Assay Detail
Functional
CHEMBL1794445
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Fluorescence polarization-based cell-based high throughput dose response assay to identify activators of insulin-degrading enzyme (IDE). (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID493087, AID493124, AID588681]
231
Total Activities
231
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 231 | 4.90 | 6.05 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1568474 | — | — | 1 | 6.05 |
| CHEMBL857 | BIOTIN | 4.0 | 1 | 5.62 |
| CHEMBL1705738 | — | — | 1 | 5.50 |
| CHEMBL1984581 | — | — | 1 | 5.26 |
| CHEMBL1514790 | — | — | 1 | 5.19 |
| CHEMBL1481849 | — | — | 1 | 5.18 |
| CHEMBL1464261 | — | — | 1 | 5.16 |
| CHEMBL1491847 | — | — | 1 | 5.15 |
| CHEMBL1458111 | — | — | 1 | 5.13 |
| CHEMBL1513972 | — | — | 1 | 5.12 |
| CHEMBL1232381 | — | — | 1 | 5.11 |
| CHEMBL1574420 | — | — | 1 | 5.10 |
| CHEMBL1578670 | — | — | 1 | 5.05 |
| CHEMBL250711 | OLEOYL DOPAMINE | — | 1 | 5.05 |
| CHEMBL1500686 | — | — | 1 | 5.03 |
| CHEMBL1322645 | — | — | 1 | 5.01 |
| CHEMBL1369287 | — | — | 1 | 5.00 |
| CHEMBL1455530 | — | — | 1 | 4.96 |
| CHEMBL1497597 | — | — | 1 | 4.95 |
| CHEMBL1527972 | — | — | 1 | 4.95 |
| CHEMBL1403262 | — | — | 1 | 4.91 |
| CHEMBL3189224 | — | — | 1 | 4.86 |
| CHEMBL1309448 | — | — | 1 | 4.84 |
| CHEMBL1605224 | — | — | 1 | 4.82 |
| CHEMBL1460004 | — | — | 1 | 4.81 |
| CHEMBL532160 | — | — | 1 | 4.81 |
| CHEMBL1393761 | — | — | 1 | 4.80 |
| CHEMBL3191688 | — | — | 1 | 4.78 |
| CHEMBL1474759 | — | — | 1 | 4.75 |
| CHEMBL1558968 | — | — | 1 | 4.70 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1568474 | — | EC50 | = | 891.5 | nM | 6.05 |
| CHEMBL857 | BIOTIN | EC50 | = | 2373.0 | nM | 5.62 |
| CHEMBL1705738 | — | EC50 | = | 3160.0 | nM | 5.50 |
| CHEMBL1984581 | — | EC50 | = | 5519.0 | nM | 5.26 |
| CHEMBL1514790 | — | EC50 | = | 6410.0 | nM | 5.19 |
| CHEMBL1481849 | — | EC50 | = | 6621.0 | nM | 5.18 |
| CHEMBL1464261 | — | EC50 | = | 6954.0 | nM | 5.16 |
| CHEMBL1491847 | — | EC50 | = | 7021.0 | nM | 5.15 |
| CHEMBL1458111 | — | EC50 | = | 7379.0 | nM | 5.13 |
| CHEMBL1513972 | — | EC50 | = | 7520.0 | nM | 5.12 |
| CHEMBL1232381 | — | EC50 | = | 7797.0 | nM | 5.11 |
| CHEMBL1574420 | — | EC50 | = | 7992.0 | nM | 5.10 |
| CHEMBL1578670 | — | EC50 | = | 8801.0 | nM | 5.05 |
| CHEMBL250711 | OLEOYL DOPAMINE | EC50 | = | 8943.0 | nM | 5.05 |
| CHEMBL1500686 | — | EC50 | = | 9391.0 | nM | 5.03 |
| CHEMBL1322645 | — | EC50 | = | 9709.0 | nM | 5.01 |
| CHEMBL1369287 | — | EC50 | = | 9931.0 | nM | 5.00 |
| CHEMBL1455530 | — | EC50 | = | 11082.0 | nM | 4.96 |
| CHEMBL1497597 | — | EC50 | = | 11177.0 | nM | 4.95 |
| CHEMBL1527972 | — | EC50 | = | 11125.0 | nM | 4.95 |
| CHEMBL1403262 | — | EC50 | = | 12176.0 | nM | 4.91 |
| CHEMBL3189224 | — | EC50 | = | 13879.0 | nM | 4.86 |
| CHEMBL1309448 | — | EC50 | = | 14344.0 | nM | 4.84 |
| CHEMBL1605224 | — | EC50 | = | 15106.0 | nM | 4.82 |
| CHEMBL1460004 | — | EC50 | = | 15541.0 | nM | 4.81 |
| CHEMBL532160 | — | EC50 | = | 15475.0 | nM | 4.81 |
| CHEMBL1393761 | — | EC50 | = | 15884.0 | nM | 4.80 |
| CHEMBL3191688 | — | EC50 | = | 16644.0 | nM | 4.78 |
| CHEMBL1474759 | — | EC50 | = | 17571.0 | nM | 4.75 |
| CHEMBL1558968 | — | EC50 | = | 20119.0 | nM | 4.70 |
| CHEMBL1504972 | — | EC50 | = | 20750.0 | nM | 4.68 |
| CHEMBL1591898 | — | EC50 | = | 22031.0 | nM | 4.66 |
| CHEMBL1530087 | — | EC50 | = | 21750.0 | nM | 4.66 |
| CHEMBL1442125 | — | EC50 | = | 22311.0 | nM | 4.65 |
| CHEMBL1542526 | — | EC50 | = | 22815.0 | nM | 4.64 |
| CHEMBL1388543 | — | EC50 | = | 23152.0 | nM | 4.63 |
| CHEMBL1526165 | — | EC50 | = | 25247.0 | nM | 4.60 |
| CHEMBL1485551 | — | EC50 | = | 29467.0 | nM | 4.53 |
| CHEMBL1536835 | — | EC50 | = | 32305.0 | nM | 4.49 |
| CHEMBL496633 | — | EC50 | = | 41004.0 | nM | 4.39 |
| CHEMBL1376516 | — | EC50 | = | 42517.0 | nM | 4.37 |
| CHEMBL1576059 | — | EC50 | = | 43763.0 | nM | 4.36 |
| CHEMBL1415720 | — | EC50 | = | 54495.0 | nM | 4.26 |
| CHEMBL1419164 | — | EC50 | > | 54680.0 | nM | - |
| CHEMBL1982108 | — | EC50 | > | 54705.0 | nM | - |
| CHEMBL1986183 | — | EC50 | > | 2025.0 | nM | - |
| CHEMBL1587031 | — | EC50 | > | 54727.0 | nM | - |
| CHEMBL354349 | EUFLAVINE | EC50 | > | 54727.0 | nM | - |
| CHEMBL1492019 | — | EC50 | > | 54727.0 | nM | - |
| CHEMBL1547938 | — | EC50 | > | 54732.0 | nM | - |