| Cyclin-dependent kinase 9 CHEMBL3116 | Ki | 9.2 | 9.2 | 0.6 | 2 |
| Cyclin-dependent kinase 8 CHEMBL5719 | Ki | 8.7 | 8.7 | 2.0 | 2 |
| CDK9/cyclin T1 CHEMBL2111389 | IC50 | 7.7 | 7.7 | 20.0 | 1 |
| Cyclin-dependent kinase 5 CHEMBL4036 | Ki | 7.6 | 7.6 | 25.1 | 2 |
| Cyclin-dependent kinase 1 CHEMBL308 | Ki | 7.5 | 7.5 | 31.6 | 2 |
| Cyclin-dependent kinase 2 CHEMBL301 | Ki | 7.4 | 7.4 | 39.8 | 2 |
| Protein kinase C theta type CHEMBL3920 | Ki | 7.1 | 7.1 | 79.4 | 1 |
| Cyclin-dependent kinase 7 CHEMBL3055 | Ki | 7.0 | 7.0 | 100.0 | 2 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1B CHEMBL5543 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| CDK2/Cyclin A2 CHEMBL3038469 | IC50 | 6.77 | 6.77 | 170.0 | 1 |
| Proto-oncogene tyrosine-protein kinase ROS CHEMBL5568 | Ki | 6.6 | 6.6 | 251.2 | 1 |
| Megakaryocyte-associated tyrosine-protein kinase CHEMBL4175 | Ki | 6.5 | 6.5 | 316.2 | 1 |
| Serine/threonine-protein kinase D3 CHEMBL2595 | Ki | 6.5 | 6.5 | 316.2 | 1 |
| Mitogen-activated protein kinase 12 CHEMBL4674 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Glycogen synthase kinase-3 beta CHEMBL262 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Mitogen-activated protein kinase 13 CHEMBL2939 | Ki | 6.3 | 6.3 | 501.2 | 1 |
| SRSF protein kinase 1 CHEMBL4375 | Ki | 6.3 | 6.3 | 501.2 | 1 |
| Serine/threonine-protein kinase MRCK alpha CHEMBL4516 | Ki | 6.2 | 6.2 | 631.0 | 2 |
| Leukocyte tyrosine kinase receptor CHEMBL5627 | Ki | 6.2 | 6.2 | 631.0 | 1 |
| ALK tyrosine kinase receptor CHEMBL4247 | Ki | 6.2 | 6.2 | 631.0 | 2 |
| Serine/threonine-protein kinase TAO1 CHEMBL5261 | Ki | 6.1 | 6.1 | 794.3 | 1 |
| Glycogen synthase kinase-3 alpha CHEMBL2850 | Ki | 6.1 | 6.1 | 794.3 | 1 |
| Tyrosine-protein kinase SYK CHEMBL2599 | Ki | 6.1 | 6.1 | 794.3 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1A CHEMBL2292 | Ki | 6.1 | 6.1 | 794.3 | 1 |
| Serine/threonine-protein kinase pim-1 CHEMBL2147 | Ki | 6.1 | 6.1 | 794.3 | 1 |
| Serine/threonine-protein kinase pim-2 CHEMBL4523 | Ki | 6.0 | 6.0 | 1000.0 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 5 CHEMBL4852 | Ki | 6.0 | 6.0 | 1000.0 | 1 |
| Tyrosine-protein kinase receptor UFO CHEMBL4895 | Ki | 6.0 | 6.0 | 1000.0 | 2 |
| Leucine-rich repeat serine/threonine-protein kinase 2 CHEMBL1075104 | Ki | 6.0 | 6.0 | 1000.0 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 2 CHEMBL5330 | Ki | 6.0 | 6.0 | 1000.0 | 1 |
| Calcium/calmodulin-dependent protein kinase type II subunit gamma CHEMBL3829 | Ki | 6.0 | 6.0 | 1000.0 | 2 |
| Dual specificity protein kinase CLK4 CHEMBL4203 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Serine/threonine-protein kinase pim-3 CHEMBL5407 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Protein kinase C delta type CHEMBL2996 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Ribosomal protein S6 kinase alpha-3 CHEMBL2345 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Serine/threonine-protein kinase D2 CHEMBL4900 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Protein-tyrosine kinase 2-beta CHEMBL5469 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| Activin receptor type-1 CHEMBL5903 | Ki | 5.7 | 5.7 | 1995.3 | 2 |
| Calcium/calmodulin-dependent protein kinase type II subunit delta CHEMBL2801 | Ki | 5.7 | 5.7 | 1995.3 | 2 |
| Ephrin type-A receptor 2 CHEMBL2068 | Ki | 5.7 | 5.7 | 1995.3 | 1 |
| Interleukin-1 receptor-associated kinase 1 CHEMBL3357 | Ki | 5.6 | 5.6 | 2511.9 | 1 |
| G protein-coupled receptor kinase 5 CHEMBL5678 | Ki | 5.6 | 5.6 | 2511.9 | 1 |
| Serine/threonine-protein kinase PLK4 CHEMBL3788 | Ki | 5.5 | 5.5 | 3162.3 | 1 |
| Serine/threonine-protein kinase TBK1 CHEMBL5408 | Ki | 5.5 | 5.5 | 3162.3 | 1 |
| Mitogen-activated protein kinase 14 CHEMBL260 | Ki | 5.4 | 5.4 | 3981.1 | 1 |
| MAP kinase-interacting serine/threonine-protein kinase 2 CHEMBL4204 | Ki | 5.3 | 5.3 | 5011.9 | 1 |
| Calcium/calmodulin-dependent protein kinase type II subunit beta CHEMBL4121 | Ki | 5.3 | 5.3 | 5011.9 | 2 |
| Interleukin-1 receptor-associated kinase 4 CHEMBL3778 | Ki | 5.3 | 5.3 | 5011.9 | 1 |
| Serine/threonine-protein kinase N2 CHEMBL3032 | Ki | 5.3 | 5.3 | 5011.9 | 1 |