| Dual specificity protein kinase CLK4 CHEMBL4203 | Ki | 7.6 | 7.6 | 25.1 | 1 |
| Ribosomal protein S6 kinase alpha-5 CHEMBL4237 | Ki | 7.4 | 7.4 | 39.8 | 1 |
| Hepatocyte growth factor receptor CHEMBL3717 | Ki | 7.0 | 7.0 | 100.0 | 1 |
| Serine/threonine-protein kinase 3 CHEMBL4708 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| PAS domain-containing serine/threonine-protein kinase CHEMBL6054 | Ki | 6.6 | 6.6 | 251.2 | 1 |
| cAMP-dependent protein kinase catalytic subunit PRKX CHEMBL5818 | Ki | 6.6 | 6.6 | 251.2 | 1 |
| Aurora kinase B CHEMBL2185 | Ki | 6.6 | 6.6 | 251.2 | 1 |
| Cell division cycle 7-related protein kinase CHEMBL5443 | Ki | 6.6 | 6.6 | 251.2 | 1 |
| Serine/threonine-protein kinase PLK4 CHEMBL3788 | Ki | 6.5 | 6.5 | 316.2 | 1 |
| Aurora kinase A CHEMBL4722 | Ki | 6.5 | 6.5 | 316.2 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 2 CHEMBL5330 | Ki | 6.5 | 6.5 | 316.2 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 5 CHEMBL4852 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Serine/threonine-protein kinase Sgk2 CHEMBL5794 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| cGMP-dependent protein kinase 2 CHEMBL2896 | Ki | 6.2 | 6.2 | 631.0 | 1 |
| Tyrosine-protein kinase JAK2 CHEMBL2971 | Ki | 6.2 | 6.2 | 631.0 | 1 |
| cGMP-dependent protein kinase 1 CHEMBL4273 | Ki | 6.1 | 6.1 | 794.3 | 1 |
| Macrophage colony-stimulating factor 1 receptor CHEMBL1844 | Ki | 6.0 | 6.0 | 1000.0 | 1 |
| Vascular endothelial growth factor receptor 2 CHEMBL279 | Ki | 6.0 | 6.0 | 1000.0 | 1 |
| Glycogen synthase kinase-3 alpha CHEMBL2850 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Dual specificity protein kinase CLK2 CHEMBL4225 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Casein kinase I isoform gamma-2 CHEMBL2543 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 4 CHEMBL6166 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| Receptor-type tyrosine-protein kinase FLT3 CHEMBL1974 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| Tyrosine-protein kinase JAK3 CHEMBL2148 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| Casein kinase II subunit alpha CHEMBL3629 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| Rho-associated protein kinase 2 CHEMBL2973 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| Interleukin-1 receptor-associated kinase 4 CHEMBL3778 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| Cyclin-dependent kinase 2 CHEMBL301 | Ki | 5.7 | 5.7 | 1995.3 | 1 |
| Homeodomain-interacting protein kinase 4 CHEMBL1075167 | Ki | 5.7 | 5.7 | 1995.3 | 1 |
| Glycogen synthase kinase-3 beta CHEMBL262 | Ki | 5.7 | 5.7 | 1995.3 | 1 |
| Serine/threonine-protein kinase TAO1 CHEMBL5261 | Ki | 5.7 | 5.7 | 1995.3 | 1 |
| cAMP-dependent protein kinase catalytic subunit alpha CHEMBL4101 | Ki | 5.7 | 5.7 | 1995.3 | 1 |
| Serine/threonine-protein kinase MARK2 CHEMBL3831 | Ki | 5.7 | 5.7 | 1995.3 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 3 CHEMBL4575 | Ki | 5.6 | 5.6 | 2511.9 | 1 |
| MAP/microtubule affinity-regulating kinase 3 CHEMBL5600 | Ki | 5.6 | 5.6 | 2511.9 | 1 |
| Serine/threonine-protein kinase PLK3 CHEMBL4897 | Ki | 5.6 | 5.6 | 2511.9 | 1 |
| SRSF protein kinase 1 CHEMBL4375 | Ki | 5.6 | 5.6 | 2511.9 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1A CHEMBL2292 | Ki | 5.6 | 5.6 | 2511.9 | 1 |
| Interleukin-1 receptor-associated kinase 1 CHEMBL3357 | Ki | 5.5 | 5.5 | 3162.3 | 1 |
| Rho-associated protein kinase 1 CHEMBL3231 | Ki | 5.5 | 5.5 | 3162.3 | 1 |
| Cyclin-dependent kinase 5 CHEMBL4036 | Ki | 5.4 | 5.4 | 3981.1 | 1 |
| Cyclin-dependent kinase 1 CHEMBL308 | Ki | 5.4 | 5.4 | 3981.1 | 1 |
| Vascular endothelial growth factor receptor 3 CHEMBL1955 | Ki | 5.4 | 5.4 | 3981.1 | 1 |
| Mitogen-activated protein kinase kinase kinase 20 CHEMBL3886 | Ki | 5.4 | 5.4 | 3981.1 | 1 |
| Lymphokine-activated killer T-cell-originated protein kinase CHEMBL4896 | Ki | 5.3 | 5.3 | 5011.9 | 1 |
| Casein kinase I isoform delta CHEMBL2828 | Ki | 5.3 | 5.3 | 5011.9 | 1 |
| Ribosomal protein S6 kinase beta-1 CHEMBL4501 | Ki | 5.3 | 5.3 | 5011.9 | 1 |
| MAP kinase-interacting serine/threonine-protein kinase 2 CHEMBL4204 | Ki | 5.2 | 5.2 | 6309.6 | 1 |
| Misshapen-like kinase 1 CHEMBL5518 | Ki | 5.1 | 5.1 | 7943.3 | 1 |
| Serine/threonine-protein kinase BRSK1 CHEMBL5650 | Ki | 5.1 | 5.1 | 7943.3 | 1 |