Assay Detail
Binding
CHEMBL1614122
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Fluorescent Polarization Homogeneous Dose Response HTS to Identify Inhibitors of Mex-5 Binding to TCR-2. (Class of assay: confirmatory) [Related pubchem assays: 1833 (Project Summary), 1832 (Primary HTS)]
1676
Total Activities
1675
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Caenorhabditis elegans |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Zinc finger protein mex-5 (CHEMBL1293319) ↗| Type | SINGLE PROTEIN |
| Organism | Caenorhabditis elegans |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 1676 | 4.81 | 7.09 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL175266 | — | — | 1 | 7.09 |
| CHEMBL3194876 | — | — | 1 | 7.07 |
| CHEMBL391877 | — | — | 1 | 7.00 |
| CHEMBL1255778 | BENSERAZIDE HYDROCHLORIDE | — | 1 | 6.95 |
| CHEMBL1412067 | — | — | 1 | 6.94 |
| CHEMBL66953 | PURPUROGALLIN | — | 1 | 6.82 |
| CHEMBL1419164 | — | — | 1 | 6.74 |
| CHEMBL3197557 | — | — | 1 | 6.71 |
| CHEMBL1307886 | — | — | 1 | 6.62 |
| CHEMBL1372920 | — | — | 1 | 6.54 |
| CHEMBL1340338 | — | — | 1 | 6.53 |
| CHEMBL1522155 | — | — | 1 | 6.38 |
| CHEMBL1987928 | — | — | 1 | 6.17 |
| CHEMBL1360509 | — | — | 1 | 6.14 |
| CHEMBL297453 | EPIGALOCATECHIN GALLATE | 3.0 | 1 | 6.14 |
| CHEMBL1359469 | — | — | 1 | 6.11 |
| CHEMBL470881 | OXOGLAUCINE | — | 1 | 6.08 |
| CHEMBL1325819 | — | — | 1 | 6.07 |
| CHEMBL1313485 | — | — | 1 | 6.06 |
| CHEMBL1986342 | — | — | 1 | 6.05 |
| CHEMBL1321098 | — | — | 1 | 6.03 |
| CHEMBL1413142 | — | — | 1 | 6.03 |
| CHEMBL1462002 | — | — | 1 | 5.99 |
| CHEMBL1486886 | — | — | 1 | 5.96 |
| CHEMBL1501508 | — | — | 1 | 5.96 |
| CHEMBL3199468 | — | — | 1 | 5.95 |
| CHEMBL1353004 | — | — | 1 | 5.95 |
| CHEMBL1524225 | — | — | 1 | 5.94 |
| CHEMBL1344339 | — | — | 1 | 5.93 |
| CHEMBL1335905 | — | — | 1 | 5.92 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL175266 | — | EC50 | = | 82.0 | nM | 7.09 |
| CHEMBL3194876 | — | EC50 | = | 86.0 | nM | 7.07 |
| CHEMBL391877 | — | EC50 | = | 100.0 | nM | 7.00 |
| CHEMBL1255778 | BENSERAZIDE HYDROCHLORIDE | EC50 | = | 112.0 | nM | 6.95 |
| CHEMBL1412067 | — | EC50 | = | 116.0 | nM | 6.94 |
| CHEMBL66953 | PURPUROGALLIN | EC50 | = | 152.0 | nM | 6.82 |
| CHEMBL1419164 | — | EC50 | = | 183.0 | nM | 6.74 |
| CHEMBL3197557 | — | EC50 | = | 193.0 | nM | 6.71 |
| CHEMBL1307886 | — | EC50 | = | 241.0 | nM | 6.62 |
| CHEMBL1372920 | — | EC50 | = | 289.0 | nM | 6.54 |
| CHEMBL1340338 | — | EC50 | = | 294.0 | nM | 6.53 |
| CHEMBL1522155 | — | EC50 | = | 421.0 | nM | 6.38 |
| CHEMBL1987928 | — | EC50 | = | 668.0 | nM | 6.17 |
| CHEMBL1360509 | — | EC50 | = | 731.0 | nM | 6.14 |
| CHEMBL297453 | EPIGALOCATECHIN GALLATE | EC50 | = | 727.0 | nM | 6.14 |
| CHEMBL1359469 | — | EC50 | = | 770.0 | nM | 6.11 |
| CHEMBL470881 | OXOGLAUCINE | EC50 | = | 834.0 | nM | 6.08 |
| CHEMBL1325819 | — | EC50 | = | 851.0 | nM | 6.07 |
| CHEMBL1313485 | — | EC50 | = | 868.0 | nM | 6.06 |
| CHEMBL1986342 | — | EC50 | = | 899.0 | nM | 6.05 |
| CHEMBL1321098 | — | EC50 | = | 945.0 | nM | 6.03 |
| CHEMBL1413142 | — | EC50 | = | 930.0 | nM | 6.03 |
| CHEMBL1462002 | — | EC50 | = | 1027.0 | nM | 5.99 |
| CHEMBL1486886 | — | EC50 | = | 1096.0 | nM | 5.96 |
| CHEMBL1501508 | — | EC50 | = | 1096.0 | nM | 5.96 |
| CHEMBL1353004 | — | EC50 | = | 1125.0 | nM | 5.95 |
| CHEMBL3199468 | — | EC50 | = | 1114.0 | nM | 5.95 |
| CHEMBL1524225 | — | EC50 | = | 1153.0 | nM | 5.94 |
| CHEMBL1344339 | — | EC50 | = | 1165.0 | nM | 5.93 |
| CHEMBL1540401 | — | EC50 | = | 1200.0 | nM | 5.92 |
| CHEMBL1335905 | — | EC50 | = | 1211.0 | nM | 5.92 |
| CHEMBL1401891 | — | EC50 | = | 1232.0 | nM | 5.91 |
| CHEMBL1421819 | — | EC50 | = | 1251.0 | nM | 5.90 |
| CHEMBL1452945 | — | EC50 | = | 1273.0 | nM | 5.89 |
| CHEMBL1560833 | — | EC50 | = | 1375.0 | nM | 5.86 |
| CHEMBL1605960 | — | EC50 | = | 1387.0 | nM | 5.86 |
| CHEMBL1463477 | — | EC50 | = | 1414.0 | nM | 5.85 |
| CHEMBL1500850 | — | EC50 | = | 1451.0 | nM | 5.84 |
| CHEMBL1327409 | — | EC50 | = | 1454.0 | nM | 5.84 |
| CHEMBL1970867 | — | EC50 | = | 1556.0 | nM | 5.81 |
| CHEMBL1584730 | — | EC50 | = | 1585.0 | nM | 5.80 |
| CHEMBL1562320 | — | EC50 | = | 1637.0 | nM | 5.79 |
| CHEMBL1472200 | — | EC50 | = | 1620.0 | nM | 5.79 |
| CHEMBL1481493 | — | EC50 | = | 1680.0 | nM | 5.78 |
| CHEMBL1429070 | — | EC50 | = | 1670.0 | nM | 5.78 |
| CHEMBL1576762 | — | EC50 | = | 1723.0 | nM | 5.76 |
| CHEMBL1481417 | — | EC50 | = | 1740.0 | nM | 5.76 |
| CHEMBL1601229 | — | EC50 | = | 1717.0 | nM | 5.76 |
| CHEMBL1484956 | — | EC50 | = | 1753.0 | nM | 5.76 |
| CHEMBL1613004 | — | EC50 | = | 1768.0 | nM | 5.75 |