Assay Detail
Functional
CHEMBL5520188
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Cytostatic activity against human CoC1 cells after 24 hrs by CCK-8 assay
10
Total Activities
10
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | CoC1 |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Three Rounds of Stability-Guided Optimization and Systematical Evaluation of Oncolytic Peptide LTX-315.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 10 | 4.79 | 4.93 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5555708 | — | — | 1 | 4.93 |
| CHEMBL5561453 | — | — | 1 | 4.90 |
| CHEMBL5555594 | — | — | 1 | 4.88 |
| CHEMBL5556048 | — | — | 1 | 4.80 |
| CHEMBL5559375 | — | — | 1 | 4.73 |
| CHEMBL5564867 | — | — | 1 | 4.72 |
| CHEMBL5561051 | — | — | 1 | 4.72 |
| CHEMBL4297628 | RUXOTEMITIDE | 2.0 | 1 | 4.65 |
| CHEMBL5566008 | — | — | 1 | - |
| CHEMBL5549764 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5555708 | — | IC50 | = | 11700.0 | nM | 4.93 |
| CHEMBL5561453 | — | IC50 | = | 12600.0 | nM | 4.90 |
| CHEMBL5555594 | — | IC50 | = | 13300.0 | nM | 4.88 |
| CHEMBL5556048 | — | IC50 | = | 15700.0 | nM | 4.80 |
| CHEMBL5559375 | — | IC50 | = | 18700.0 | nM | 4.73 |
| CHEMBL5564867 | — | IC50 | = | 18900.0 | nM | 4.72 |
| CHEMBL5561051 | — | IC50 | = | 18900.0 | nM | 4.72 |
| CHEMBL4297628 | RUXOTEMITIDE | IC50 | = | 22300.0 | nM | 4.65 |
| CHEMBL5566008 | — | IC50 | = | 136600.0 | nM | - |
| CHEMBL5549764 | — | IC50 | = | 105200.0 | nM | - |