Assay Detail
Functional
CHEMBL1217012
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Antimicrobial activity against Cryptosporidium parvum
258
Total Activities
258
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Cryptosporidium parvum |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 258 | 5.68 | 6.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL104787 | — | — | 1 | 6.00 |
| CHEMBL323960 | — | — | 1 | 6.00 |
| CHEMBL7586 | — | — | 1 | 6.00 |
| CHEMBL52947 | — | — | 1 | 6.00 |
| CHEMBL1213324 | — | — | 1 | 6.00 |
| CHEMBL1213323 | — | — | 1 | 6.00 |
| CHEMBL1213321 | — | — | 1 | 6.00 |
| CHEMBL1213269 | — | — | 1 | 6.00 |
| CHEMBL1213540 | — | — | 1 | 6.00 |
| CHEMBL1213435 | — | — | 1 | 6.00 |
| CHEMBL1213436 | — | — | 1 | 5.70 |
| CHEMBL1214610 | — | — | 1 | 5.70 |
| CHEMBL322315 | — | — | 1 | 5.70 |
| CHEMBL7535 | — | — | 1 | 5.70 |
| CHEMBL1213683 | — | — | 1 | 5.52 |
| CHEMBL1213585 | — | — | 1 | 5.52 |
| CHEMBL343543 | — | — | 1 | 5.52 |
| CHEMBL22 | TRIMETHOPRIM | 4.0 | 1 | 5.40 |
| CHEMBL1213320 | — | — | 1 | 5.40 |
| CHEMBL1214609 | — | — | 1 | 5.30 |
| CHEMBL6696 | — | — | 1 | 5.05 |
| CHEMBL1213662 | — | — | 1 | 4.52 |
| CHEMBL343382 | — | — | 1 | - |
| CHEMBL88430 | — | — | 1 | - |
| CHEMBL138265 | — | — | 1 | - |
| CHEMBL137942 | — | — | 1 | - |
| CHEMBL138060 | — | — | 1 | - |
| CHEMBL1213493 | — | — | 1 | - |
| CHEMBL1213686 | — | — | 1 | - |
| CHEMBL1213685 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL104787 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL1213540 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL323960 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL7586 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL52947 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL1213324 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL1213323 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL1213321 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL1213269 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL1213435 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL1213436 | — | IC50 | = | 2000.0 | nM | 5.70 |
| CHEMBL7535 | — | IC50 | = | 2000.0 | nM | 5.70 |
| CHEMBL322315 | — | IC50 | = | 2000.0 | nM | 5.70 |
| CHEMBL1214610 | — | IC50 | = | 2000.0 | nM | 5.70 |
| CHEMBL1213585 | — | IC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL1213683 | — | IC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL343543 | — | IC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL1213320 | — | IC50 | = | 4000.0 | nM | 5.40 |
| CHEMBL22 | TRIMETHOPRIM | IC50 | = | 4000.0 | nM | 5.40 |
| CHEMBL1214609 | — | IC50 | = | 5000.0 | nM | 5.30 |
| CHEMBL6696 | — | IC50 | = | 9000.0 | nM | 5.05 |
| CHEMBL1213662 | — | IC50 | = | 30000.0 | nM | 4.52 |
| CHEMBL384467 | DEXAMETHASONE | IC50 | - | — | - | |
| CHEMBL898 | DIFLUNISAL | IC50 | - | — | - | |
| CHEMBL1201353 | DEXCHLORPHENIRAMINE | IC50 | - | — | - | |
| CHEMBL248702 | DEXFENFLURAMINE | IC50 | - | — | - | |
| CHEMBL1213351 | PROPOXYPHENE | IC50 | - | — | - | |
| CHEMBL12 | DIAZEPAM | IC50 | - | — | - | |
| CHEMBL181 | DIAZOXIDE | IC50 | - | — | - | |
| CHEMBL139 | DICLOFENAC | IC50 | - | — | - | |
| CHEMBL23 | DILTIAZEM | IC50 | - | — | - | |
| CHEMBL989 | FLUOCINOLONE ACETONIDE | IC50 | - | — | - | |
| CHEMBL59 | DOPAMINE | IC50 | - | — | - | |
| CHEMBL219916 | DOMPERIDONE | IC50 | - | — | - | |
| CHEMBL1597 | DIMERCAPROL | IC50 | - | — | - | |
| CHEMBL254219 | DIGITOXIN | IC50 | - | — | - | |
| CHEMBL1201891 | DEFLAZACORT | IC50 | - | — | - | |
| CHEMBL509924 | DIFLUCORTOLONE | IC50 | - | — | - | |
| CHEMBL135 | ESTRADIOL | IC50 | - | — | - | |
| CHEMBL1575 | ESTRAMUSTINE | IC50 | - | — | - | |
| CHEMBL456 | ETHACRYNIC ACID | IC50 | - | — | - | |
| CHEMBL1441 | ETHIONAMIDE | IC50 | - | — | - | |
| CHEMBL696 | ETHOSUXIMIDE | IC50 | - | — | - | |
| CHEMBL1213460 | ETHYL LOFLAZEPATE | IC50 | - | — | - | |
| CHEMBL358150 | ETOFIBRATE | IC50 | - | — | - | |
| CHEMBL44657 | ETOPOSIDE | IC50 | - | — | - | |
| CHEMBL1480 | FELODIPINE | IC50 | - | — | - | |
| CHEMBL32800 | FENOTEROL | IC50 | - | — | - | |
| CHEMBL596 | FENTANYL | IC50 | - | — | - | |
| CHEMBL1213420 | DROXICAM | IC50 | - | — | - |