Assay Detail
Functional
CHEMBL1963883
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Dose-response secondary confirmation of microRNA-mediated mRNA deacetylation inhibitors by fluorescence polarization assay using Cy5 labeled peptide. (Class of assay: confirmatory)
1186
Total Activities
1186
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1186 | 4.39 | 4.48 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1342622 | — | — | 1 | 4.48 |
| CHEMBL1370330 | — | — | 1 | 4.48 |
| CHEMBL1471090 | — | — | 1 | 4.48 |
| CHEMBL1446983 | — | — | 1 | 4.48 |
| CHEMBL1874130 | — | — | 1 | 4.48 |
| CHEMBL1541254 | — | — | 1 | 4.47 |
| CHEMBL1718610 | — | — | 1 | 4.47 |
| CHEMBL1981093 | — | — | 1 | 4.46 |
| CHEMBL1497838 | — | — | 1 | 4.46 |
| CHEMBL1480605 | — | — | 1 | 4.45 |
| CHEMBL1869639 | — | — | 1 | 4.45 |
| CHEMBL3145283 | — | — | 1 | 4.45 |
| CHEMBL1429797 | — | — | 1 | 4.45 |
| CHEMBL1969088 | — | — | 1 | 4.44 |
| CHEMBL1519796 | — | — | 1 | 4.43 |
| CHEMBL1562280 | — | — | 1 | 4.42 |
| CHEMBL1469144 | — | — | 1 | 4.42 |
| CHEMBL1702548 | — | — | 1 | 4.38 |
| CHEMBL1459684 | — | — | 1 | 4.38 |
| CHEMBL253348 | — | — | 1 | 4.36 |
| CHEMBL1570587 | — | — | 1 | 4.35 |
| CHEMBL1573280 | — | — | 1 | 4.35 |
| CHEMBL1575046 | — | — | 1 | 4.35 |
| CHEMBL1530966 | — | — | 1 | 4.34 |
| CHEMBL1304508 | — | — | 1 | 4.33 |
| CHEMBL1613576 | — | — | 1 | 4.32 |
| CHEMBL1979932 | — | — | 1 | 4.29 |
| CHEMBL426 | — | — | 1 | 4.28 |
| CHEMBL1363719 | — | — | 1 | 4.27 |
| CHEMBL1868523 | — | — | 1 | 4.21 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1471090 | — | IC50 | = | 33400.0 | nM | 4.48 |
| CHEMBL1370330 | — | IC50 | = | 33200.0 | nM | 4.48 |
| CHEMBL1446983 | — | IC50 | = | 33100.0 | nM | 4.48 |
| CHEMBL1874130 | — | IC50 | = | 33100.0 | nM | 4.48 |
| CHEMBL1342622 | — | IC50 | = | 33300.0 | nM | 4.48 |
| CHEMBL1541254 | — | IC50 | = | 34100.0 | nM | 4.47 |
| CHEMBL1718610 | — | IC50 | = | 33500.0 | nM | 4.47 |
| CHEMBL1981093 | — | IC50 | = | 35100.0 | nM | 4.46 |
| CHEMBL1497838 | — | IC50 | = | 35100.0 | nM | 4.46 |
| CHEMBL1480605 | — | IC50 | = | 35700.0 | nM | 4.45 |
| CHEMBL3145283 | — | IC50 | = | 35300.0 | nM | 4.45 |
| CHEMBL1869639 | — | IC50 | = | 35700.0 | nM | 4.45 |
| CHEMBL1429797 | — | IC50 | = | 35200.0 | nM | 4.45 |
| CHEMBL1969088 | — | IC50 | = | 36400.0 | nM | 4.44 |
| CHEMBL1519796 | — | IC50 | = | 37300.0 | nM | 4.43 |
| CHEMBL1562280 | — | IC50 | = | 37900.0 | nM | 4.42 |
| CHEMBL1469144 | — | IC50 | = | 38300.0 | nM | 4.42 |
| CHEMBL1459684 | — | IC50 | = | 41700.0 | nM | 4.38 |
| CHEMBL1702548 | — | IC50 | = | 41400.0 | nM | 4.38 |
| CHEMBL253348 | — | IC50 | = | 43300.0 | nM | 4.36 |
| CHEMBL1573280 | — | IC50 | = | 44800.0 | nM | 4.35 |
| CHEMBL1575046 | — | IC50 | = | 45100.0 | nM | 4.35 |
| CHEMBL1570587 | — | IC50 | = | 44500.0 | nM | 4.35 |
| CHEMBL1530966 | — | IC50 | = | 45800.0 | nM | 4.34 |
| CHEMBL1304508 | — | IC50 | = | 46200.0 | nM | 4.33 |
| CHEMBL1613576 | — | IC50 | = | 48200.0 | nM | 4.32 |
| CHEMBL1979932 | — | IC50 | = | 51200.0 | nM | 4.29 |
| CHEMBL426 | — | IC50 | = | 52100.0 | nM | 4.28 |
| CHEMBL1363719 | — | IC50 | = | 53900.0 | nM | 4.27 |
| CHEMBL1575084 | — | IC50 | = | 62100.0 | nM | 4.21 |
| CHEMBL1868523 | — | IC50 | = | 61600.0 | nM | 4.21 |
| CHEMBL1865656 | — | IC50 | > | 66000.0 | nM | - |
| CHEMBL1506226 | — | IC50 | > | 66000.0 | nM | - |
| CHEMBL1429377 | — | IC50 | > | 66000.0 | nM | - |
| CHEMBL1361913 | — | IC50 | > | 66000.0 | nM | - |
| CHEMBL505209 | — | IC50 | > | 66000.0 | nM | - |
| CHEMBL1497766 | — | IC50 | > | 66000.0 | nM | - |
| CHEMBL1508001 | — | IC50 | > | 66000.0 | nM | - |
| CHEMBL1407756 | — | IC50 | > | 66000.0 | nM | - |
| CHEMBL1876600 | — | IC50 | > | 66000.0 | nM | - |
| CHEMBL1411507 | — | IC50 | > | 66000.0 | nM | - |
| CHEMBL1429408 | — | IC50 | > | 66000.0 | nM | - |
| CHEMBL1566257 | — | IC50 | > | 66000.0 | nM | - |
| CHEMBL1434250 | — | IC50 | > | 66000.0 | nM | - |
| CHEMBL1551103 | — | IC50 | > | 66000.0 | nM | - |
| CHEMBL1498790 | — | IC50 | > | 66000.0 | nM | - |
| CHEMBL1350038 | — | IC50 | > | 66000.0 | nM | - |
| CHEMBL1303188 | — | IC50 | > | 66000.0 | nM | - |
| CHEMBL581225 | — | IC50 | > | 66000.0 | nM | - |
| CHEMBL1422849 | — | IC50 | > | 66000.0 | nM | - |