| Dual specificity protein kinase CLK4 CHEMBL4203 | Ki | 8.0 | 8.0 | 10.0 | 1 |
| Casein kinase I isoform gamma-2 CHEMBL2543 | Ki | 7.3 | 7.3 | 50.1 | 1 |
| Cyclin-dependent kinase 9 CHEMBL3116 | Ki | 7.2 | 7.2 | 63.1 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 3 CHEMBL4575 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| Interleukin-1 receptor-associated kinase 1 CHEMBL3357 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1B CHEMBL5543 | Ki | 6.8 | 6.8 | 158.5 | 1 |
| Casein kinase I isoform gamma-1 CHEMBL2426 | Ki | 6.8 | 6.8 | 158.5 | 1 |
| Cyclin-dependent kinase 7 CHEMBL3055 | Ki | 6.7 | 6.7 | 199.5 | 1 |
| Interleukin-1 receptor-associated kinase 4 CHEMBL3778 | Ki | 6.6 | 6.6 | 251.2 | 1 |
| Vascular endothelial growth factor receptor 2 CHEMBL279 | Ki | 6.6 | 6.6 | 251.2 | 1 |
| Dual specificity protein kinase CLK2 CHEMBL4225 | Ki | 6.6 | 6.6 | 251.2 | 1 |
| Cyclin-dependent kinase 5 CHEMBL4036 | Ki | 6.5 | 6.5 | 316.2 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1A CHEMBL2292 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Cyclin-dependent kinase 1 CHEMBL308 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Tyrosine-protein kinase ITK/TSK CHEMBL2959 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| STE20-like serine/threonine-protein kinase CHEMBL4202 | Ki | 6.3 | 6.3 | 501.2 | 1 |
| Mitogen-activated protein kinase 8 CHEMBL2276 | Ki | 6.2 | 6.2 | 631.0 | 1 |
| Homeodomain-interacting protein kinase 2 CHEMBL4576 | Ki | 6.2 | 6.2 | 631.0 | 1 |
| Leucine-rich repeat serine/threonine-protein kinase 2 CHEMBL1075104 | Ki | 6.1 | 6.1 | 794.3 | 1 |
| Casein kinase I isoform delta CHEMBL2828 | Ki | 6.1 | 6.1 | 794.3 | 1 |
| Macrophage colony-stimulating factor 1 receptor CHEMBL1844 | Ki | 6.1 | 6.1 | 794.3 | 1 |
| Serine/threonine-protein kinase Sgk2 CHEMBL5794 | Ki | 6.1 | 6.1 | 794.3 | 1 |
| Tyrosine-protein kinase ABL1 CHEMBL1862 | Ki | 6.1 | 6.1 | 794.3 | 1 |
| Serine/threonine-protein kinase Nek4 CHEMBL5819 | Ki | 6.1 | 6.1 | 794.3 | 1 |
| Platelet-derived growth factor receptor beta CHEMBL1913 | Ki | 6.1 | 6.1 | 794.3 | 1 |
| Vascular endothelial growth factor receptor 3 CHEMBL1955 | Ki | 6.0 | 6.0 | 1000.0 | 1 |
| SRSF protein kinase 1 CHEMBL4375 | Ki | 6.0 | 6.0 | 1000.0 | 1 |
| Mitogen-activated protein kinase kinase kinase 20 CHEMBL3886 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Cyclin-dependent kinase 2 CHEMBL301 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Misshapen-like kinase 1 CHEMBL5518 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 5 CHEMBL4852 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Aurora kinase B CHEMBL2185 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| MAP/microtubule affinity-regulating kinase 3 CHEMBL5600 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| Maternal embryonic leucine zipper kinase CHEMBL4578 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| Serine/threonine-protein kinase TAO1 CHEMBL5261 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 2 CHEMBL5330 | Ki | 5.7 | 5.7 | 1995.3 | 1 |
| Hepatocyte growth factor receptor CHEMBL3717 | Ki | 5.7 | 5.7 | 1995.3 | 1 |
| Glycogen synthase kinase-3 beta CHEMBL262 | Ki | 5.6 | 5.6 | 2511.9 | 1 |
| Homeodomain-interacting protein kinase 4 CHEMBL1075167 | Ki | 5.5 | 5.5 | 3162.3 | 1 |
| Casein kinase I isoform alpha CHEMBL2793 | Ki | 5.5 | 5.5 | 3162.3 | 1 |
| Phosphorylase b kinase gamma catalytic chain, liver/testis isoform CHEMBL2349 | Ki | 5.5 | 5.5 | 3162.3 | 1 |
| Serine/threonine-protein kinase MARK2 CHEMBL3831 | Ki | 5.4 | 5.4 | 3981.1 | 1 |
| Serine/threonine-protein kinase D2 CHEMBL4900 | Ki | 5.3 | 5.3 | 5011.9 | 1 |
| Serine/threonine-protein kinase 3 CHEMBL4708 | Ki | 5.3 | 5.3 | 5011.9 | 1 |
| Casein kinase II subunit alpha CHEMBL3629 | Ki | 5.3 | 5.3 | 5011.9 | 1 |
| Calcium/calmodulin-dependent protein kinase type II subunit delta CHEMBL2801 | Ki | 5.3 | 5.3 | 5011.9 | 1 |
| MAP kinase-interacting serine/threonine-protein kinase 2 CHEMBL4204 | Ki | 5.2 | 5.2 | 6309.6 | 1 |