Assay Detail
Functional
CHEMBL1613791
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: A counter screen for small molecule screen for inhibitors of the PhoP region in Salmonella typhi. (Class of assay: confirmatory) [Related pubchem assays: 1850, 1864, 2252, 1985 ]
1126
Total Activities
1121
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1126 | 4.50 | 6.62 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1594055 | — | — | 1 | 6.62 |
| CHEMBL1523989 | — | — | 1 | 6.57 |
| CHEMBL1551640 | — | — | 1 | 6.51 |
| CHEMBL458019 | PARAQUAT DICHLORIDE | — | 1 | 6.32 |
| CHEMBL9 | NORFLOXACIN | 4.0 | 1 | 6.31 |
| CHEMBL1430611 | — | — | 1 | 6.28 |
| CHEMBL15511 | ENROFLOXACIN | 2.0 | 1 | 6.28 |
| CHEMBL1572266 | — | — | 1 | 6.19 |
| CHEMBL1485275 | — | — | 1 | 6.17 |
| CHEMBL5315124 | LEVOFLOXACIN | 4.0 | 1 | 6.16 |
| CHEMBL1454910 | NITROXOLINE | 4.0 | 1 | 6.10 |
| CHEMBL1513204 | — | — | 1 | 6.09 |
| CHEMBL22 | TRIMETHOPRIM | 4.0 | 1 | 6.09 |
| CHEMBL1593697 | — | — | 1 | 6.08 |
| CHEMBL240163 | PAZUFLOXACIN | 3.0 | 1 | 6.05 |
| CHEMBL283849 | — | — | 1 | 5.97 |
| CHEMBL31 | GATIFLOXACIN | 4.0 | 1 | 5.96 |
| CHEMBL1428564 | PEFLOXACIN MESYLATE | -1.0 | 1 | 5.91 |
| CHEMBL1200735 | MOXIFLOXACIN HYDROCHLORIDE | 4.0 | 1 | 5.90 |
| CHEMBL529 | AZITHROMYCIN | 4.0 | 1 | 5.89 |
| CHEMBL104270 | TOSUFLOXACIN TOSYLATE | — | 1 | 5.82 |
| CHEMBL1200567 | — | — | 1 | 5.81 |
| CHEMBL130 | CHLORAMPHENICOL | 4.0 | 1 | 5.80 |
| CHEMBL1545940 | — | — | 1 | 5.77 |
| CHEMBL1315061 | — | — | 1 | 5.77 |
| CHEMBL4 | OFLOXACIN | 4.0 | 1 | 5.76 |
| CHEMBL1364939 | — | — | 1 | 5.75 |
| CHEMBL1456906 | — | — | 1 | 5.66 |
| CHEMBL601757 | — | — | 1 | 5.63 |
| CHEMBL578512 | — | — | 1 | 5.60 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1594055 | — | IC50 | = | 240.0 | nM | 6.62 |
| CHEMBL1523989 | — | IC50 | = | 270.0 | nM | 6.57 |
| CHEMBL1551640 | — | IC50 | = | 310.0 | nM | 6.51 |
| CHEMBL458019 | PARAQUAT DICHLORIDE | IC50 | = | 480.0 | nM | 6.32 |
| CHEMBL9 | NORFLOXACIN | IC50 | = | 490.0 | nM | 6.31 |
| CHEMBL1430611 | — | IC50 | = | 530.0 | nM | 6.28 |
| CHEMBL15511 | ENROFLOXACIN | IC50 | = | 520.0 | nM | 6.28 |
| CHEMBL1572266 | — | IC50 | = | 650.0 | nM | 6.19 |
| CHEMBL1485275 | — | IC50 | = | 680.0 | nM | 6.17 |
| CHEMBL5315124 | LEVOFLOXACIN | IC50 | = | 690.0 | nM | 6.16 |
| CHEMBL1454910 | NITROXOLINE | IC50 | = | 790.0 | nM | 6.10 |
| CHEMBL22 | TRIMETHOPRIM | IC50 | = | 820.0 | nM | 6.09 |
| CHEMBL1513204 | — | IC50 | = | 820.0 | nM | 6.09 |
| CHEMBL1593697 | — | IC50 | = | 830.0 | nM | 6.08 |
| CHEMBL240163 | PAZUFLOXACIN | IC50 | = | 900.0 | nM | 6.05 |
| CHEMBL283849 | — | IC50 | = | 1060.0 | nM | 5.97 |
| CHEMBL31 | GATIFLOXACIN | IC50 | = | 1100.0 | nM | 5.96 |
| CHEMBL1428564 | PEFLOXACIN MESYLATE | IC50 | = | 1230.0 | nM | 5.91 |
| CHEMBL1200735 | MOXIFLOXACIN HYDROCHLORIDE | IC50 | = | 1260.0 | nM | 5.90 |
| CHEMBL529 | AZITHROMYCIN | IC50 | = | 1280.0 | nM | 5.89 |
| CHEMBL104270 | TOSUFLOXACIN TOSYLATE | IC50 | = | 1530.0 | nM | 5.82 |
| CHEMBL1200567 | — | IC50 | = | 1560.0 | nM | 5.81 |
| CHEMBL130 | CHLORAMPHENICOL | IC50 | = | 1570.0 | nM | 5.80 |
| CHEMBL1545940 | — | IC50 | = | 1690.0 | nM | 5.77 |
| CHEMBL1315061 | — | IC50 | = | 1710.0 | nM | 5.77 |
| CHEMBL4 | OFLOXACIN | IC50 | = | 1730.0 | nM | 5.76 |
| CHEMBL1364939 | — | IC50 | = | 1780.0 | nM | 5.75 |
| CHEMBL1456906 | — | IC50 | = | 2190.0 | nM | 5.66 |
| CHEMBL601757 | — | IC50 | = | 2320.0 | nM | 5.63 |
| CHEMBL578512 | — | IC50 | = | 2530.0 | nM | 5.60 |
| CHEMBL185 | FLUOROURACIL | IC50 | = | 2530.0 | nM | 5.60 |
| CHEMBL414400 | — | IC50 | = | 3020.0 | nM | 5.52 |
| CHEMBL521078 | PORFIROMYCIN | IC50 | = | 3120.0 | nM | 5.51 |
| CHEMBL466853 | — | IC50 | = | 3100.0 | nM | 5.51 |
| CHEMBL428064 | — | IC50 | = | 3320.0 | nM | 5.48 |
| CHEMBL1342852 | — | IC50 | = | 3740.0 | nM | 5.43 |
| CHEMBL1327202 | — | IC50 | = | 3820.0 | nM | 5.42 |
| CHEMBL1385808 | — | IC50 | = | 3900.0 | nM | 5.41 |
| CHEMBL2373661 | — | IC50 | = | 3950.0 | nM | 5.40 |
| CHEMBL334707 | — | IC50 | = | 4250.0 | nM | 5.37 |
| CHEMBL1487183 | ALEXIDINE HYDROCHLORIDE | IC50 | = | 4650.0 | nM | 5.33 |
| CHEMBL251670 | (R)-GATIFLOXACIN | IC50 | = | 4980.0 | nM | 5.30 |
| CHEMBL1241590 | FLORFENICOL | IC50 | = | 5150.0 | nM | 5.29 |
| CHEMBL790 | CHLORHEXIDINE | IC50 | = | 5130.0 | nM | 5.29 |
| CHEMBL1330113 | — | IC50 | = | 5200.0 | nM | 5.28 |
| CHEMBL1318861 | — | IC50 | = | 5310.0 | nM | 5.28 |
| CHEMBL1330113 | — | IC50 | = | 5400.0 | nM | 5.27 |
| CHEMBL1237072 | DIRITHROMYCIN | IC50 | = | 5520.0 | nM | 5.26 |
| CHEMBL1389315 | — | IC50 | = | 5670.0 | nM | 5.25 |
| CHEMBL497 | CLIOQUINOL | IC50 | = | 5620.0 | nM | 5.25 |