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Assay Detail

CHEMBL1614169

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
PUBCHEM_BIOASSAY: Luminescence-based Microorganism Dose Response HTS to Identify Inhibitors of E. Coli Growth. (Class of assay: confirmatory) [Related pubchem assays: 1833 (Project Summary), 1832 (Primary HTS)]
1691
Total Activities
1690
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Category confirmatory
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

PubChem BioAssay data set

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1691 5.11 6.63

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1563623 1 6.63
CHEMBL927 CEFDINIR 4.0 1 6.28
CHEMBL1485275 1 5.34
CHEMBL1200567 1 5.33
CHEMBL1545940 1 5.19
CHEMBL1551640 1 5.13
CHEMBL1593697 1 5.06
CHEMBL1448592 1 5.03
CHEMBL3195762 1 4.85
CHEMBL3195360 1 4.79
CHEMBL1429365 1 4.74
CHEMBL339587 1 4.71
CHEMBL3194726 1 4.64
CHEMBL1414746 1 4.47
CHEMBL1492585 1 4.42
CHEMBL1538244 1 -
CHEMBL1400103 1 -
CHEMBL1301297 1 -
CHEMBL1567874 1 -
CHEMBL3198142 1 -
CHEMBL1514691 1 -
CHEMBL1577068 1 -
CHEMBL1556891 1 -
CHEMBL1301252 1 -
CHEMBL1595587 1 -
CHEMBL1301239 1 -
CHEMBL1329597 1 -
CHEMBL1360323 1 -
CHEMBL1567652 1 -
CHEMBL1987928 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1563623 EC50 = 232.0 nM 6.63
CHEMBL927 CEFDINIR EC50 = 521.0 nM 6.28
CHEMBL1485275 EC50 = 4585.0 nM 5.34
CHEMBL1200567 EC50 = 4674.0 nM 5.33
CHEMBL1545940 EC50 = 6493.0 nM 5.19
CHEMBL1551640 EC50 = 7378.0 nM 5.13
CHEMBL1593697 EC50 = 8681.0 nM 5.06
CHEMBL1448592 EC50 = 9414.0 nM 5.03
CHEMBL3195762 EC50 = 14269.0 nM 4.85
CHEMBL3195360 EC50 = 16173.0 nM 4.79
CHEMBL1429365 EC50 = 18252.0 nM 4.74
CHEMBL339587 EC50 = 19514.0 nM 4.71
CHEMBL3194726 EC50 = 22981.0 nM 4.64
CHEMBL1414746 EC50 = 34123.0 nM 4.47
CHEMBL1492585 EC50 = 37827.0 nM 4.42
CHEMBL1406795 EC50 > 110000.0 nM -
CHEMBL3189560 EC50 > 110000.0 nM -
CHEMBL1586152 EC50 > 110000.0 nM -
CHEMBL1563624 EC50 > 110000.0 nM -
CHEMBL1469444 EC50 > 110000.0 nM -
CHEMBL1508788 EC50 > 110000.0 nM -
CHEMBL1358059 EC50 > 110000.0 nM -
CHEMBL1508847 EC50 > 110000.0 nM -
CHEMBL1430184 EC50 > 110000.0 nM -
CHEMBL1327262 EC50 > 110000.0 nM -
CHEMBL1356350 EC50 > 110000.0 nM -
CHEMBL1508769 EC50 > 110000.0 nM -
CHEMBL1398052 EC50 > 110000.0 nM -
CHEMBL1413137 EC50 > 110000.0 nM -
CHEMBL1333555 EC50 > 110000.0 nM -
CHEMBL1390702 EC50 > 110000.0 nM -
CHEMBL1469130 EC50 > 110000.0 nM -
CHEMBL1429861 EC50 > 110000.0 nM -
CHEMBL1508544 EC50 > 110000.0 nM -
CHEMBL1585982 EC50 > 110000.0 nM -
CHEMBL1976839 EC50 > 110000.0 nM -
CHEMBL1350455 EC50 > 110000.0 nM -
CHEMBL1310375 EC50 > 110000.0 nM -
CHEMBL1563370 EC50 > 110000.0 nM -
CHEMBL246446 EC50 > 110000.0 nM -
CHEMBL3192762 EC50 > 110000.0 nM -
CHEMBL1602261 EC50 > 110000.0 nM -
CHEMBL1530689 EC50 > 110000.0 nM -
CHEMBL3213030 EC50 > 110000.0 nM -
CHEMBL1547446 EC50 > 110000.0 nM -
CHEMBL1469043 EC50 > 110000.0 nM -
CHEMBL1445820 EC50 > 110000.0 nM -
CHEMBL1508461 EC50 > 110000.0 nM -
CHEMBL305978 EC50 > 110000.0 nM -
CHEMBL1508452 EC50 > 110000.0 nM -