Assay Detail
Functional
CHEMBL5520186
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Cytostatic activity against mouse A20 cells after 24 hrs by CCK-8 assay
20
Total Activities
18
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Mus musculus |
| Cell Type | A20 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Three Rounds of Stability-Guided Optimization and Systematical Evaluation of Oncolytic Peptide LTX-315.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 20 | 4.86 | 5.41 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5566800 | — | — | 1 | 5.41 |
| CHEMBL5561652 | — | — | 1 | 5.39 |
| CHEMBL5555708 | — | — | 2 | 5.19 |
| CHEMBL5555594 | — | — | 1 | 5.19 |
| CHEMBL5561453 | — | — | 1 | 5.01 |
| CHEMBL5560630 | — | — | 1 | 4.97 |
| CHEMBL5555895 | — | — | 1 | 4.95 |
| CHEMBL4297628 | RUXOTEMITIDE | 2.0 | 2 | 4.95 |
| CHEMBL5561211 | — | — | 1 | 4.93 |
| CHEMBL5561051 | — | — | 1 | 4.83 |
| CHEMBL5556048 | — | — | 1 | 4.79 |
| CHEMBL5564867 | — | — | 1 | 4.77 |
| CHEMBL5559375 | — | — | 1 | 4.64 |
| CHEMBL5556816 | — | — | 1 | 4.39 |
| CHEMBL5549764 | — | — | 1 | 4.09 |
| CHEMBL5566008 | — | — | 1 | 4.05 |
| CHEMBL5558457 | — | — | 1 | - |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5566800 | — | IC50 | = | 3900.0 | nM | 5.41 |
| CHEMBL5561652 | — | IC50 | = | 4100.0 | nM | 5.39 |
| CHEMBL5555708 | — | IC50 | = | 6500.0 | nM | 5.19 |
| CHEMBL5555594 | — | IC50 | = | 6400.0 | nM | 5.19 |
| CHEMBL5555708 | — | IC50 | = | 7800.0 | nM | 5.11 |
| CHEMBL5561453 | — | IC50 | = | 9800.0 | nM | 5.01 |
| CHEMBL5560630 | — | IC50 | = | 10800.0 | nM | 4.97 |
| CHEMBL4297628 | RUXOTEMITIDE | IC50 | = | 11300.0 | nM | 4.95 |
| CHEMBL5555895 | — | IC50 | = | 11200.0 | nM | 4.95 |
| CHEMBL5561211 | — | IC50 | = | 11800.0 | nM | 4.93 |
| CHEMBL4297628 | RUXOTEMITIDE | IC50 | = | 13200.0 | nM | 4.88 |
| CHEMBL5561051 | — | IC50 | = | 14900.0 | nM | 4.83 |
| CHEMBL5556048 | — | IC50 | = | 16400.0 | nM | 4.79 |
| CHEMBL5564867 | — | IC50 | = | 16900.0 | nM | 4.77 |
| CHEMBL5559375 | — | IC50 | = | 23000.0 | nM | 4.64 |
| CHEMBL5556816 | — | IC50 | = | 40600.0 | nM | 4.39 |
| CHEMBL5549764 | — | IC50 | = | 80500.0 | nM | 4.09 |
| CHEMBL5566008 | — | IC50 | = | 89900.0 | nM | 4.05 |
| CHEMBL5558457 | — | IC50 | > | 300000.0 | nM | - |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 179200.0 | nM | - |