Assay Detail
Functional
CHEMBL1614374
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Absorbance Microorganism-Based Dose Response Follow up to Identify Inhibitors of Streptokinase Expression. (Class of assay: confirmatory) [Related pubchem assays: 1677 (Project Summary), 1915, 1914, 1902 (Retest at Dose), 1900 (Counter Screen), 1662 (Primary HTS)]
63
Total Activities
62
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Streptococcus pyogenes M1 GAS |
| Category | confirmatory |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
Streptokinase A (CHEMBL1293228) ↗| Type | SINGLE PROTEIN |
| Organism | Streptococcus pyogenes serotype M1 |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 63 | 5.17 | 6.38 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1393959 | — | — | 1 | 6.38 |
| CHEMBL1407961 | — | — | 1 | 5.93 |
| CHEMBL1530048 | — | — | 1 | 5.79 |
| CHEMBL1422105 | — | — | 1 | 5.79 |
| CHEMBL1587193 | — | — | 1 | 5.76 |
| CHEMBL1336879 | — | — | 1 | 5.65 |
| CHEMBL1450241 | — | — | 1 | 5.64 |
| CHEMBL1341100 | — | — | 1 | 5.54 |
| CHEMBL1369724 | — | — | 1 | 5.53 |
| CHEMBL1591750 | — | — | 1 | 5.51 |
| CHEMBL1331239 | — | — | 1 | 5.50 |
| CHEMBL1380929 | — | — | 1 | 5.47 |
| CHEMBL1478693 | — | — | 1 | 5.45 |
| CHEMBL1358236 | — | — | 1 | 5.45 |
| CHEMBL1333583 | — | — | 1 | 5.44 |
| CHEMBL1305704 | — | — | 1 | 5.44 |
| CHEMBL1437208 | — | — | 1 | 5.40 |
| CHEMBL1314635 | — | — | 1 | 5.40 |
| CHEMBL1327366 | — | — | 1 | 5.40 |
| CHEMBL1429121 | — | — | 1 | 5.39 |
| CHEMBL1394006 | — | — | 1 | 5.39 |
| CHEMBL1338958 | — | — | 1 | 5.38 |
| CHEMBL1544494 | — | — | 1 | 5.36 |
| CHEMBL1351184 | — | — | 1 | 5.36 |
| CHEMBL1567814 | — | — | 1 | 5.31 |
| CHEMBL1511988 | — | — | 1 | 5.27 |
| CHEMBL1371202 | — | — | 2 | 5.25 |
| CHEMBL1527478 | — | — | 1 | 5.24 |
| CHEMBL1449558 | — | — | 1 | 5.23 |
| CHEMBL1488460 | — | — | 1 | 5.23 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1393959 | — | EC50 | = | 419.0 | nM | 6.38 |
| CHEMBL1407961 | — | EC50 | = | 1165.0 | nM | 5.93 |
| CHEMBL1422105 | — | EC50 | = | 1606.0 | nM | 5.79 |
| CHEMBL1530048 | — | EC50 | = | 1641.0 | nM | 5.79 |
| CHEMBL1587193 | — | EC50 | = | 1731.0 | nM | 5.76 |
| CHEMBL1336879 | — | EC50 | = | 2261.0 | nM | 5.65 |
| CHEMBL1450241 | — | EC50 | = | 2267.0 | nM | 5.64 |
| CHEMBL1341100 | — | EC50 | = | 2893.0 | nM | 5.54 |
| CHEMBL1369724 | — | EC50 | = | 2932.0 | nM | 5.53 |
| CHEMBL1591750 | — | EC50 | = | 3096.0 | nM | 5.51 |
| CHEMBL1331239 | — | EC50 | = | 3132.0 | nM | 5.50 |
| CHEMBL1380929 | — | EC50 | = | 3374.0 | nM | 5.47 |
| CHEMBL1478693 | — | EC50 | = | 3540.0 | nM | 5.45 |
| CHEMBL1358236 | — | EC50 | = | 3529.0 | nM | 5.45 |
| CHEMBL1305704 | — | EC50 | = | 3652.0 | nM | 5.44 |
| CHEMBL1333583 | — | EC50 | = | 3627.0 | nM | 5.44 |
| CHEMBL1327366 | — | EC50 | = | 3942.0 | nM | 5.40 |
| CHEMBL1437208 | — | EC50 | = | 4003.0 | nM | 5.40 |
| CHEMBL1314635 | — | EC50 | = | 3966.0 | nM | 5.40 |
| CHEMBL1429121 | — | EC50 | = | 4025.0 | nM | 5.39 |
| CHEMBL1394006 | — | EC50 | = | 4095.0 | nM | 5.39 |
| CHEMBL1338958 | — | EC50 | = | 4147.0 | nM | 5.38 |
| CHEMBL1544494 | — | EC50 | = | 4387.0 | nM | 5.36 |
| CHEMBL1351184 | — | EC50 | = | 4400.0 | nM | 5.36 |
| CHEMBL1567814 | — | EC50 | = | 4940.0 | nM | 5.31 |
| CHEMBL1511988 | — | EC50 | = | 5418.0 | nM | 5.27 |
| CHEMBL1371202 | — | EC50 | = | 5597.0 | nM | 5.25 |
| CHEMBL1527478 | — | EC50 | = | 5698.0 | nM | 5.24 |
| CHEMBL1488460 | — | EC50 | = | 5929.0 | nM | 5.23 |
| CHEMBL1449558 | — | EC50 | = | 5898.0 | nM | 5.23 |
| CHEMBL1318434 | — | EC50 | = | 6357.0 | nM | 5.20 |
| CHEMBL1589740 | — | EC50 | = | 6274.0 | nM | 5.20 |
| CHEMBL1475828 | — | EC50 | = | 6537.0 | nM | 5.18 |
| CHEMBL1394162 | — | EC50 | = | 6624.0 | nM | 5.18 |
| CHEMBL1302315 | — | EC50 | = | 6675.0 | nM | 5.18 |
| CHEMBL1383137 | — | EC50 | = | 7089.0 | nM | 5.15 |
| CHEMBL1368435 | — | EC50 | = | 7588.0 | nM | 5.12 |
| CHEMBL1371202 | — | EC50 | = | 7602.0 | nM | 5.12 |
| CHEMBL1435608 | — | EC50 | = | 7953.0 | nM | 5.10 |
| CHEMBL1473390 | — | EC50 | = | 8380.0 | nM | 5.08 |
| CHEMBL1240975 | HYPOSTATIN | EC50 | = | 8369.0 | nM | 5.08 |
| CHEMBL1589702 | — | EC50 | = | 9115.0 | nM | 5.04 |
| CHEMBL1533974 | — | EC50 | = | 9181.0 | nM | 5.04 |
| CHEMBL1414059 | — | EC50 | = | 9541.0 | nM | 5.02 |
| CHEMBL1565485 | — | EC50 | = | 10085.0 | nM | 5.00 |
| CHEMBL1528266 | — | EC50 | = | 10357.0 | nM | 4.99 |
| CHEMBL1447853 | — | EC50 | = | 12553.0 | nM | 4.90 |
| CHEMBL1314004 | — | EC50 | = | 13731.0 | nM | 4.86 |
| CHEMBL1487309 | — | EC50 | = | 14159.0 | nM | 4.85 |
| CHEMBL1471371 | — | EC50 | = | 14954.0 | nM | 4.83 |