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Compound Detail

CHEMBL4447775

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Nc1ncnc2c1c1occc1n2[C@@H]1O[C@H](CO)[C@@H](O)[C@H]1O

Basic Information

ChEMBL ID CHEMBL4447775
Phase Preclinical
Structure Type MOL
InChI Key WQNNJYMNIVAWCW-HTVVRFAVSA-N
8
Targets
9
Activities
2
Assay Types
0
PK Parameters
19
Publications
0
Known Names

Molecular Properties

306.3
MW (Da)
-0.63
ALogP
9
HBA
4
HBD
139.8
PSA (Ų)
0.49
QED
0
Ro5 Violations
2
Rot. Bonds

Drug Information

Molecule Type Unknown
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C13H14N4O5
MW 306.28
Aromatic Rings 3
Heavy Atoms 22
NP-Likeness 0.87

Activity Summary

IC50 7 meas. best 6.29
EC50 2 meas. best 6.52

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Hepatitis C virus
CHEMBL379
EC50 6.52 6.5 300.0 2
HL-60
CHEMBL383
IC50 6.29 6.29 510.0 1
HeLa S3
CHEMBL4296436
IC50 5.77 5.77 1710.0 1
HepG2
CHEMBL395
IC50 5.35 5.35 4510.0 1
K562
CHEMBL385
IC50 5.22 5.22 6040.0 1
U2OS
CHEMBL615023
IC50 5.15 5.15 7090.0 1
HCT-116
CHEMBL394
IC50 4.32 4.32 48420.0 1
Unchecked
CHEMBL612545
IC50 4.3 4.3 50000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

Data from ChEMBL 36 via Core Engine