| Receptor-type tyrosine-protein kinase FLT3 CHEMBL1974 | Ki | 8.3 | 8.3 | 5.0 | 1 |
| Macrophage colony-stimulating factor 1 receptor CHEMBL1844 | Ki | 7.7 | 7.7 | 19.9 | 1 |
| Vascular endothelial growth factor receptor 1 CHEMBL1868 | Ki | 7.7 | 7.7 | 19.9 | 1 |
| NT-3 growth factor receptor CHEMBL5608 | Ki | 7.7 | 7.7 | 19.9 | 1 |
| Proto-oncogene tyrosine-protein kinase receptor Ret CHEMBL2041 | Ki | 7.5 | 7.5 | 31.6 | 1 |
| Aurora kinase B CHEMBL2185 | Ki | 7.4 | 7.4 | 39.8 | 1 |
| Tyrosine-protein kinase receptor UFO CHEMBL4895 | Ki | 7.4 | 7.4 | 39.8 | 1 |
| Serine/threonine-protein kinase Chk2 CHEMBL2527 | Ki | 7.1 | 7.1 | 79.4 | 1 |
| Tyrosine-protein kinase Blk CHEMBL2250 | Ki | 7.0 | 7.0 | 100.0 | 1 |
| Vascular endothelial growth factor receptor 2 CHEMBL279 | Ki | 7.0 | 7.0 | 100.0 | 1 |
| Serine/threonine-protein kinase 17A CHEMBL4525 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| Ribosomal protein S6 kinase beta-1 CHEMBL4501 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| Insulin receptor CHEMBL1981 | Ki | 6.8 | 6.8 | 158.5 | 1 |
| Ribosomal protein S6 kinase alpha-3 CHEMBL2345 | Ki | 6.8 | 6.8 | 158.5 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 4 CHEMBL6166 | Ki | 6.7 | 6.7 | 199.5 | 1 |
| ALK tyrosine kinase receptor CHEMBL4247 | Ki | 6.7 | 6.7 | 199.5 | 1 |
| Tyrosine-protein kinase JAK2 CHEMBL2971 | Ki | 6.7 | 6.7 | 199.5 | 1 |
| High affinity nerve growth factor receptor CHEMBL2815 | Ki | 6.6 | 6.6 | 251.2 | 1 |
| Tyrosine-protein kinase Fer CHEMBL3982 | Ki | 6.5 | 6.5 | 316.2 | 1 |
| Vascular endothelial growth factor receptor 3 CHEMBL1955 | Ki | 6.5 | 6.5 | 316.2 | 1 |
| Protein-tyrosine kinase 2-beta CHEMBL5469 | Ki | 6.5 | 6.5 | 316.2 | 1 |
| Casein kinase I isoform delta CHEMBL2828 | Ki | 6.5 | 6.5 | 316.2 | 1 |
| Serine/threonine-protein kinase PLK4 CHEMBL3788 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Dual specificity protein kinase CLK4 CHEMBL4203 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Dual specificity protein kinase CLK2 CHEMBL4225 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Tyrosine-protein kinase ITK/TSK CHEMBL2959 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 5 CHEMBL4852 | Ki | 6.3 | 6.3 | 501.2 | 1 |
| Aurora kinase A CHEMBL4722 | Ki | 6.3 | 6.3 | 501.2 | 1 |
| BDNF/NT-3 growth factors receptor CHEMBL4898 | Ki | 6.3 | 6.3 | 501.2 | 1 |
| Tyrosine-protein kinase Lyn CHEMBL3905 | Ki | 6.3 | 6.3 | 501.2 | 1 |
| Calcium/calmodulin-dependent protein kinase type II subunit delta CHEMBL2801 | Ki | 6.2 | 6.2 | 631.0 | 1 |
| Serine/threonine-protein kinase 3 CHEMBL4708 | Ki | 6.2 | 6.2 | 631.0 | 1 |
| Tyrosine-protein kinase JAK3 CHEMBL2148 | Ki | 6.2 | 6.2 | 631.0 | 1 |
| Tyrosine-protein kinase Fyn CHEMBL1841 | Ki | 6.1 | 6.1 | 794.3 | 1 |
| Calcium/calmodulin-dependent protein kinase type II subunit gamma CHEMBL3829 | Ki | 6.1 | 6.1 | 794.3 | 1 |
| Tyrosine-protein kinase SYK CHEMBL2599 | Ki | 6.1 | 6.1 | 794.3 | 1 |
| Fibroblast growth factor receptor 3 CHEMBL2742 | Ki | 6.1 | 6.1 | 794.3 | 1 |
| Non-receptor tyrosine-protein kinase TYK2 CHEMBL3553 | Ki | 6.0 | 6.0 | 1000.0 | 1 |
| Tyrosine-protein kinase Lck CHEMBL258 | Ki | 6.0 | 6.0 | 1000.0 | 1 |
| Interleukin-1 receptor-associated kinase 4 CHEMBL3778 | Ki | 6.0 | 6.0 | 1000.0 | 1 |
| Phosphorylase b kinase gamma catalytic chain, liver/testis isoform CHEMBL2349 | Ki | 6.0 | 6.0 | 1000.0 | 1 |
| Fibroblast growth factor receptor 1 CHEMBL3650 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Serine/threonine-protein kinase N2 CHEMBL3032 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Misshapen-like kinase 1 CHEMBL5518 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Serine/threonine-protein kinase MARK2 CHEMBL3831 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 2 CHEMBL5330 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| Tyrosine-protein kinase FRK CHEMBL4223 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| STE20-like serine/threonine-protein kinase CHEMBL4202 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| Unchecked CHEMBL612545 | IC50 | 5.79 | 5.2125 | 1616.3 | 4 |
| MAP/microtubule affinity-regulating kinase 3 CHEMBL5600 | Ki | 5.7 | 5.7 | 1995.3 | 1 |