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Assay Detail

CHEMBL1963811

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: CAMK1D
ChEMBL ↗
352
Total Activities
342
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Category other
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Calcium/calmodulin-dependent protein kinase type 1D (CHEMBL5073) ↗
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

PubChem BioAssay data set

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 352 5.57 8.40

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1980995 — — 1 8.40
CHEMBL1988581 — — 1 7.30
CHEMBL1980407 — — 1 7.20
CHEMBL2007421 — — 1 6.80
CHEMBL1991078 — — 1 6.60
CHEMBL1988141 — — 1 6.50
CHEMBL509032 TAE-684 — 1 6.40
CHEMBL2002099 — — 2 6.40
CHEMBL1996048 — — 1 6.40
CHEMBL1997193 — — 1 6.40
CHEMBL1978371 — — 1 6.40
CHEMBL1972355 — — 1 6.30
CHEMBL1983111 — — 1 6.30
CHEMBL1973359 — — 1 6.30
CHEMBL1992073 — — 1 6.30
CHEMBL1972346 — — 1 6.30
CHEMBL1991734 — — 1 6.30
CHEMBL1980329 — — 1 6.30
CHEMBL1983980 — — 1 6.30
CHEMBL1992042 — — 1 6.20
CHEMBL2004025 — — 1 6.20
CHEMBL1975923 — — 1 6.20
CHEMBL1978166 — — 2 6.20
CHEMBL379975 — — 1 6.20
CHEMBL1995811 — — 1 6.20
CHEMBL1965351 — — 1 6.10
CHEMBL1966175 — — 1 6.10
CHEMBL1979690 — — 1 6.10
CHEMBL1982413 — — 1 6.10
CHEMBL1993335 — — 1 6.10

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1980995 — Ki = 3.981 nM 8.40
CHEMBL1988581 — Ki = 50.12 nM 7.30
CHEMBL1980407 — Ki = 63.1 nM 7.20
CHEMBL2007421 — Ki = 158.49 nM 6.80
CHEMBL1991078 — Ki = 251.19 nM 6.60
CHEMBL1988141 — Ki = 316.23 nM 6.50
CHEMBL1997193 — Ki = 398.11 nM 6.40
CHEMBL1996048 — Ki = 398.11 nM 6.40
CHEMBL2002099 — Ki = 398.11 nM 6.40
CHEMBL509032 TAE-684 Ki = 398.11 nM 6.40
CHEMBL1978371 — Ki = 398.11 nM 6.40
CHEMBL1972355 — Ki = 501.19 nM 6.30
CHEMBL1980329 — Ki = 501.19 nM 6.30
CHEMBL1991734 — Ki = 501.19 nM 6.30
CHEMBL1983111 — Ki = 501.19 nM 6.30
CHEMBL1992073 — Ki = 501.19 nM 6.30
CHEMBL2002099 — Ki = 501.19 nM 6.30
CHEMBL1973359 — Ki = 501.19 nM 6.30
CHEMBL1983980 — Ki = 501.19 nM 6.30
CHEMBL1972346 — Ki = 501.19 nM 6.30
CHEMBL1978166 — Ki = 630.96 nM 6.20
CHEMBL1992042 — Ki = 630.96 nM 6.20
CHEMBL379975 — Ki = 630.96 nM 6.20
CHEMBL2004025 — Ki = 630.96 nM 6.20
CHEMBL1978166 — Ki = 630.96 nM 6.20
CHEMBL1975923 — Ki = 630.96 nM 6.20
CHEMBL1995811 — Ki = 630.96 nM 6.20
CHEMBL1979690 — Ki = 794.33 nM 6.10
CHEMBL1966175 — Ki = 794.33 nM 6.10
CHEMBL1982413 — Ki = 794.33 nM 6.10
CHEMBL1965351 — Ki = 794.33 nM 6.10
CHEMBL1993335 — Ki = 794.33 nM 6.10
CHEMBL1974480 — Ki = 1000.0 nM 6.00
CHEMBL1980167 — Ki = 1000.0 nM 6.00
CHEMBL1983348 — Ki = 1000.0 nM 6.00
CHEMBL1980297 ILORASERTIB Ki = 1000.0 nM 6.00
CHEMBL2005449 — Ki = 1000.0 nM 6.00
CHEMBL1976196 — Ki = 1000.0 nM 6.00
CHEMBL1421720 — Ki = 1000.0 nM 6.00
CHEMBL1967998 — Ki = 1258.93 nM 5.90
CHEMBL1993374 — Ki = 1258.93 nM 5.90
CHEMBL1972220 — Ki = 1258.93 nM 5.90
CHEMBL2002723 — Ki = 1258.93 nM 5.90
CHEMBL1973013 — Ki = 1258.93 nM 5.90
CHEMBL1982711 — Ki = 1584.89 nM 5.80
CHEMBL1980391 RG-1530 Ki = 1584.89 nM 5.80
CHEMBL2005478 — Ki = 1584.89 nM 5.80
CHEMBL1971227 — Ki = 1584.89 nM 5.80
CHEMBL1977138 — Ki = 1584.89 nM 5.80
CHEMBL565612 SOTRASTAURIN Ki = 1584.89 nM 5.80