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Assay Detail

CHEMBL1963822

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: DCAMKL1
ChEMBL ↗
615
Total Activities
605
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Category other
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Serine/threonine-protein kinase DCLK1 (CHEMBL5683) ↗
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

PubChem BioAssay data set

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 615 5.62 7.40

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1981047 — — 1 7.40
CHEMBL509032 TAE-684 — 1 7.40
CHEMBL1993661 — — 1 6.90
CHEMBL2000114 — — 1 6.50
CHEMBL1971029 — — 1 6.50
CHEMBL1983309 — — 1 6.20
CHEMBL1973540 — — 1 6.20
CHEMBL1987034 — — 1 6.10
CHEMBL1998159 — — 1 6.10
CHEMBL1966628 — — 1 6.00
CHEMBL1984367 — — 1 6.00
CHEMBL2001751 — — 1 6.00
CHEMBL1987007 — — 1 6.00
CHEMBL1825138 — — 1 5.80
CHEMBL2001239 — — 1 5.80
CHEMBL1082440 — — 1 5.80
CHEMBL2000568 — — 1 5.70
CHEMBL1991063 — — 1 5.70
CHEMBL1993424 — — 1 5.60
CHEMBL1966035 — — 1 5.60
CHEMBL1983111 — — 1 5.60
CHEMBL592030 — — 1 5.60
CHEMBL1998121 — — 1 5.60
CHEMBL1974416 — — 1 5.60
CHEMBL1995813 — — 1 5.50
CHEMBL1975233 — — 1 5.50
CHEMBL1974870 — — 1 5.50
CHEMBL2000393 — — 1 5.50
CHEMBL1991356 — — 1 5.40
CHEMBL246970 — — 1 5.40

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1981047 — Ki = 39.81 nM 7.40
CHEMBL509032 TAE-684 Ki = 39.81 nM 7.40
CHEMBL1993661 — Ki = 125.89 nM 6.90
CHEMBL2000114 — Ki = 316.23 nM 6.50
CHEMBL1971029 — Ki = 316.23 nM 6.50
CHEMBL1973540 — Ki = 630.96 nM 6.20
CHEMBL1983309 — Ki = 630.96 nM 6.20
CHEMBL1987034 — Ki = 794.33 nM 6.10
CHEMBL1998159 — Ki = 794.33 nM 6.10
CHEMBL1966628 — Ki = 1000.0 nM 6.00
CHEMBL1987007 — Ki = 1000.0 nM 6.00
CHEMBL1984367 — Ki = 1000.0 nM 6.00
CHEMBL2001751 — Ki = 1000.0 nM 6.00
CHEMBL1825138 — Ki = 1584.89 nM 5.80
CHEMBL2001239 — Ki = 1584.89 nM 5.80
CHEMBL1082440 — Ki = 1584.89 nM 5.80
CHEMBL2000568 — Ki = 1995.26 nM 5.70
CHEMBL1991063 — Ki = 1995.26 nM 5.70
CHEMBL1974416 — Ki = 2511.89 nM 5.60
CHEMBL1993424 — Ki = 2511.89 nM 5.60
CHEMBL1983111 — Ki = 2511.89 nM 5.60
CHEMBL1998121 — Ki = 2511.89 nM 5.60
CHEMBL1966035 — Ki = 2511.89 nM 5.60
CHEMBL592030 — Ki = 2511.89 nM 5.60
CHEMBL1974870 — Ki = 3162.28 nM 5.50
CHEMBL1995813 — Ki = 3162.28 nM 5.50
CHEMBL1975233 — Ki = 3162.28 nM 5.50
CHEMBL2000393 — Ki = 3162.28 nM 5.50
CHEMBL2003638 — Ki = 3981.07 nM 5.40
CHEMBL1999931 — Ki = 3981.07 nM 5.40
CHEMBL1990885 — Ki = 3981.07 nM 5.40
CHEMBL246970 — Ki = 3981.07 nM 5.40
CHEMBL1984191 — Ki = 3981.07 nM 5.40
CHEMBL1991356 — Ki = 3981.07 nM 5.40
CHEMBL1967878 CENISERTIB Ki = 3981.07 nM 5.40
CHEMBL1997617 — Ki = 3981.07 nM 5.40
CHEMBL1992342 — Ki = 5011.87 nM 5.30
CHEMBL1975128 — Ki = 5011.87 nM 5.30
CHEMBL1991078 — Ki = 5011.87 nM 5.30
CHEMBL1973937 — Ki = 5011.87 nM 5.30
CHEMBL1966343 — Ki = 5011.87 nM 5.30
CHEMBL1988163 — Ki = 5011.87 nM 5.30
CHEMBL1970903 — Ki = 6309.57 nM 5.20
CHEMBL1994074 — Ki = 6309.57 nM 5.20
CHEMBL1988838 — Ki = 6309.57 nM 5.20
CHEMBL1988437 — Ki = 6309.57 nM 5.20
CHEMBL458997 — Ki = 6309.57 nM 5.20
CHEMBL1968791 — Ki = 7943.28 nM 5.10
CHEMBL1241473 — Ki = 7943.28 nM 5.10
CHEMBL1984274 — Ki = 7943.28 nM 5.10