = | 7413.1 | nM | 5.13 |
| CHEMBL3922285 | — | IC50 | = | 9120.11 | nM | 5.04 |