Assay Detail
Functional
CHEMBL5520189
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Cytostatic activity against human HeLa cells after 24 hrs by CCK-8 assay
19
Total Activities
17
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HeLa |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Three Rounds of Stability-Guided Optimization and Systematical Evaluation of Oncolytic Peptide LTX-315.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 19 | 4.45 | 4.97 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5566800 | — | — | 1 | 4.97 |
| CHEMBL5561652 | — | — | 1 | 4.90 |
| CHEMBL5555895 | — | — | 1 | 4.76 |
| CHEMBL5556816 | — | — | 1 | 4.55 |
| CHEMBL5560630 | — | — | 1 | 4.48 |
| CHEMBL5555708 | — | — | 2 | 4.41 |
| CHEMBL4297628 | RUXOTEMITIDE | 2.0 | 2 | 4.37 |
| CHEMBL5561453 | — | — | 1 | 4.35 |
| CHEMBL5555594 | — | — | 1 | 4.32 |
| CHEMBL5556048 | — | — | 1 | 4.30 |
| CHEMBL5561051 | — | — | 1 | 4.28 |
| CHEMBL5559375 | — | — | 1 | 4.28 |
| CHEMBL5558457 | — | — | 1 | 4.26 |
| CHEMBL5564867 | — | — | 1 | 4.24 |
| CHEMBL5549764 | — | — | 1 | - |
| CHEMBL5566008 | — | — | 1 | - |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5566800 | — | IC50 | = | 10700.0 | nM | 4.97 |
| CHEMBL5561652 | — | IC50 | = | 12600.0 | nM | 4.90 |
| CHEMBL5555895 | — | IC50 | = | 17500.0 | nM | 4.76 |
| CHEMBL5556816 | — | IC50 | = | 28200.0 | nM | 4.55 |
| CHEMBL5560630 | — | IC50 | = | 33400.0 | nM | 4.48 |
| CHEMBL5555708 | — | IC50 | = | 39100.0 | nM | 4.41 |
| CHEMBL4297628 | RUXOTEMITIDE | IC50 | = | 43000.0 | nM | 4.37 |
| CHEMBL5555708 | — | IC50 | = | 44300.0 | nM | 4.35 |
| CHEMBL5561453 | — | IC50 | = | 44300.0 | nM | 4.35 |
| CHEMBL4297628 | RUXOTEMITIDE | IC50 | = | 45800.0 | nM | 4.34 |
| CHEMBL5555594 | — | IC50 | = | 47700.0 | nM | 4.32 |
| CHEMBL5556048 | — | IC50 | = | 50000.0 | nM | 4.30 |
| CHEMBL5561051 | — | IC50 | = | 52700.0 | nM | 4.28 |
| CHEMBL5559375 | — | IC50 | = | 52900.0 | nM | 4.28 |
| CHEMBL5558457 | — | IC50 | = | 54300.0 | nM | 4.26 |
| CHEMBL5564867 | — | IC50 | = | 57000.0 | nM | 4.24 |
| CHEMBL5549764 | — | IC50 | > | 300000.0 | nM | - |
| CHEMBL5566008 | — | IC50 | > | 300000.0 | nM | - |
| CHEMBL65 | CAMPTOTHECIN | IC50 | > | 300000.0 | nM | - |