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Assay Detail

CHEMBL5232718

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of human PDE4 catalytic domain expressed in Escherichia coli
12
Total Activities
12
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

3',5'-cyclic-AMP phosphodiesterase 4B (CHEMBL275)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Targeting Metalloenzymes by Boron-Containing Metal-Binding Pharmacophores.
Xiao YC, Yu JL, Dai QQ, Li G, Li GB.
J Med Chem (2021) 64 : 17706 -17727
PubMed 34875836 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 12 8.43 10.30

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5268572 1 10.30
CHEMBL5268265 1 9.92
CHEMBL5289939 1 9.62
CHEMBL4872870 1 9.38
CHEMBL5290174 1 9.15
CHEMBL5278590 1 7.62
CHEMBL1093373 1 7.33
CHEMBL4467344 1 7.22
CHEMBL484785 CRISABOROLE 4.0 1 6.96
CHEMBL1093962 1 6.75
CHEMBL5281157 1 -
CHEMBL1093374 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5268572 IC50 = 0.05 nM 10.30
CHEMBL5268265 IC50 = 0.12 nM 9.92
CHEMBL5289939 IC50 = 0.24 nM 9.62
CHEMBL4872870 IC50 = 0.42 nM 9.38
CHEMBL5290174 IC50 = 0.7 nM 9.15
CHEMBL5278590 IC50 = 24.0 nM 7.62
CHEMBL1093373 IC50 = 47.0 nM 7.33
CHEMBL4467344 IC50 = 60.0 nM 7.22
CHEMBL484785 CRISABOROLE IC50 = 110.0 nM 6.96
CHEMBL1093962 IC50 = 180.0 nM 6.75
CHEMBL5281157 IC50 > 100.0 nM -
CHEMBL1093374 IC50 > 10.0 nM -