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Compound Detail

CHEMBL2359093

ROSE BENGAL SODIUM
🧪 Phase II
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🧪 Phase II
O=C([O-])c1c(Cl)c(Cl)c(Cl)c(Cl)c1-c1c2cc(I)c(=O)c(I)c-2oc2c(I)c([O-])c(I)cc12.[Na+].[Na+]

Basic Information

ChEMBL ID CHEMBL2359093
Name ROSE BENGAL SODIUM
Phase Phase II
Structure Type MOL
InChI Key UWBXIFCTIZXXLS-UHFFFAOYSA-L
Parent Compound CHEMBL1208422
Active Moiety CHEMBL1208422

Known Names

Acid red 94 Aka105(1) Bengal rose b sodium salt Japan red 105-1 Red no. 105-1 Rose bengal disodium Rose bengal disodium salt Rose bengal extra Rose bengal sodium Rose bengal sodium salt Rose bengale sodique Rose de bengala de sodio
8
Targets
17
Activities
2
Assay Types
0
PK Parameters
20
Publications
12
Known Names

Molecular Properties

973.7
MW (Da)
9.00
ALogP
4
HBA
2
HBD
87.7
PSA (Ų)
0.09
QED
2
Ro5 Violations
2
Rot. Bonds

Drug Information

Molecule Type Small molecule
Chirality Achiral

Flags

Natural Product

Extended Properties

Molecular Formula C20H2Cl4I4Na2O5
MW 1017.64
Aromatic Rings 2
Heavy Atoms 33
NP-Likeness 0.29

ATC Classification

S01JA02
rose bengal sodium
Level 1: SENSORY ORGANS
Level 2: OPHTHALMOLOGICALS

Activity Summary

IC50 16 meas. best 8.1
Ki 1 meas. best 7.72

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Vesicular stomatitis virus
CHEMBL613739
IC50 8.1 8.1 8.0 1
Unchecked
CHEMBL612545
IC50 7.72 5.3017 19.0 6
Unchecked
CHEMBL612545
Ki 7.72 7.72 19.0 1
Human immunodeficiency virus
CHEMBL613758
IC50 7.3 7.3 50.0 1
unidentified influenza virus
CHEMBL613128
IC50 6.52 6.52 300.0 1
Protein translocase subunit SecA 1
CHEMBL3832949
IC50 6.3 6.15 500.0 2
Protein translocase subunit SecA 2
CHEMBL3832955
IC50 5.7 5.7 2000.0 1
Vesicular acetylcholine transporter
CHEMBL2125
IC50 5.01 5.01 9700.0 1
Fibroblast
CHEMBL613838
IC50 4.14 4.13 73000.0 2

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Vesicular stomatitis virus IC50 = 8.0 nM 8.1 Antiviral activity against Vesicular stomatitis virus 33310284
Unchecked IC50 = 19.0 nM 7.72 Inhibition of VGLUT in rat synaptic vesicles assessed as [3H]glutamate uptake pr... 20708942
Unchecked Ki = 19.0 nM 7.72 Inhibition of VGLUT 20708942
Human immunodeficiency virus IC50 = 50.0 nM 7.3 Antiviral activity against Human immunodeficiency virus 33310284
Unchecked IC50 = 64.0 nM 7.19 Inhibition of VMAT in rat synaptic vesicles assessed as [3H]HT uptake pretreated... 20708942
unidentified influenza virus IC50 = 300.0 nM 6.52 Antiviral activity against influenza virus 33310284
Protein translocase subunit SecA 1 IC50 = 500.0 nM 6.3 Inhibition of Staphylococcus aureus ATCC 35556 SecA1 liposomal ion channel activ... 26432604
Protein translocase subunit SecA 1 IC50 = 1000.0 nM 6.0 Inhibition of Staphylococcus aureus ATCC 35556 SecA1 expressed in Escherichia co... 26432604
Protein translocase subunit SecA 2 IC50 = 2000.0 nM 5.7 Inhibition of Staphylococcus aureus ATCC 35556 SecA2 expressed in Escherichia co... 26432604
Vesicular acetylcholine transporter IC50 = 9700.0 nM 5.01 Inhibition of VACHT in rat synaptic vesicles assessed as [3H]HT uptake pretreate... 20708942
Unchecked IC50 = 45000.0 nM 4.35 Cytotoxicity against ewing sarcoma cells (unknown origin) 33310284
Unchecked IC50 = 51000.0 nM 4.29 Cytotoxicity against rhabdomyosarcoma cells (unknown origin) 33310284
Unchecked IC50 = 73000.0 nM 4.14 Cytotoxicity against neuroblastoma cells (unknown origin) 33310284
Fibroblast IC50 = 73000.0 nM 4.14 Cytotoxicity against normal foreskin fibroblast cells (unknown origin) 33310284
Unchecked IC50 = 75000.0 nM 4.12 Cytotoxicity against osteosarcoma cells (unknown origin) 33310284
Fibroblast IC50 = 75000.0 nM 4.12 Cytotoxicity against normal lung fibroblast cells (unknown origin) 33310284

Literature References

Data from ChEMBL 36 via Core Engine