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Assay Detail

CHEMBL1963787

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: CAMK2B
ChEMBL ↗
606
Total Activities
593
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Category other
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Calcium/calmodulin-dependent protein kinase type II subunit beta (CHEMBL4121) ↗
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

PubChem BioAssay data set

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 606 5.54 7.10

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1966628 — — 1 7.10
CHEMBL1986943 — — 2 7.00
CHEMBL1974870 — — 2 7.00
CHEMBL1998159 — — 1 7.00
CHEMBL1970903 — — 1 7.00
CHEMBL1988537 — — 1 6.70
CHEMBL1973540 — — 1 6.60
CHEMBL2001751 — — 1 6.60
CHEMBL1991063 — — 1 6.60
CHEMBL1995813 — — 1 6.50
CHEMBL1982711 — — 1 6.50
CHEMBL1996817 — — 1 6.50
CHEMBL2002726 — — 1 6.50
CHEMBL1993661 — — 1 6.40
CHEMBL1992634 — — 1 6.40
CHEMBL1982957 — — 1 6.40
CHEMBL1965836 — — 1 6.30
CHEMBL1967887 — — 1 6.20
CHEMBL1975128 — — 2 6.10
CHEMBL509032 TAE-684 — 1 6.10
CHEMBL1965131 — — 1 6.00
CHEMBL1996979 — — 1 6.00
CHEMBL1973860 — — 1 6.00
CHEMBL2000071 — — 1 6.00
CHEMBL2001920 — — 1 6.00
CHEMBL1969588 — — 1 6.00
CHEMBL1973142 — — 1 5.90
CHEMBL1966425 — — 1 5.90
CHEMBL482767 SNS-314 1.0 1 5.90
CHEMBL2003405 — — 1 5.90

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1966628 — Ki = 79.43 nM 7.10
CHEMBL1986943 — Ki = 100.0 nM 7.00
CHEMBL1974870 — Ki = 100.0 nM 7.00
CHEMBL1970903 — Ki = 100.0 nM 7.00
CHEMBL1998159 — Ki = 100.0 nM 7.00
CHEMBL1986943 — Ki = 100.0 nM 7.00
CHEMBL1974870 — Ki = 100.0 nM 7.00
CHEMBL1988537 — Ki = 199.53 nM 6.70
CHEMBL1973540 — Ki = 251.19 nM 6.60
CHEMBL1991063 — Ki = 251.19 nM 6.60
CHEMBL2001751 — Ki = 251.19 nM 6.60
CHEMBL1995813 — Ki = 316.23 nM 6.50
CHEMBL2002726 — Ki = 316.23 nM 6.50
CHEMBL1996817 — Ki = 316.23 nM 6.50
CHEMBL1982711 — Ki = 316.23 nM 6.50
CHEMBL1982957 — Ki = 398.11 nM 6.40
CHEMBL1992634 — Ki = 398.11 nM 6.40
CHEMBL1993661 — Ki = 398.11 nM 6.40
CHEMBL1965836 — Ki = 501.19 nM 6.30
CHEMBL1967887 — Ki = 630.96 nM 6.20
CHEMBL509032 TAE-684 Ki = 794.33 nM 6.10
CHEMBL1975128 — Ki = 794.33 nM 6.10
CHEMBL1975128 — Ki = 794.33 nM 6.10
CHEMBL2000071 — Ki = 1000.0 nM 6.00
CHEMBL2001920 — Ki = 1000.0 nM 6.00
CHEMBL1965131 — Ki = 1000.0 nM 6.00
CHEMBL1969588 — Ki = 1000.0 nM 6.00
CHEMBL1973860 — Ki = 1000.0 nM 6.00
CHEMBL1996979 — Ki = 1000.0 nM 6.00
CHEMBL482767 SNS-314 Ki = 1258.93 nM 5.90
CHEMBL1973142 — Ki = 1258.93 nM 5.90
CHEMBL1974416 — Ki = 1258.93 nM 5.90
CHEMBL2003405 — Ki = 1258.93 nM 5.90
CHEMBL1991078 — Ki = 1258.93 nM 5.90
CHEMBL1990885 — Ki = 1258.93 nM 5.90
CHEMBL1966425 — Ki = 1258.93 nM 5.90
CHEMBL1988173 — Ki = 1584.89 nM 5.80
CHEMBL1997764 — Ki = 1584.89 nM 5.80
CHEMBL1982924 — Ki = 1584.89 nM 5.80
CHEMBL2001646 — Ki = 1584.89 nM 5.80
CHEMBL246970 — Ki = 1584.89 nM 5.80
CHEMBL2006439 — Ki = 1584.89 nM 5.80
CHEMBL1992922 — Ki = 1584.89 nM 5.80
CHEMBL1978448 — Ki = 1584.89 nM 5.80
CHEMBL1974803 — Ki = 1584.89 nM 5.80
CHEMBL1966343 — Ki = 1584.89 nM 5.80
CHEMBL1993424 — Ki = 1584.89 nM 5.80
CHEMBL1988163 — Ki = 1995.26 nM 5.70
CHEMBL1972158 — Ki = 1995.26 nM 5.70
CHEMBL1986499 — Ki = 1995.26 nM 5.70