Assay Detail
Binding
CHEMBL1794358
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Counterscreen for IDE activators: Fluorescence polarization-based biochemical high throughput dose response assay for activators of recombinant IDE. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID493087, AID493124, AID588439, AID588440, AID588442]
231
Total Activities
231
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Category | confirmatory |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 231 | 4.94 | 5.88 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1568474 | — | — | 1 | 5.88 |
| CHEMBL1989158 | — | — | 1 | 5.63 |
| CHEMBL1320463 | — | — | 1 | 5.63 |
| CHEMBL857 | BIOTIN | 4.0 | 1 | 5.60 |
| CHEMBL1984581 | — | — | 1 | 5.54 |
| CHEMBL1705738 | — | — | 1 | 5.44 |
| CHEMBL1973159 | — | — | 1 | 5.34 |
| CHEMBL1316468 | — | — | 1 | 5.18 |
| CHEMBL1458111 | — | — | 1 | 5.17 |
| CHEMBL1527972 | — | — | 1 | 5.17 |
| CHEMBL1593621 | — | — | 1 | 5.15 |
| CHEMBL1232381 | — | — | 1 | 5.13 |
| CHEMBL1474028 | — | — | 1 | 5.07 |
| CHEMBL1995720 | — | — | 1 | 5.01 |
| CHEMBL1971127 | — | — | 1 | 5.01 |
| CHEMBL1437186 | — | — | 1 | 4.95 |
| CHEMBL1574420 | — | — | 1 | 4.86 |
| CHEMBL1370780 | — | — | 1 | 4.78 |
| CHEMBL1496705 | — | — | 1 | 4.77 |
| CHEMBL1403262 | — | — | 1 | 4.77 |
| CHEMBL1578670 | — | — | 1 | 4.76 |
| CHEMBL1572827 | — | — | 1 | 4.60 |
| CHEMBL3196438 | — | — | 1 | 4.58 |
| CHEMBL1442125 | — | — | 1 | 4.57 |
| CHEMBL1536835 | — | — | 1 | 4.53 |
| CHEMBL1591898 | — | — | 1 | 4.48 |
| CHEMBL1497597 | — | — | 1 | 4.40 |
| CHEMBL1528386 | — | — | 1 | 4.30 |
| CHEMBL1376516 | — | — | 1 | 4.28 |
| CHEMBL589694 | — | — | 1 | 4.27 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1568474 | — | EC50 | = | 1317.0 | nM | 5.88 |
| CHEMBL1320463 | — | EC50 | = | 2324.0 | nM | 5.63 |
| CHEMBL1989158 | — | EC50 | = | 2356.0 | nM | 5.63 |
| CHEMBL857 | BIOTIN | EC50 | = | 2526.0 | nM | 5.60 |
| CHEMBL1984581 | — | EC50 | = | 2853.0 | nM | 5.54 |
| CHEMBL1705738 | — | EC50 | = | 3639.0 | nM | 5.44 |
| CHEMBL1973159 | — | EC50 | = | 4597.0 | nM | 5.34 |
| CHEMBL1316468 | — | EC50 | = | 6551.0 | nM | 5.18 |
| CHEMBL1458111 | — | EC50 | = | 6694.0 | nM | 5.17 |
| CHEMBL1527972 | — | EC50 | = | 6733.0 | nM | 5.17 |
| CHEMBL1593621 | — | EC50 | = | 7077.0 | nM | 5.15 |
| CHEMBL1232381 | — | EC50 | = | 7406.0 | nM | 5.13 |
| CHEMBL1474028 | — | EC50 | = | 8554.0 | nM | 5.07 |
| CHEMBL1971127 | — | EC50 | = | 9708.0 | nM | 5.01 |
| CHEMBL1995720 | — | EC50 | = | 9666.0 | nM | 5.01 |
| CHEMBL1437186 | — | EC50 | = | 11159.0 | nM | 4.95 |
| CHEMBL1574420 | — | EC50 | = | 13975.0 | nM | 4.86 |
| CHEMBL1370780 | — | EC50 | = | 16789.0 | nM | 4.78 |
| CHEMBL1496705 | — | EC50 | = | 16931.0 | nM | 4.77 |
| CHEMBL1403262 | — | EC50 | = | 16936.0 | nM | 4.77 |
| CHEMBL1578670 | — | EC50 | = | 17262.0 | nM | 4.76 |
| CHEMBL1572827 | — | EC50 | = | 25196.0 | nM | 4.60 |
| CHEMBL3196438 | — | EC50 | = | 25995.0 | nM | 4.58 |
| CHEMBL1442125 | — | EC50 | = | 26856.0 | nM | 4.57 |
| CHEMBL1536835 | — | EC50 | = | 29821.0 | nM | 4.53 |
| CHEMBL1591898 | — | EC50 | = | 32976.0 | nM | 4.48 |
| CHEMBL1497597 | — | EC50 | = | 40117.0 | nM | 4.40 |
| CHEMBL1528386 | — | EC50 | = | 50087.0 | nM | 4.30 |
| CHEMBL1376516 | — | EC50 | = | 52109.0 | nM | 4.28 |
| CHEMBL589694 | — | EC50 | = | 53428.0 | nM | 4.27 |
| CHEMBL1200883 | THONZONIUM BROMIDE | EC50 | = | 53305.0 | nM | 4.27 |
| CHEMBL1486690 | PYRONIN Y | EC50 | > | 54732.0 | nM | - |
| CHEMBL1471509 | — | EC50 | > | 54705.0 | nM | - |
| CHEMBL1528271 | — | EC50 | > | 54690.0 | nM | - |
| CHEMBL1302748 | — | EC50 | > | 54732.0 | nM | - |
| CHEMBL1378294 | — | EC50 | > | 54710.0 | nM | - |
| CHEMBL1708021 | — | EC50 | > | 54689.0 | nM | - |
| CHEMBL1331010 | — | EC50 | > | 54689.0 | nM | - |
| CHEMBL1598570 | — | EC50 | > | 54705.0 | nM | - |
| CHEMBL1331762 | — | EC50 | > | 54705.0 | nM | - |
| CHEMBL1513972 | — | EC50 | > | 54705.0 | nM | - |
| CHEMBL496633 | — | EC50 | > | 54690.0 | nM | - |
| CHEMBL1542526 | — | EC50 | > | 54710.0 | nM | - |
| CHEMBL1337599 | — | EC50 | > | 54705.0 | nM | - |
| CHEMBL1315987 | — | EC50 | > | 2026.0 | nM | - |
| CHEMBL1369287 | — | EC50 | > | 54748.0 | nM | - |
| CHEMBL1345866 | — | EC50 | > | 54687.0 | nM | - |
| CHEMBL1980281 | — | EC50 | > | 54721.0 | nM | - |
| CHEMBL1418096 | — | EC50 | > | 54743.0 | nM | - |
| CHEMBL1372920 | — | EC50 | > | 54683.0 | nM | - |