Assay Detail
Functional
CHEMBL1963941
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Dose-response confirmation of microRNA-mediated mRNA deacetylation inhibitors by fluorescence polarization assay. (Class of assay: confirmatory)
1186
Total Activities
1186
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1186 | 4.42 | 4.88 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1608481 | — | — | 1 | 4.88 |
| CHEMBL1579180 | — | — | 1 | 4.83 |
| CHEMBL1482177 | — | — | 1 | 4.82 |
| CHEMBL1373688 | — | — | 1 | 4.81 |
| CHEMBL1370330 | — | — | 1 | 4.78 |
| CHEMBL1443008 | — | — | 1 | 4.77 |
| CHEMBL1497838 | — | — | 1 | 4.75 |
| CHEMBL1560136 | — | — | 1 | 4.73 |
| CHEMBL1387807 | — | — | 1 | 4.71 |
| CHEMBL1362862 | — | — | 1 | 4.70 |
| CHEMBL282433 | DITOLYLGUANIDINE | — | 1 | 4.70 |
| CHEMBL1520090 | — | — | 1 | 4.68 |
| CHEMBL1568818 | — | — | 1 | 4.67 |
| CHEMBL1309254 | — | — | 1 | 4.67 |
| CHEMBL1568292 | — | — | 1 | 4.66 |
| CHEMBL3145283 | — | — | 1 | 4.66 |
| CHEMBL1710159 | — | — | 1 | 4.64 |
| CHEMBL1409735 | — | — | 1 | 4.63 |
| CHEMBL1419909 | — | — | 1 | 4.63 |
| CHEMBL1304508 | — | — | 1 | 4.62 |
| CHEMBL269410 | — | — | 1 | 4.62 |
| CHEMBL581225 | — | — | 1 | 4.62 |
| CHEMBL88326 | — | — | 1 | 4.62 |
| CHEMBL2002995 | — | — | 1 | 4.60 |
| CHEMBL1988862 | — | — | 1 | 4.59 |
| CHEMBL1572807 | — | — | 1 | 4.59 |
| CHEMBL1347598 | — | — | 1 | 4.59 |
| CHEMBL1480605 | — | — | 1 | 4.56 |
| CHEMBL1316631 | — | — | 1 | 4.56 |
| CHEMBL1573564 | — | — | 1 | 4.55 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1608481 | — | IC50 | = | 13100.0 | nM | 4.88 |
| CHEMBL1579180 | — | IC50 | = | 14900.0 | nM | 4.83 |
| CHEMBL1482177 | — | IC50 | = | 15200.0 | nM | 4.82 |
| CHEMBL1373688 | — | IC50 | = | 15400.0 | nM | 4.81 |
| CHEMBL1370330 | — | IC50 | = | 16700.0 | nM | 4.78 |
| CHEMBL1443008 | — | IC50 | = | 17000.0 | nM | 4.77 |
| CHEMBL1497838 | — | IC50 | = | 18000.0 | nM | 4.75 |
| CHEMBL1560136 | — | IC50 | = | 18500.0 | nM | 4.73 |
| CHEMBL1387807 | — | IC50 | = | 19300.0 | nM | 4.71 |
| CHEMBL1362862 | — | IC50 | = | 20000.0 | nM | 4.70 |
| CHEMBL282433 | DITOLYLGUANIDINE | IC50 | = | 19800.0 | nM | 4.70 |
| CHEMBL1520090 | — | IC50 | = | 21000.0 | nM | 4.68 |
| CHEMBL1309254 | — | IC50 | = | 21200.0 | nM | 4.67 |
| CHEMBL1568818 | — | IC50 | = | 21400.0 | nM | 4.67 |
| CHEMBL3145283 | — | IC50 | = | 22000.0 | nM | 4.66 |
| CHEMBL1568292 | — | IC50 | = | 21800.0 | nM | 4.66 |
| CHEMBL1710159 | — | IC50 | = | 22800.0 | nM | 4.64 |
| CHEMBL1419909 | — | IC50 | = | 23400.0 | nM | 4.63 |
| CHEMBL1409735 | — | IC50 | = | 23500.0 | nM | 4.63 |
| CHEMBL88326 | — | IC50 | = | 24250.0 | nM | 4.62 |
| CHEMBL269410 | — | IC50 | = | 24000.0 | nM | 4.62 |
| CHEMBL581225 | — | IC50 | = | 23800.0 | nM | 4.62 |
| CHEMBL1304508 | — | IC50 | = | 24200.0 | nM | 4.62 |
| CHEMBL2002995 | — | IC50 | = | 25100.0 | nM | 4.60 |
| CHEMBL1572807 | — | IC50 | = | 25970.0 | nM | 4.59 |
| CHEMBL1347598 | — | IC50 | = | 25800.0 | nM | 4.59 |
| CHEMBL1988862 | — | IC50 | = | 25500.0 | nM | 4.59 |
| CHEMBL1316631 | — | IC50 | = | 27320.0 | nM | 4.56 |
| CHEMBL1480605 | — | IC50 | = | 27500.0 | nM | 4.56 |
| CHEMBL1573564 | — | IC50 | = | 28000.0 | nM | 4.55 |
| CHEMBL1573280 | — | IC50 | = | 28020.0 | nM | 4.55 |
| CHEMBL1068 | OXCARBAZEPINE | IC50 | = | 28100.0 | nM | 4.55 |
| CHEMBL1329990 | — | IC50 | = | 29130.0 | nM | 4.54 |
| CHEMBL1543180 | — | IC50 | = | 28720.0 | nM | 4.54 |
| CHEMBL1529134 | — | IC50 | = | 29000.0 | nM | 4.54 |
| CHEMBL1517097 | — | IC50 | = | 29300.0 | nM | 4.53 |
| CHEMBL1718610 | — | IC50 | = | 29710.0 | nM | 4.53 |
| CHEMBL1332240 | — | IC50 | = | 29390.0 | nM | 4.53 |
| CHEMBL1515332 | — | IC50 | = | 30300.0 | nM | 4.52 |
| CHEMBL1725279 | SP-600125 | IC50 | = | 30850.0 | nM | 4.51 |
| CHEMBL1304640 | — | IC50 | = | 31200.0 | nM | 4.51 |
| CHEMBL1495219 | — | IC50 | = | 30800.0 | nM | 4.51 |
| CHEMBL1985537 | — | IC50 | = | 30800.0 | nM | 4.51 |
| CHEMBL1308769 | — | IC50 | = | 32000.0 | nM | 4.50 |
| CHEMBL1380812 | — | IC50 | = | 31600.0 | nM | 4.50 |
| CHEMBL1541254 | — | IC50 | = | 31600.0 | nM | 4.50 |
| CHEMBL1493286 | — | IC50 | = | 32600.0 | nM | 4.49 |
| CHEMBL1389248 | — | IC50 | = | 32200.0 | nM | 4.49 |
| CHEMBL1200938 | METHYSERGIDE MALEATE | IC50 | = | 32230.0 | nM | 4.49 |
| CHEMBL1425966 | — | IC50 | = | 33300.0 | nM | 4.48 |