Assay Detail
Binding
CHEMBL1613896
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Fluorescent Polarization Homogeneous Dose Response HTS to Identify Inhibitors of POS-1 Binding to mex-3-RNA. (Class of assay: confirmatory) [Related pubchem assays: 1833 (Project Summary), 1832 (Primary HTS)]
1690
Total Activities
1689
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Caenorhabditis elegans |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
RNA-binding protein pos-1 (CHEMBL1293304) ↗| Type | SINGLE PROTEIN |
| Organism | Caenorhabditis elegans |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 1690 | 4.66 | 6.76 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1569232 | — | — | 1 | 6.76 |
| CHEMBL1412067 | — | — | 1 | 6.44 |
| CHEMBL3190340 | — | — | 1 | 6.43 |
| CHEMBL391877 | — | — | 1 | 6.26 |
| CHEMBL1307886 | — | — | 1 | 6.26 |
| CHEMBL1506185 | — | — | 1 | 6.18 |
| CHEMBL1483095 | — | — | 1 | 6.06 |
| CHEMBL1524225 | — | — | 1 | 5.98 |
| CHEMBL1986342 | — | — | 1 | 5.97 |
| CHEMBL1452945 | — | — | 1 | 5.85 |
| CHEMBL3198643 | — | — | 1 | 5.80 |
| CHEMBL1508788 | — | — | 1 | 5.80 |
| CHEMBL1560833 | — | — | 1 | 5.75 |
| CHEMBL175266 | — | — | 1 | 5.72 |
| CHEMBL1509842 | — | — | 1 | 5.67 |
| CHEMBL1501508 | — | — | 1 | 5.66 |
| CHEMBL1466582 | — | — | 1 | 5.66 |
| CHEMBL1308830 | — | — | 1 | 5.65 |
| CHEMBL1540401 | — | — | 1 | 5.64 |
| CHEMBL1481493 | — | — | 1 | 5.62 |
| CHEMBL1598570 | — | — | 1 | 5.62 |
| CHEMBL1536682 | — | — | 1 | 5.60 |
| CHEMBL1419164 | — | — | 1 | 5.58 |
| CHEMBL1401891 | — | — | 1 | 5.58 |
| CHEMBL1531566 | — | — | 1 | 5.55 |
| CHEMBL1311174 | — | — | 1 | 5.55 |
| CHEMBL1458456 | — | — | 1 | 5.53 |
| CHEMBL1370447 | — | — | 1 | 5.50 |
| CHEMBL1598223 | — | — | 1 | 5.50 |
| CHEMBL1521250 | — | — | 1 | 5.50 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1569232 | — | EC50 | = | 173.0 | nM | 6.76 |
| CHEMBL1412067 | — | EC50 | = | 363.0 | nM | 6.44 |
| CHEMBL3190340 | — | EC50 | = | 374.0 | nM | 6.43 |
| CHEMBL1307886 | — | EC50 | = | 548.0 | nM | 6.26 |
| CHEMBL391877 | — | EC50 | = | 549.0 | nM | 6.26 |
| CHEMBL1506185 | — | EC50 | = | 660.0 | nM | 6.18 |
| CHEMBL1483095 | — | EC50 | = | 862.0 | nM | 6.06 |
| CHEMBL1524225 | — | EC50 | = | 1046.0 | nM | 5.98 |
| CHEMBL1986342 | — | EC50 | = | 1066.0 | nM | 5.97 |
| CHEMBL1452945 | — | EC50 | = | 1411.0 | nM | 5.85 |
| CHEMBL1508788 | — | EC50 | = | 1597.0 | nM | 5.80 |
| CHEMBL3198643 | — | EC50 | = | 1572.0 | nM | 5.80 |
| CHEMBL1560833 | — | EC50 | = | 1759.0 | nM | 5.75 |
| CHEMBL175266 | — | EC50 | = | 1897.0 | nM | 5.72 |
| CHEMBL1509842 | — | EC50 | = | 2126.0 | nM | 5.67 |
| CHEMBL1501508 | — | EC50 | = | 2197.0 | nM | 5.66 |
| CHEMBL1466582 | — | EC50 | = | 2180.0 | nM | 5.66 |
| CHEMBL1308830 | — | EC50 | = | 2237.0 | nM | 5.65 |
| CHEMBL1540401 | — | EC50 | = | 2295.0 | nM | 5.64 |
| CHEMBL1481493 | — | EC50 | = | 2408.0 | nM | 5.62 |
| CHEMBL1598570 | — | EC50 | = | 2370.0 | nM | 5.62 |
| CHEMBL1536682 | — | EC50 | = | 2498.0 | nM | 5.60 |
| CHEMBL1419164 | — | EC50 | = | 2619.0 | nM | 5.58 |
| CHEMBL1401891 | — | EC50 | = | 2601.0 | nM | 5.58 |
| CHEMBL1311174 | — | EC50 | = | 2826.0 | nM | 5.55 |
| CHEMBL1531566 | — | EC50 | = | 2822.0 | nM | 5.55 |
| CHEMBL1458456 | — | EC50 | = | 2974.0 | nM | 5.53 |
| CHEMBL1521250 | — | EC50 | = | 3155.0 | nM | 5.50 |
| CHEMBL1370447 | — | EC50 | = | 3152.0 | nM | 5.50 |
| CHEMBL1598223 | — | EC50 | = | 3144.0 | nM | 5.50 |
| CHEMBL1492305 | — | EC50 | = | 3393.0 | nM | 5.47 |
| CHEMBL1613004 | — | EC50 | = | 3632.0 | nM | 5.44 |
| CHEMBL1532412 | — | EC50 | = | 3956.0 | nM | 5.40 |
| CHEMBL1500850 | — | EC50 | = | 4095.0 | nM | 5.39 |
| CHEMBL1374016 | — | EC50 | = | 4194.0 | nM | 5.38 |
| CHEMBL1602950 | — | EC50 | = | 4129.0 | nM | 5.38 |
| CHEMBL1583838 | — | EC50 | = | 4266.0 | nM | 5.37 |
| CHEMBL1464656 | — | EC50 | = | 4365.0 | nM | 5.36 |
| CHEMBL1582403 | — | EC50 | = | 4357.0 | nM | 5.36 |
| CHEMBL1518827 | — | EC50 | = | 4469.0 | nM | 5.35 |
| CHEMBL1342776 | — | EC50 | = | 4557.0 | nM | 5.34 |
| CHEMBL1391547 | — | EC50 | = | 4605.0 | nM | 5.34 |
| CHEMBL1378413 | — | EC50 | = | 4601.0 | nM | 5.34 |
| CHEMBL1392231 | — | EC50 | = | 4671.0 | nM | 5.33 |
| CHEMBL1402117 | — | EC50 | = | 4856.0 | nM | 5.31 |
| CHEMBL1414842 | — | EC50 | = | 4951.0 | nM | 5.30 |
| CHEMBL3192451 | — | EC50 | = | 5066.0 | nM | 5.29 |
| CHEMBL1418568 | — | EC50 | = | 5111.0 | nM | 5.29 |
| CHEMBL1987928 | — | EC50 | = | 5165.0 | nM | 5.29 |
| CHEMBL1310138 | — | EC50 | = | 5148.0 | nM | 5.29 |