Assay Detail
Functional
CHEMBL1963971
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PubChem BioAssay. Dose response confirmation of uHTS antagonist hits from Gli-SUFU in a luminescent reporter assay. (Class of assay: confirmatory)
344
Total Activities
344
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 344 | 5.25 | 6.53 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1393367 | — | — | 1 | 6.53 |
| CHEMBL1543258 | — | — | 1 | 6.43 |
| CHEMBL1438842 | — | — | 1 | 6.42 |
| CHEMBL1336211 | — | — | 1 | 6.38 |
| CHEMBL1509493 | — | — | 1 | 6.27 |
| CHEMBL1581759 | — | — | 1 | 6.21 |
| CHEMBL1463207 | — | — | 1 | 6.19 |
| CHEMBL1452840 | — | — | 1 | 6.18 |
| CHEMBL1704304 | — | — | 1 | 6.18 |
| CHEMBL1553781 | — | — | 1 | 6.13 |
| CHEMBL1534358 | — | — | 1 | 6.11 |
| CHEMBL1401057 | — | — | 1 | 6.05 |
| CHEMBL1523428 | — | — | 1 | 6.03 |
| CHEMBL1507347 | — | — | 1 | 6.02 |
| CHEMBL1713017 | — | — | 1 | 5.99 |
| CHEMBL1386479 | — | — | 1 | 5.99 |
| CHEMBL1300193 | — | — | 1 | 5.97 |
| CHEMBL1976317 | — | — | 1 | 5.95 |
| CHEMBL1310132 | — | — | 1 | 5.90 |
| CHEMBL1714938 | — | — | 1 | 5.89 |
| CHEMBL1542594 | — | — | 1 | 5.88 |
| CHEMBL1410925 | — | — | 1 | 5.83 |
| CHEMBL1387401 | — | — | 1 | 5.82 |
| CHEMBL2003587 | — | — | 1 | 5.82 |
| CHEMBL56170 | — | — | 1 | 5.80 |
| CHEMBL1706173 | — | — | 1 | 5.80 |
| CHEMBL1457690 | — | — | 1 | 5.75 |
| CHEMBL1379608 | — | — | 1 | 5.71 |
| CHEMBL1497797 | — | — | 1 | 5.70 |
| CHEMBL1573186 | — | — | 1 | 5.70 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1393367 | — | IC50 | = | 294.0 | nM | 6.53 |
| CHEMBL1543258 | — | IC50 | = | 368.0 | nM | 6.43 |
| CHEMBL1438842 | — | IC50 | = | 377.0 | nM | 6.42 |
| CHEMBL1336211 | — | IC50 | = | 421.0 | nM | 6.38 |
| CHEMBL1509493 | — | IC50 | = | 535.0 | nM | 6.27 |
| CHEMBL1581759 | — | IC50 | = | 619.0 | nM | 6.21 |
| CHEMBL1463207 | — | IC50 | = | 647.0 | nM | 6.19 |
| CHEMBL1452840 | — | IC50 | = | 663.0 | nM | 6.18 |
| CHEMBL1704304 | — | IC50 | = | 666.0 | nM | 6.18 |
| CHEMBL1553781 | — | IC50 | = | 735.0 | nM | 6.13 |
| CHEMBL1534358 | — | IC50 | = | 771.0 | nM | 6.11 |
| CHEMBL1401057 | — | IC50 | = | 887.0 | nM | 6.05 |
| CHEMBL1523428 | — | IC50 | = | 940.0 | nM | 6.03 |
| CHEMBL1507347 | — | IC50 | = | 954.0 | nM | 6.02 |
| CHEMBL1713017 | — | IC50 | = | 1020.0 | nM | 5.99 |
| CHEMBL1386479 | — | IC50 | = | 1020.0 | nM | 5.99 |
| CHEMBL1300193 | — | IC50 | = | 1060.0 | nM | 5.97 |
| CHEMBL1976317 | — | IC50 | = | 1120.0 | nM | 5.95 |
| CHEMBL1310132 | — | IC50 | = | 1260.0 | nM | 5.90 |
| CHEMBL1714938 | — | IC50 | = | 1280.0 | nM | 5.89 |
| CHEMBL1542594 | — | IC50 | = | 1320.0 | nM | 5.88 |
| CHEMBL1410925 | — | IC50 | = | 1470.0 | nM | 5.83 |
| CHEMBL1387401 | — | IC50 | = | 1530.0 | nM | 5.82 |
| CHEMBL2003587 | — | IC50 | = | 1510.0 | nM | 5.82 |
| CHEMBL1706173 | — | IC50 | = | 1600.0 | nM | 5.80 |
| CHEMBL56170 | — | IC50 | = | 1570.0 | nM | 5.80 |
| CHEMBL1457690 | — | IC50 | = | 1780.0 | nM | 5.75 |
| CHEMBL1379608 | — | IC50 | = | 1960.0 | nM | 5.71 |
| CHEMBL1423564 | — | IC50 | = | 1980.0 | nM | 5.70 |
| CHEMBL1497797 | — | IC50 | = | 2020.0 | nM | 5.70 |
| CHEMBL1573186 | — | IC50 | = | 1990.0 | nM | 5.70 |
| CHEMBL1423708 | — | IC50 | = | 2060.0 | nM | 5.69 |
| CHEMBL1705113 | — | IC50 | = | 2120.0 | nM | 5.67 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 2230.0 | nM | 5.65 |
| CHEMBL1429289 | — | IC50 | = | 2220.0 | nM | 5.65 |
| CHEMBL1494441 | — | IC50 | = | 2290.0 | nM | 5.64 |
| CHEMBL1412273 | — | IC50 | = | 2280.0 | nM | 5.64 |
| CHEMBL1394105 | — | IC50 | = | 2440.0 | nM | 5.61 |
| CHEMBL1571603 | — | IC50 | = | 2510.0 | nM | 5.60 |
| CHEMBL1500404 | — | IC50 | = | 2520.0 | nM | 5.60 |
| CHEMBL1530686 | — | IC50 | = | 2720.0 | nM | 5.57 |
| CHEMBL1304383 | — | IC50 | = | 2750.0 | nM | 5.56 |
| CHEMBL1425183 | — | IC50 | = | 2790.0 | nM | 5.55 |
| CHEMBL1712863 | PIRITREXIM ISETHIONATE | IC50 | = | 2800.0 | nM | 5.55 |
| CHEMBL1495292 | — | IC50 | = | 2790.0 | nM | 5.55 |
| CHEMBL1371706 | — | IC50 | = | 2900.0 | nM | 5.54 |
| CHEMBL1441701 | — | IC50 | = | 2930.0 | nM | 5.53 |
| CHEMBL1203698 | — | IC50 | = | 3020.0 | nM | 5.52 |
| CHEMBL1360505 | — | IC50 | = | 3010.0 | nM | 5.52 |
| CHEMBL1993889 | — | IC50 | = | 3110.0 | nM | 5.51 |