| Vascular endothelial growth factor receptor 1 CHEMBL1868 | Ki | 8.9 | 8.9 | 1.3 | 1 |
| Receptor-type tyrosine-protein kinase FLT3 CHEMBL1974 | Ki | 8.4 | 8.4 | 4.0 | 1 |
| Aurora kinase B CHEMBL2185 | Ki | 8.4 | 8.4 | 4.0 | 1 |
| Vascular endothelial growth factor receptor 2 CHEMBL279 | Ki | 8.3 | 8.3 | 5.0 | 1 |
| Macrophage colony-stimulating factor 1 receptor CHEMBL1844 | Ki | 8.0 | 8.0 | 10.0 | 1 |
| Tyrosine-protein kinase ABL1 CHEMBL1862 | Ki | 7.4 | 7.4 | 39.8 | 1 |
| Aurora kinase A CHEMBL4722 | Ki | 7.2 | 7.2 | 63.1 | 1 |
| Vascular endothelial growth factor receptor 3 CHEMBL1955 | Ki | 7.1 | 7.1 | 79.4 | 1 |
| Tyrosine-protein kinase Lck CHEMBL258 | Ki | 7.1 | 7.1 | 79.4 | 1 |
| Tyrosine-protein kinase Blk CHEMBL2250 | Ki | 7.0 | 7.0 | 100.0 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 2 CHEMBL5330 | Ki | 7.0 | 7.0 | 100.0 | 1 |
| Tyrosine-protein kinase receptor UFO CHEMBL4895 | Ki | 7.0 | 7.0 | 100.0 | 1 |
| Tyrosine-protein kinase Lyn CHEMBL3905 | Ki | 6.8 | 6.8 | 158.5 | 1 |
| Serine/threonine-protein kinase PLK4 CHEMBL3788 | Ki | 6.8 | 6.8 | 158.5 | 1 |
| Homeodomain-interacting protein kinase 2 CHEMBL4576 | Ki | 6.8 | 6.8 | 158.5 | 1 |
| Serine/threonine-protein kinase Nek2 CHEMBL3835 | Ki | 6.7 | 6.7 | 199.5 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 4 CHEMBL6166 | Ki | 6.6 | 6.6 | 251.2 | 1 |
| Homeodomain-interacting protein kinase 4 CHEMBL1075167 | Ki | 6.6 | 6.6 | 251.2 | 1 |
| Misshapen-like kinase 1 CHEMBL5518 | Ki | 6.5 | 6.5 | 316.2 | 1 |
| Serine/threonine-protein kinase 3 CHEMBL4708 | Ki | 6.5 | 6.5 | 316.2 | 1 |
| Hepatocyte growth factor receptor CHEMBL3717 | Ki | 6.5 | 6.5 | 316.2 | 1 |
| Tyrosine-protein kinase Fer CHEMBL3982 | Ki | 6.5 | 6.5 | 316.2 | 1 |
| NT-3 growth factor receptor CHEMBL5608 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Tyrosine-protein kinase FRK CHEMBL4223 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| STE20-like serine/threonine-protein kinase CHEMBL4202 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Tyrosine-protein kinase Fyn CHEMBL1841 | Ki | 6.3 | 6.3 | 501.2 | 1 |
| Mast/stem cell growth factor receptor Kit CHEMBL1936 | Ki | 6.2 | 6.2 | 631.0 | 1 |
| Rho-associated protein kinase 2 CHEMBL2973 | Ki | 6.2 | 6.2 | 631.0 | 1 |
| Fibroblast growth factor receptor 1 CHEMBL3650 | Ki | 6.2 | 6.2 | 631.0 | 1 |
| Focal adhesion kinase 1 CHEMBL2695 | Ki | 6.1 | 6.1 | 794.3 | 1 |
| Casein kinase I isoform gamma-2 CHEMBL2543 | Ki | 6.0 | 6.0 | 1000.0 | 1 |
| Rho-associated protein kinase 1 CHEMBL3231 | Ki | 6.0 | 6.0 | 1000.0 | 1 |
| Tyrosine-protein kinase Fes/Fps CHEMBL5455 | Ki | 6.0 | 6.0 | 1000.0 | 1 |
| ALK tyrosine kinase receptor CHEMBL4247 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Casein kinase I isoform gamma-1 CHEMBL2426 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| 5'-AMP-activated protein kinase catalytic subunit alpha-1 CHEMBL4045 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| Tyrosine-protein kinase SYK CHEMBL2599 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| LIM domain kinase 1 CHEMBL3836 | Ki | 5.7 | 5.7 | 1995.3 | 1 |
| Serine/threonine-protein kinase TAO1 CHEMBL5261 | Ki | 5.7 | 5.7 | 1995.3 | 1 |
| BDNF/NT-3 growth factors receptor CHEMBL4898 | Ki | 5.6 | 5.6 | 2511.9 | 1 |
| High affinity nerve growth factor receptor CHEMBL2815 | Ki | 5.6 | 5.6 | 2511.9 | 1 |
| SRSF protein kinase 1 CHEMBL4375 | Ki | 5.5 | 5.5 | 3162.3 | 1 |
| MAP/microtubule affinity-regulating kinase 3 CHEMBL5600 | Ki | 5.4 | 5.4 | 3981.1 | 1 |
| Serine/threonine-protein kinase Nek4 CHEMBL5819 | Ki | 5.4 | 5.4 | 3981.1 | 1 |
| Serine/threonine-protein kinase MARK2 CHEMBL3831 | Ki | 5.4 | 5.4 | 3981.1 | 1 |
| MAP kinase-interacting serine/threonine-protein kinase 2 CHEMBL4204 | Ki | 5.3 | 5.3 | 5011.9 | 1 |
| Mitogen-activated protein kinase kinase kinase 20 CHEMBL3886 | Ki | 5.3 | 5.3 | 5011.9 | 1 |
| Serine/threonine-protein kinase D2 CHEMBL4900 | Ki | 5.2 | 5.2 | 6309.6 | 1 |
| Dual specificity protein kinase CLK2 CHEMBL4225 | Ki | 5.2 | 5.2 | 6309.6 | 1 |
| Lymphokine-activated killer T-cell-originated protein kinase CHEMBL4896 | Ki | 5.1 | 5.1 | 7943.3 | 1 |