Assay Detail
Functional
CHEMBL1963766
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: EGFR
601
Total Activities
596
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | other |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 601 | 6.57 | 8.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2006715 | — | — | 1 | 8.70 |
| CHEMBL1090360 | — | — | 1 | 8.40 |
| CHEMBL1981725 | — | — | 1 | 8.20 |
| CHEMBL1999749 | — | — | 1 | 8.20 |
| CHEMBL509032 | TAE-684 | — | 1 | 8.00 |
| CHEMBL1991429 | — | — | 1 | 7.80 |
| CHEMBL1999590 | — | — | 1 | 7.70 |
| CHEMBL302449 | GO-6976 | — | 1 | 7.70 |
| CHEMBL1980995 | — | — | 1 | 7.60 |
| CHEMBL1982866 | — | — | 1 | 7.60 |
| CHEMBL1970879 | — | — | 1 | 7.60 |
| CHEMBL458997 | — | — | 1 | 7.50 |
| CHEMBL1090356 | — | — | 1 | 7.50 |
| CHEMBL1997617 | — | — | 1 | 7.50 |
| CHEMBL1682558 | — | — | 1 | 7.40 |
| CHEMBL117697 | — | — | 1 | 7.30 |
| CHEMBL1984191 | — | — | 1 | 7.30 |
| CHEMBL2003657 | — | — | 1 | 7.20 |
| CHEMBL475251 | R-406 | 2.0 | 1 | 7.20 |
| CHEMBL2004419 | — | — | 1 | 7.20 |
| CHEMBL2005886 | — | — | 1 | 7.10 |
| CHEMBL289959 | — | — | 1 | 7.10 |
| CHEMBL1967878 | CENISERTIB | 2.0 | 1 | 7.10 |
| CHEMBL1993661 | — | — | 1 | 7.10 |
| CHEMBL1980163 | — | — | 1 | 7.00 |
| CHEMBL1971029 | — | — | 1 | 7.00 |
| CHEMBL1989474 | — | — | 1 | 6.90 |
| CHEMBL1982992 | — | — | 1 | 6.80 |
| CHEMBL590109 | — | — | 1 | 6.80 |
| CHEMBL363648 | TAK-715 | 2.0 | 1 | 6.70 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2006715 | — | Ki | = | 1.995 | nM | 8.70 |
| CHEMBL1090360 | — | Ki | = | 3.981 | nM | 8.40 |
| CHEMBL1999749 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL1981725 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL509032 | TAE-684 | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL1991429 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1999590 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL302449 | GO-6976 | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1982866 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1980995 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1970879 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1997617 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL1090356 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL458997 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL1682558 | — | Ki | = | 39.81 | nM | 7.40 |
| CHEMBL117697 | — | Ki | = | 50.12 | nM | 7.30 |
| CHEMBL1984191 | — | Ki | = | 50.12 | nM | 7.30 |
| CHEMBL2004419 | — | Ki | = | 63.1 | nM | 7.20 |
| CHEMBL2003657 | — | Ki | = | 63.1 | nM | 7.20 |
| CHEMBL475251 | R-406 | Ki | = | 63.1 | nM | 7.20 |
| CHEMBL2005886 | — | Ki | = | 79.43 | nM | 7.10 |
| CHEMBL1993661 | — | Ki | = | 79.43 | nM | 7.10 |
| CHEMBL1967878 | CENISERTIB | Ki | = | 79.43 | nM | 7.10 |
| CHEMBL289959 | — | Ki | = | 79.43 | nM | 7.10 |
| CHEMBL1980163 | — | Ki | = | 100.0 | nM | 7.00 |
| CHEMBL1971029 | — | Ki | = | 100.0 | nM | 7.00 |
| CHEMBL1989474 | — | Ki | = | 125.89 | nM | 6.90 |
| CHEMBL1982992 | — | Ki | = | 158.49 | nM | 6.80 |
| CHEMBL590109 | — | Ki | = | 158.49 | nM | 6.80 |
| CHEMBL1969588 | — | Ki | = | 199.53 | nM | 6.70 |
| CHEMBL103667 | DORAMAPIMOD | Ki | = | 199.53 | nM | 6.70 |
| CHEMBL306380 | — | Ki | = | 199.53 | nM | 6.70 |
| CHEMBL243088 | — | Ki | = | 199.53 | nM | 6.70 |
| CHEMBL483158 | ALISERTIB | Ki | = | 199.53 | nM | 6.70 |
| CHEMBL363648 | TAK-715 | Ki | = | 199.53 | nM | 6.70 |
| CHEMBL1994938 | — | Ki | = | 199.53 | nM | 6.70 |
| CHEMBL1984162 | — | Ki | = | 199.53 | nM | 6.70 |
| CHEMBL1614705 | — | Ki | = | 199.53 | nM | 6.70 |
| CHEMBL1970522 | — | Ki | = | 199.53 | nM | 6.70 |
| CHEMBL2006778 | — | Ki | = | 251.19 | nM | 6.60 |
| CHEMBL2001239 | — | Ki | = | 251.19 | nM | 6.60 |
| CHEMBL1996066 | — | Ki | = | 251.19 | nM | 6.60 |
| CHEMBL2001751 | — | Ki | = | 251.19 | nM | 6.60 |
| CHEMBL1968380 | — | Ki | = | 251.19 | nM | 6.60 |
| CHEMBL1997623 | — | Ki | = | 251.19 | nM | 6.60 |
| CHEMBL514499 | GW843682X | Ki | = | 251.19 | nM | 6.60 |
| CHEMBL1996979 | — | Ki | = | 251.19 | nM | 6.60 |
| CHEMBL2006276 | — | Ki | = | 251.19 | nM | 6.60 |
| CHEMBL1964692 | — | Ki | = | 316.23 | nM | 6.50 |
| CHEMBL1970317 | — | Ki | = | 316.23 | nM | 6.50 |