| Cell division cycle 7-related protein kinase CHEMBL5443 | Ki | 7.9 | 7.9 | 12.6 | 1 |
| Serine/threonine-protein kinase 3 CHEMBL4708 | Ki | 7.6 | 7.6 | 25.1 | 1 |
| Tyrosine-protein kinase JAK3 CHEMBL2148 | Ki | 7.2 | 7.2 | 63.1 | 1 |
| MAP/microtubule affinity-regulating kinase 3 CHEMBL5600 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| Serine/threonine-protein kinase MARK2 CHEMBL3831 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| Aurora kinase A CHEMBL4722 | Ki | 6.8 | 6.8 | 158.5 | 1 |
| Serine/threonine-protein kinase PLK4 CHEMBL3788 | Ki | 6.6 | 6.6 | 251.2 | 1 |
| Cyclin-dependent kinase 2 CHEMBL301 | Ki | 6.6 | 6.6 | 251.2 | 1 |
| Cyclin-dependent kinase 1 CHEMBL308 | Ki | 6.5 | 6.5 | 316.2 | 1 |
| Cyclin-dependent kinase 5 CHEMBL4036 | Ki | 6.5 | 6.5 | 316.2 | 1 |
| Tyrosine-protein kinase JAK2 CHEMBL2971 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Ribosomal protein S6 kinase beta-1 CHEMBL4501 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Interleukin-1 receptor-associated kinase 4 CHEMBL3778 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1A CHEMBL2292 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Aurora kinase B CHEMBL2185 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Rho-associated protein kinase 2 CHEMBL2973 | Ki | 6.3 | 6.3 | 501.2 | 1 |
| Protein kinase C delta type CHEMBL2996 | Ki | 6.2 | 6.2 | 631.0 | 1 |
| High affinity nerve growth factor receptor CHEMBL2815 | Ki | 6.2 | 6.2 | 631.0 | 1 |
| Fibroblast growth factor receptor 3 CHEMBL2742 | Ki | 6.2 | 6.2 | 631.0 | 1 |
| Tyrosine-protein kinase Blk CHEMBL2250 | Ki | 6.2 | 6.2 | 631.0 | 1 |
| LIM domain kinase 1 CHEMBL3836 | Ki | 6.2 | 6.2 | 631.0 | 1 |
| Tyrosine-protein kinase Fyn CHEMBL1841 | Ki | 6.1 | 6.1 | 794.3 | 1 |
| Tyrosine-protein kinase Lck CHEMBL258 | Ki | 6.1 | 6.1 | 794.3 | 1 |
| Vascular endothelial growth factor receptor 2 CHEMBL279 | Ki | 6.0 | 6.0 | 1000.0 | 1 |
| Tyrosine-protein kinase Lyn CHEMBL3905 | Ki | 6.0 | 6.0 | 1000.0 | 1 |
| Protein kinase C gamma type CHEMBL2938 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Glycogen synthase kinase-3 alpha CHEMBL2850 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| cAMP-dependent protein kinase catalytic subunit alpha CHEMBL4101 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| 5'-AMP-activated protein kinase catalytic subunit alpha-1 CHEMBL4045 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| MAP kinase-activated protein kinase 2 CHEMBL2208 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| BDNF/NT-3 growth factors receptor CHEMBL4898 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Vascular endothelial growth factor receptor 3 CHEMBL1955 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| Hepatocyte growth factor receptor CHEMBL3717 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| Fibroblast growth factor receptor 1 CHEMBL3650 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| Rho-associated protein kinase 1 CHEMBL3231 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| Glycogen synthase kinase-3 beta CHEMBL262 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| 3-phosphoinositide-dependent protein kinase 1 CHEMBL2534 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| Epidermal growth factor receptor CHEMBL203 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| Serine/threonine-protein kinase D2 CHEMBL4900 | Ki | 5.7 | 5.7 | 1995.3 | 1 |
| Insulin receptor CHEMBL1981 | Ki | 5.7 | 5.7 | 1995.3 | 1 |
| Serine/threonine-protein kinase PAK 4 CHEMBL4482 | Ki | 5.4 | 5.4 | 3981.1 | 1 |
| Serine/threonine-protein kinase Chk1 CHEMBL4630 | Ki | 5.4 | 5.4 | 3981.1 | 1 |
| Serine/threonine-protein kinase Chk2 CHEMBL2527 | Ki | 5.4 | 5.4 | 3981.1 | 1 |
| Serine/threonine-protein kinase Sgk2 CHEMBL5794 | Ki | 5.4 | 5.4 | 3981.1 | 1 |
| Mitogen-activated protein kinase 1 CHEMBL4040 | Ki | 5.3 | 5.3 | 5011.9 | 1 |
| Serine/threonine-protein kinase MRCK alpha CHEMBL4516 | Ki | 5.3 | 5.3 | 5011.9 | 1 |
| Mitogen-activated protein kinase 12 CHEMBL4674 | Ki | 5.2 | 5.2 | 6309.6 | 1 |
| Serine/threonine-protein kinase pim-1 CHEMBL2147 | Ki | 5.1 | 5.1 | 7943.3 | 1 |