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Compound Detail

CHEMBL1504429

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CC(=O)OCCCNc1cc(Sc2nc3ccccc3s2)c2nonc2c1[N+](=O)[O-]

Basic Information

ChEMBL ID CHEMBL1504429
Phase Preclinical
Structure Type MOL
InChI Key JVJXCUAWYNIAOL-UHFFFAOYSA-N
6
Targets
9
Activities
2
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

445.5
MW (Da)
4.26
ALogP
11
HBA
1
HBD
133.3
PSA (Ų)
0.18
QED
1
Ro5 Violations
8
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C18H15N5O5S2
MW 445.48
Aromatic Rings 4
Heavy Atoms 30
NP-Likeness -1.61

Activity Summary

EC50 5 meas. best 5.86
IC50 4 meas. best 5.69

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
EC50 5.86 5.59 1377.0 2
Type-1 angiotensin II receptor
CHEMBL227
IC50 5.69 5.69 2057.0 1
Streptokinase A
CHEMBL1293228
EC50 5.62 5.62 2429.0 1
Streptococcus sp. 'group A'
CHEMBL612389
EC50 5.49 5.49 3262.0 1
Streptococcus
CHEMBL612313
EC50 5.43 5.43 3700.0 1
Glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase
CHEMBL1741212
IC50 5.41 5.12 3920.0 2
Unchecked
CHEMBL612545
IC50 5.11 5.11 7736.0 1

Activity Data Samples

Top measurements by pChEMBL value

Data from ChEMBL 36 via Core Engine