Assay Detail
Binding
CHEMBL1614548
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: uHTS fluorescence polarization assay for the identification of translation initiation inhibitors (PABP). (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID2012, AID2030, AID435011, AID435018, AID449744, AID449751, AID449752]
156
Total Activities
156
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 156 | 4.95 | 5.73 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL592588 | — | — | 1 | 5.73 |
| CHEMBL1423915 | — | — | 1 | 5.73 |
| CHEMBL589711 | — | — | 1 | 5.65 |
| CHEMBL1383779 | — | — | 1 | 5.61 |
| CHEMBL1577127 | — | — | 1 | 5.57 |
| CHEMBL1445700 | — | — | 1 | 5.56 |
| CHEMBL1563641 | — | — | 1 | 5.55 |
| CHEMBL1301276 | — | — | 1 | 5.49 |
| CHEMBL1303289 | — | — | 1 | 5.49 |
| CHEMBL1377588 | — | — | 1 | 5.48 |
| CHEMBL1497097 | — | — | 1 | 5.46 |
| CHEMBL3197066 | — | — | 1 | 5.45 |
| CHEMBL1789987 | — | — | 1 | 5.43 |
| CHEMBL1342158 | — | — | 1 | 5.42 |
| CHEMBL1464460 | — | — | 1 | 5.40 |
| CHEMBL1324692 | — | — | 1 | 5.39 |
| CHEMBL1505531 | — | — | 1 | 5.39 |
| CHEMBL1359526 | — | — | 1 | 5.37 |
| CHEMBL1364684 | — | — | 1 | 5.37 |
| CHEMBL3195960 | — | — | 1 | 5.36 |
| CHEMBL1416798 | — | — | 1 | 5.36 |
| CHEMBL1469272 | — | — | 1 | 5.35 |
| CHEMBL1469858 | — | — | 1 | 5.34 |
| CHEMBL1332525 | — | — | 1 | 5.34 |
| CHEMBL1562954 | — | — | 1 | 5.34 |
| CHEMBL1480280 | — | — | 1 | 5.31 |
| CHEMBL1319469 | — | — | 1 | 5.31 |
| CHEMBL3196705 | — | — | 1 | 5.29 |
| CHEMBL1388052 | — | — | 1 | 5.28 |
| CHEMBL1573412 | — | — | 1 | 5.27 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL592588 | — | IC50 | = | 1870.0 | nM | 5.73 |
| CHEMBL1423915 | — | IC50 | = | 1850.0 | nM | 5.73 |
| CHEMBL589711 | — | IC50 | = | 2220.0 | nM | 5.65 |
| CHEMBL1383779 | — | IC50 | = | 2480.0 | nM | 5.61 |
| CHEMBL1577127 | — | IC50 | = | 2725.0 | nM | 5.57 |
| CHEMBL1445700 | — | IC50 | = | 2760.0 | nM | 5.56 |
| CHEMBL1563641 | — | IC50 | = | 2810.0 | nM | 5.55 |
| CHEMBL1301276 | — | IC50 | = | 3250.0 | nM | 5.49 |
| CHEMBL1303289 | — | IC50 | = | 3265.0 | nM | 5.49 |
| CHEMBL1377588 | — | IC50 | = | 3290.0 | nM | 5.48 |
| CHEMBL1497097 | — | IC50 | = | 3495.0 | nM | 5.46 |
| CHEMBL3197066 | — | IC50 | = | 3565.0 | nM | 5.45 |
| CHEMBL1789987 | — | IC50 | = | 3685.0 | nM | 5.43 |
| CHEMBL1342158 | — | IC50 | = | 3830.0 | nM | 5.42 |
| CHEMBL1464460 | — | IC50 | = | 4000.0 | nM | 5.40 |
| CHEMBL1324692 | — | IC50 | = | 4075.0 | nM | 5.39 |
| CHEMBL1505531 | — | IC50 | = | 4085.0 | nM | 5.39 |
| CHEMBL1364684 | — | IC50 | = | 4320.0 | nM | 5.37 |
| CHEMBL1359526 | — | IC50 | = | 4320.0 | nM | 5.37 |
| CHEMBL3195960 | — | IC50 | = | 4395.0 | nM | 5.36 |
| CHEMBL1416798 | — | IC50 | = | 4405.0 | nM | 5.36 |
| CHEMBL1469272 | — | IC50 | = | 4470.0 | nM | 5.35 |
| CHEMBL1562954 | — | IC50 | = | 4585.0 | nM | 5.34 |
| CHEMBL1469858 | — | IC50 | = | 4535.0 | nM | 5.34 |
| CHEMBL1332525 | — | IC50 | = | 4550.0 | nM | 5.34 |
| CHEMBL1480280 | — | IC50 | = | 4860.0 | nM | 5.31 |
| CHEMBL1319469 | — | IC50 | = | 4910.0 | nM | 5.31 |
| CHEMBL3196705 | — | IC50 | = | 5140.0 | nM | 5.29 |
| CHEMBL1388052 | — | IC50 | = | 5270.0 | nM | 5.28 |
| CHEMBL1320897 | — | IC50 | = | 5405.0 | nM | 5.27 |
| CHEMBL1318253 | — | IC50 | = | 5325.0 | nM | 5.27 |
| CHEMBL1423236 | — | IC50 | = | 5425.0 | nM | 5.27 |
| CHEMBL1573412 | — | IC50 | = | 5320.0 | nM | 5.27 |
| CHEMBL1432423 | — | IC50 | = | 5515.0 | nM | 5.26 |
| CHEMBL1480992 | — | IC50 | = | 5470.0 | nM | 5.26 |
| CHEMBL3210843 | — | IC50 | = | 5575.0 | nM | 5.25 |
| CHEMBL1355123 | — | IC50 | = | 5630.0 | nM | 5.25 |
| CHEMBL1343383 | — | IC50 | = | 5700.0 | nM | 5.24 |
| CHEMBL3213476 | — | IC50 | = | 5825.0 | nM | 5.24 |
| CHEMBL1312519 | — | IC50 | = | 5920.0 | nM | 5.23 |
| CHEMBL1610821 | — | IC50 | = | 5930.0 | nM | 5.23 |
| CHEMBL1378601 | — | IC50 | = | 6050.0 | nM | 5.22 |
| CHEMBL1483521 | — | IC50 | = | 6055.0 | nM | 5.22 |
| CHEMBL1535072 | — | IC50 | = | 5955.0 | nM | 5.22 |
| CHEMBL1422684 | — | IC50 | = | 6205.0 | nM | 5.21 |
| CHEMBL1383109 | — | IC50 | = | 6160.0 | nM | 5.21 |
| CHEMBL1379062 | — | IC50 | = | 6350.0 | nM | 5.20 |
| CHEMBL1547939 | — | IC50 | = | 6515.0 | nM | 5.19 |
| CHEMBL1369880 | — | IC50 | = | 6535.0 | nM | 5.18 |
| CHEMBL1451147 | — | IC50 | = | 6610.0 | nM | 5.18 |