Assay Detail
Functional
CHEMBL3562130
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PubChem BioAssay. GSK3B-pretreated HCT116 viability from Cell TiterGlo-IC50. (Class of assay: confirmatory)
184
Total Activities
183
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 184 | 6.48 | 9.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL34259 | METHOTREXATE | 4.0 | 1 | 9.00 |
| CHEMBL232201 | BENZIODARONE | 4.0 | 1 | 9.00 |
| CHEMBL917 | FLOXURIDINE | 4.0 | 1 | 9.00 |
| CHEMBL1417019 | MITOXANTRONE HYDROCHLORIDE | 4.0 | 1 | 9.00 |
| CHEMBL378544 | VINBLASTINE SULFATE | 4.0 | 2 | 9.00 |
| CHEMBL1750 | CLOFARABINE | 4.0 | 1 | 9.00 |
| CHEMBL3182961 | — | — | 1 | 9.00 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 9.00 |
| CHEMBL50588 | EMETINE | 4.0 | 1 | 9.00 |
| CHEMBL290106 | BITHIONOL | 4.0 | 1 | 9.00 |
| CHEMBL24944 | TRIBROMSALAN | 4.0 | 1 | 9.00 |
| CHEMBL42442 | OXFENDAZOLE | 2.0 | 1 | 9.00 |
| CHEMBL1607 | TOPOTECAN HYDROCHLORIDE | 4.0 | 1 | 8.84 |
| CHEMBL451887 | CARFILZOMIB | 4.0 | 1 | 8.76 |
| CHEMBL140144 | — | — | 1 | 8.64 |
| CHEMBL3559830 | — | — | 1 | 8.62 |
| CHEMBL1448 | NICLOSAMIDE | 4.0 | 1 | 8.53 |
| CHEMBL1981438 | CLOFLUCARBAN | 2.0 | 1 | 8.52 |
| CHEMBL37161 | FENBENDAZOLE | 2.0 | 1 | 8.52 |
| CHEMBL2358886 | — | — | 1 | 8.41 |
| CHEMBL81782 | — | — | 1 | 8.06 |
| CHEMBL1545634 | — | — | 1 | 8.01 |
| CHEMBL2361697 | — | — | 1 | 7.70 |
| CHEMBL2360738 | — | — | 1 | 7.62 |
| CHEMBL1200596 | CHLOROXINE | 4.0 | 1 | 7.41 |
| CHEMBL2218894 | FLUVASTATIN SODIUM | 4.0 | 1 | 7.40 |
| CHEMBL1456 | MYCOPHENOLATE MOFETIL | 4.0 | 1 | 7.30 |
| CHEMBL1200563 | CERIVASTATIN SODIUM | 4.0 | 1 | 7.28 |
| CHEMBL3185933 | IODOPHTHALEIN SODIUM | 2.0 | 1 | 7.27 |
| CHEMBL178 | DAUNORUBICIN | 4.0 | 1 | 7.26 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1750 | CLOFARABINE | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL42442 | OXFENDAZOLE | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL232201 | BENZIODARONE | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL378544 | VINBLASTINE SULFATE | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL50588 | EMETINE | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL290106 | BITHIONOL | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL917 | FLOXURIDINE | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL1417019 | MITOXANTRONE HYDROCHLORIDE | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL378544 | VINBLASTINE SULFATE | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL3182961 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL24944 | TRIBROMSALAN | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL1607 | TOPOTECAN HYDROCHLORIDE | IC50 | = | 1.44 | nM | 8.84 |
| CHEMBL451887 | CARFILZOMIB | IC50 | = | 1.73 | nM | 8.76 |
| CHEMBL140144 | — | IC50 | = | 2.3 | nM | 8.64 |
| CHEMBL3559830 | — | IC50 | = | 2.41 | nM | 8.62 |
| CHEMBL1448 | NICLOSAMIDE | IC50 | = | 2.95 | nM | 8.53 |
| CHEMBL37161 | FENBENDAZOLE | IC50 | = | 3.0 | nM | 8.52 |
| CHEMBL1981438 | CLOFLUCARBAN | IC50 | = | 3.0 | nM | 8.52 |
| CHEMBL2358886 | — | IC50 | = | 3.92 | nM | 8.41 |
| CHEMBL81782 | — | IC50 | = | 8.75 | nM | 8.06 |
| CHEMBL1545634 | — | IC50 | = | 9.83 | nM | 8.01 |
| CHEMBL2361697 | — | IC50 | = | 19.79 | nM | 7.70 |
| CHEMBL2360738 | — | IC50 | = | 23.7 | nM | 7.62 |
| CHEMBL1200596 | CHLOROXINE | IC50 | = | 39.34 | nM | 7.41 |
| CHEMBL2218894 | FLUVASTATIN SODIUM | IC50 | = | 39.88 | nM | 7.40 |
| CHEMBL1456 | MYCOPHENOLATE MOFETIL | IC50 | = | 49.8 | nM | 7.30 |
| CHEMBL1200563 | CERIVASTATIN SODIUM | IC50 | = | 52.91 | nM | 7.28 |
| CHEMBL3185933 | IODOPHTHALEIN SODIUM | IC50 | = | 54.0 | nM | 7.27 |
| CHEMBL178 | DAUNORUBICIN | IC50 | = | 55.38 | nM | 7.26 |
| CHEMBL1320139 | HELIOMYCIN | IC50 | = | 57.35 | nM | 7.24 |
| CHEMBL264373 | METOPRINE | IC50 | = | 58.88 | nM | 7.23 |
| CHEMBL329522 | EXIFONE | IC50 | = | 69.11 | nM | 7.16 |
| CHEMBL254077 | — | IC50 | = | 141.18 | nM | 6.85 |
| CHEMBL473535 | FENTICLOR | IC50 | = | 147.76 | nM | 6.83 |
| CHEMBL1788401 | CYCLOBENDAZOLE | IC50 | = | 154.7 | nM | 6.81 |
| CHEMBL1483 | ALBENDAZOLE | IC50 | = | 157.93 | nM | 6.80 |
| CHEMBL727 | THIOGUANINE | IC50 | = | 163.26 | nM | 6.79 |
| CHEMBL452867 | RIBOPRINE | IC50 | = | 180.01 | nM | 6.75 |
| CHEMBL223448 | BROXYQUINOLINE | IC50 | = | 183.33 | nM | 6.74 |
| CHEMBL2359490 | — | IC50 | = | 187.64 | nM | 6.73 |
| CHEMBL550348 | DEFERASIROX | IC50 | = | 242.3 | nM | 6.62 |
| CHEMBL1324 | TOLCAPONE | IC50 | = | 264.97 | nM | 6.58 |
| CHEMBL1315136 | TIBROFAN | IC50 | = | 342.3 | nM | 6.47 |
| CHEMBL2355158 | — | IC50 | = | 344.2 | nM | 6.46 |
| CHEMBL1076347 | TRICLOCARBAN | IC50 | = | 362.24 | nM | 6.44 |
| CHEMBL1454910 | NITROXOLINE | IC50 | = | 375.09 | nM | 6.43 |
| CHEMBL242580 | CICLOPIROX OLAMINE | IC50 | = | 389.82 | nM | 6.41 |
| CHEMBL554041 | ALEXIDINE DIHYDROCHLORIDE | IC50 | = | 396.3 | nM | 6.40 |