Assay Detail
Binding
CHEMBL1613849
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Fluorescence polarization-based biochemical high throughput dose response assay for inhibitors of GLD-1 protein - TGE RNA interaction. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID2280, AID2290, AID2459]
77
Total Activities
77
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Caenorhabditis elegans |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Female germline-specific tumor suppressor gld-1 (CHEMBL1293302) ↗| Type | SINGLE PROTEIN |
| Organism | Caenorhabditis elegans |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 77 | 5.30 | 6.61 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1374066 | — | — | 1 | 6.61 |
| CHEMBL1495503 | — | — | 1 | 6.14 |
| CHEMBL1460312 | — | — | 1 | 6.08 |
| CHEMBL2000619 | — | — | 1 | 6.06 |
| CHEMBL1378107 | — | — | 1 | 5.96 |
| CHEMBL68500 | ALLOXAZINE | — | 1 | 5.83 |
| CHEMBL1391213 | — | — | 1 | 5.71 |
| CHEMBL1546264 | — | — | 1 | 5.62 |
| CHEMBL1987546 | — | — | 1 | 5.59 |
| CHEMBL1469144 | — | — | 1 | 5.57 |
| CHEMBL1864348 | — | — | 1 | 5.56 |
| CHEMBL1411766 | — | — | 1 | 5.56 |
| CHEMBL1469407 | — | — | 1 | 5.54 |
| CHEMBL269410 | — | — | 1 | 5.54 |
| CHEMBL1391235 | — | — | 1 | 5.53 |
| CHEMBL88326 | — | — | 1 | 5.52 |
| CHEMBL1357473 | — | — | 1 | 5.50 |
| CHEMBL166209 | — | — | 1 | 5.45 |
| CHEMBL1555842 | — | — | 1 | 5.44 |
| CHEMBL3190665 | — | — | 1 | 5.43 |
| CHEMBL1578982 | — | — | 1 | 5.41 |
| CHEMBL1425966 | — | — | 1 | 5.40 |
| CHEMBL1573564 | — | — | 1 | 5.39 |
| CHEMBL1415985 | — | — | 1 | 5.39 |
| CHEMBL1503865 | — | — | 1 | 5.39 |
| CHEMBL1381318 | — | — | 1 | 5.38 |
| CHEMBL1493286 | — | — | 1 | 5.37 |
| CHEMBL1579180 | — | — | 1 | 5.34 |
| CHEMBL1494927 | — | — | 1 | 5.33 |
| CHEMBL274921 | — | — | 1 | 5.30 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1374066 | — | IC50 | = | 247.51 | nM | 6.61 |
| CHEMBL1495503 | — | IC50 | = | 725.27 | nM | 6.14 |
| CHEMBL1460312 | — | IC50 | = | 840.5 | nM | 6.08 |
| CHEMBL2000619 | — | IC50 | = | 868.25 | nM | 6.06 |
| CHEMBL1378107 | — | IC50 | = | 1103.0 | nM | 5.96 |
| CHEMBL68500 | ALLOXAZINE | IC50 | = | 1471.0 | nM | 5.83 |
| CHEMBL1391213 | — | IC50 | = | 1961.0 | nM | 5.71 |
| CHEMBL1546264 | — | IC50 | = | 2427.0 | nM | 5.62 |
| CHEMBL1987546 | — | IC50 | = | 2594.0 | nM | 5.59 |
| CHEMBL1469144 | — | IC50 | = | 2670.0 | nM | 5.57 |
| CHEMBL1864348 | — | IC50 | = | 2755.0 | nM | 5.56 |
| CHEMBL1411766 | — | IC50 | = | 2737.0 | nM | 5.56 |
| CHEMBL1469407 | — | IC50 | = | 2900.0 | nM | 5.54 |
| CHEMBL269410 | — | IC50 | = | 2903.0 | nM | 5.54 |
| CHEMBL1391235 | — | IC50 | = | 2957.0 | nM | 5.53 |
| CHEMBL88326 | — | IC50 | = | 3047.0 | nM | 5.52 |
| CHEMBL1357473 | — | IC50 | = | 3124.0 | nM | 5.50 |
| CHEMBL166209 | — | IC50 | = | 3513.0 | nM | 5.45 |
| CHEMBL1555842 | — | IC50 | = | 3663.0 | nM | 5.44 |
| CHEMBL3190665 | — | IC50 | = | 3706.0 | nM | 5.43 |
| CHEMBL1578982 | — | IC50 | = | 3885.0 | nM | 5.41 |
| CHEMBL1425966 | — | IC50 | = | 3962.0 | nM | 5.40 |
| CHEMBL1573564 | — | IC50 | = | 4074.0 | nM | 5.39 |
| CHEMBL1415985 | — | IC50 | = | 4074.0 | nM | 5.39 |
| CHEMBL1503865 | — | IC50 | = | 4038.0 | nM | 5.39 |
| CHEMBL1381318 | — | IC50 | = | 4149.0 | nM | 5.38 |
| CHEMBL1493286 | — | IC50 | = | 4292.0 | nM | 5.37 |
| CHEMBL1579180 | — | IC50 | = | 4541.0 | nM | 5.34 |
| CHEMBL1494927 | — | IC50 | = | 4720.0 | nM | 5.33 |
| CHEMBL274921 | — | IC50 | = | 4974.0 | nM | 5.30 |
| CHEMBL1574146 | — | IC50 | = | 4968.0 | nM | 5.30 |
| CHEMBL1332240 | — | IC50 | = | 5004.0 | nM | 5.30 |
| CHEMBL1456904 | — | IC50 | = | 4963.0 | nM | 5.30 |
| CHEMBL282433 | DITOLYLGUANIDINE | IC50 | = | 5205.0 | nM | 5.28 |
| CHEMBL1308993 | — | IC50 | = | 5308.0 | nM | 5.28 |
| CHEMBL1421995 | — | IC50 | = | 5408.0 | nM | 5.27 |
| CHEMBL1553837 | — | IC50 | = | 5514.0 | nM | 5.26 |
| CHEMBL11475 | — | IC50 | = | 5581.0 | nM | 5.25 |
| CHEMBL1354016 | — | IC50 | = | 5862.0 | nM | 5.23 |
| CHEMBL1981093 | — | IC50 | = | 6196.0 | nM | 5.21 |
| CHEMBL1337685 | — | IC50 | = | 6115.0 | nM | 5.21 |
| CHEMBL456295 | OXOPURPUREINE | IC50 | = | 6152.0 | nM | 5.21 |
| CHEMBL1446983 | — | IC50 | = | 6133.0 | nM | 5.21 |
| CHEMBL1523792 | — | IC50 | = | 6228.0 | nM | 5.21 |
| CHEMBL1560136 | — | IC50 | = | 6284.0 | nM | 5.20 |
| CHEMBL1397154 | — | IC50 | = | 6631.0 | nM | 5.18 |
| CHEMBL294264 | PURPURIN | IC50 | = | 6688.0 | nM | 5.17 |
| CHEMBL1568292 | — | IC50 | = | 7148.0 | nM | 5.15 |
| CHEMBL41286 | DIACEREIN | IC50 | = | 7308.0 | nM | 5.14 |
| CHEMBL1585268 | — | IC50 | = | 7568.0 | nM | 5.12 |