Assay Detail
Functional
CHEMBL1614229
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: A Cell Based Assay for the Identification of Lead Compounds with Inhibitory Activity against HIV-1 Fusion (CCR5 Tropic HIV-1 Fusion Inhibition Assay) - Dose Response. (Class of assay: confirmatory)
89
Total Activities
89
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 89 | 4.80 | 6.01 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL496 | HEXACHLOROPHENE | 4.0 | 1 | 6.01 |
| CHEMBL1602800 | — | — | 1 | 5.70 |
| CHEMBL1329925 | — | — | 1 | 5.66 |
| CHEMBL3199742 | — | — | 1 | 5.52 |
| CHEMBL1498887 | — | — | 1 | 5.52 |
| CHEMBL1583537 | — | — | 1 | 5.47 |
| CHEMBL3198976 | — | — | 1 | 5.44 |
| CHEMBL1309484 | — | — | 1 | 5.37 |
| CHEMBL1543779 | — | — | 1 | 5.36 |
| CHEMBL1492305 | — | — | 1 | 5.35 |
| CHEMBL3194804 | — | — | 1 | 5.35 |
| CHEMBL223453 | — | — | 1 | 5.32 |
| CHEMBL3196762 | — | — | 1 | 5.32 |
| CHEMBL1303580 | — | — | 1 | 5.24 |
| CHEMBL1482585 | — | — | 1 | 5.22 |
| CHEMBL1430309 | — | — | 1 | 5.15 |
| CHEMBL3195965 | — | — | 1 | 5.15 |
| CHEMBL287542 | RAFOXANIDE | 2.0 | 1 | 5.13 |
| CHEMBL1417710 | — | — | 1 | 5.05 |
| CHEMBL3199737 | — | — | 1 | 5.01 |
| CHEMBL1392551 | — | — | 1 | 5.00 |
| CHEMBL1367952 | — | — | 1 | 5.00 |
| CHEMBL1605668 | — | — | 1 | 5.00 |
| CHEMBL1471907 | — | — | 1 | 4.99 |
| CHEMBL3190829 | — | — | 1 | 4.96 |
| CHEMBL1422763 | — | — | 1 | 4.96 |
| CHEMBL1400449 | — | — | 1 | 4.93 |
| CHEMBL1362734 | — | — | 1 | 4.92 |
| CHEMBL1515202 | — | — | 1 | 4.91 |
| CHEMBL1605235 | — | — | 1 | 4.79 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL496 | HEXACHLOROPHENE | IC50 | = | 970.0 | nM | 6.01 |
| CHEMBL1602800 | — | IC50 | = | 2000.0 | nM | 5.70 |
| CHEMBL1329925 | — | IC50 | = | 2170.0 | nM | 5.66 |
| CHEMBL3199742 | — | IC50 | = | 3030.0 | nM | 5.52 |
| CHEMBL1498887 | — | IC50 | = | 3030.0 | nM | 5.52 |
| CHEMBL1583537 | — | IC50 | = | 3410.0 | nM | 5.47 |
| CHEMBL3198976 | — | IC50 | = | 3610.0 | nM | 5.44 |
| CHEMBL1309484 | — | IC50 | = | 4250.0 | nM | 5.37 |
| CHEMBL1543779 | — | IC50 | = | 4410.0 | nM | 5.36 |
| CHEMBL1492305 | — | IC50 | = | 4430.0 | nM | 5.35 |
| CHEMBL3194804 | — | IC50 | = | 4450.0 | nM | 5.35 |
| CHEMBL223453 | — | IC50 | = | 4770.0 | nM | 5.32 |
| CHEMBL3196762 | — | IC50 | = | 4760.0 | nM | 5.32 |
| CHEMBL1303580 | — | IC50 | = | 5700.0 | nM | 5.24 |
| CHEMBL1482585 | — | IC50 | = | 6030.0 | nM | 5.22 |
| CHEMBL1430309 | — | IC50 | = | 7080.0 | nM | 5.15 |
| CHEMBL3195965 | — | IC50 | = | 7020.0 | nM | 5.15 |
| CHEMBL287542 | RAFOXANIDE | IC50 | = | 7360.0 | nM | 5.13 |
| CHEMBL1417710 | — | IC50 | = | 8820.0 | nM | 5.05 |
| CHEMBL3199737 | — | IC50 | = | 9870.0 | nM | 5.01 |
| CHEMBL1392551 | — | IC50 | = | 9920.0 | nM | 5.00 |
| CHEMBL1367952 | — | IC50 | = | 10090.0 | nM | 5.00 |
| CHEMBL1605668 | — | IC50 | = | 9890.0 | nM | 5.00 |
| CHEMBL1471907 | — | IC50 | = | 10260.0 | nM | 4.99 |
| CHEMBL1422763 | — | IC50 | = | 11080.0 | nM | 4.96 |
| CHEMBL3190829 | — | IC50 | = | 11020.0 | nM | 4.96 |
| CHEMBL1400449 | — | IC50 | = | 11670.0 | nM | 4.93 |
| CHEMBL1362734 | — | IC50 | = | 11920.0 | nM | 4.92 |
| CHEMBL1515202 | — | IC50 | = | 12210.0 | nM | 4.91 |
| CHEMBL1605235 | — | IC50 | = | 16280.0 | nM | 4.79 |
| CHEMBL1366367 | — | IC50 | = | 16510.0 | nM | 4.78 |
| CHEMBL1699206 | — | IC50 | = | 17000.0 | nM | 4.77 |
| CHEMBL1533561 | — | IC50 | = | 17440.0 | nM | 4.76 |
| CHEMBL1422601 | — | IC50 | = | 18810.0 | nM | 4.73 |
| CHEMBL1390211 | — | IC50 | = | 18670.0 | nM | 4.73 |
| CHEMBL1485064 | — | IC50 | = | 19570.0 | nM | 4.71 |
| CHEMBL1545384 | — | IC50 | = | 20680.0 | nM | 4.68 |
| CHEMBL1503209 | — | IC50 | = | 21660.0 | nM | 4.66 |
| CHEMBL1384843 | — | IC50 | = | 22700.0 | nM | 4.64 |
| CHEMBL3198341 | — | IC50 | = | 23640.0 | nM | 4.63 |
| CHEMBL1985327 | — | IC50 | = | 25050.0 | nM | 4.60 |
| CHEMBL1381868 | — | IC50 | = | 27060.0 | nM | 4.57 |
| CHEMBL1608106 | — | IC50 | = | 27820.0 | nM | 4.56 |
| CHEMBL1555218 | — | IC50 | = | 28510.0 | nM | 4.54 |
| CHEMBL1527520 | — | IC50 | = | 29370.0 | nM | 4.53 |
| CHEMBL1379894 | — | IC50 | = | 29940.0 | nM | 4.52 |
| CHEMBL1595563 | — | IC50 | = | 30070.0 | nM | 4.52 |
| CHEMBL1971033 | — | IC50 | = | 31720.0 | nM | 4.50 |
| CHEMBL1528476 | — | IC50 | = | 33720.0 | nM | 4.47 |
| CHEMBL3194119 | — | IC50 | = | 35240.0 | nM | 4.45 |