| Cell division cycle 7-related protein kinase CHEMBL5443 | Ki | 8.7 | 8.7 | 2.0 | 1 |
| Misshapen-like kinase 1 CHEMBL5518 | Ki | 8.2 | 8.2 | 6.3 | 1 |
| Serine/threonine-protein kinase MRCK alpha CHEMBL4516 | Ki | 7.4 | 7.4 | 39.8 | 1 |
| 3-phosphoinositide-dependent protein kinase 1 CHEMBL2534 | Ki | 7.1 | 7.1 | 79.4 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 3 CHEMBL4575 | Ki | 7.0 | 7.0 | 100.0 | 1 |
| Serine/threonine-protein kinase N2 CHEMBL3032 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| Dual specificity protein kinase CLK4 CHEMBL4203 | Ki | 6.8 | 6.8 | 158.5 | 1 |
| NT-3 growth factor receptor CHEMBL5608 | Ki | 6.7 | 6.7 | 199.5 | 1 |
| Proto-oncogene tyrosine-protein kinase ROS CHEMBL5568 | Ki | 6.7 | 6.7 | 199.5 | 1 |
| Testis-specific serine/threonine-protein kinase 1 CHEMBL6003 | Ki | 6.6 | 6.6 | 251.2 | 1 |
| Dual specificity mitogen-activated protein kinase kinase 1 CHEMBL3587 | Ki | 6.6 | 6.6 | 251.2 | 1 |
| Casein kinase II subunit alpha CHEMBL3629 | Ki | 6.6 | 6.6 | 251.2 | 1 |
| Maternal embryonic leucine zipper kinase CHEMBL4578 | Ki | 6.5 | 6.5 | 316.2 | 1 |
| Serine/threonine-protein kinase Chk2 CHEMBL2527 | Ki | 6.5 | 6.5 | 316.2 | 1 |
| Protein kinase C delta type CHEMBL2996 | Ki | 6.5 | 6.5 | 316.2 | 1 |
| Tyrosine-protein kinase SYK CHEMBL2599 | Ki | 6.5 | 6.5 | 316.2 | 1 |
| cAMP-dependent protein kinase catalytic subunit alpha CHEMBL4101 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 2 CHEMBL5330 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Tyrosine-protein kinase Fer CHEMBL3982 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Tyrosine-protein kinase Blk CHEMBL2250 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| cAMP-dependent protein kinase catalytic subunit PRKX CHEMBL5818 | Ki | 6.3 | 6.3 | 501.2 | 1 |
| Protein kinase C gamma type CHEMBL2938 | Ki | 6.3 | 6.3 | 501.2 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1B CHEMBL5543 | Ki | 6.3 | 6.3 | 501.2 | 1 |
| Serine/threonine-protein kinase PLK1 CHEMBL3024 | Ki | 6.3 | 6.3 | 501.2 | 1 |
| Ribosomal protein S6 kinase beta-1 CHEMBL4501 | Ki | 6.3 | 6.3 | 501.2 | 1 |
| cGMP-dependent protein kinase 1 CHEMBL4273 | Ki | 6.3 | 6.3 | 501.2 | 1 |
| STE20-like serine/threonine-protein kinase CHEMBL4202 | Ki | 6.3 | 6.3 | 501.2 | 1 |
| Homeodomain-interacting protein kinase 2 CHEMBL4576 | Ki | 6.2 | 6.2 | 631.0 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1A CHEMBL2292 | Ki | 6.2 | 6.2 | 631.0 | 1 |
| Tyrosine-protein kinase Lyn CHEMBL3905 | Ki | 6.2 | 6.2 | 631.0 | 1 |
| Macrophage-stimulating protein receptor CHEMBL2689 | Ki | 6.1 | 6.1 | 794.3 | 1 |
| Serine/threonine-protein kinase Sgk2 CHEMBL5794 | Ki | 6.1 | 6.1 | 794.3 | 1 |
| MAP/microtubule affinity-regulating kinase 3 CHEMBL5600 | Ki | 6.1 | 6.1 | 794.3 | 1 |
| Epidermal growth factor receptor CHEMBL203 | Ki | 6.1 | 6.1 | 794.3 | 1 |
| Serine/threonine-protein kinase PAK 4 CHEMBL4482 | Ki | 6.1 | 6.1 | 794.3 | 1 |
| Vascular endothelial growth factor receptor 3 CHEMBL1955 | Ki | 6.0 | 6.0 | 1000.0 | 1 |
| Protein kinase C iota type CHEMBL2598 | Ki | 6.0 | 6.0 | 1000.0 | 1 |
| Aurora kinase B CHEMBL2185 | Ki | 6.0 | 6.0 | 1000.0 | 1 |
| Serine/threonine-protein kinase 3 CHEMBL4708 | Ki | 6.0 | 6.0 | 1000.0 | 1 |
| Ribosomal protein S6 kinase alpha-3 CHEMBL2345 | Ki | 6.0 | 6.0 | 1000.0 | 1 |
| Serine/threonine-protein kinase Chk1 CHEMBL4630 | Ki | 6.0 | 6.0 | 1000.0 | 1 |
| Casein kinase I isoform gamma-2 CHEMBL2543 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Homeodomain-interacting protein kinase 4 CHEMBL1075167 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Glycogen synthase kinase-3 alpha CHEMBL2850 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Casein kinase I isoform delta CHEMBL2828 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 5 CHEMBL4852 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Protein kinase C zeta type CHEMBL3438 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 4 CHEMBL1075115 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Interleukin-1 receptor-associated kinase 4 CHEMBL3778 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Glycogen synthase kinase-3 beta CHEMBL262 | Ki | 5.9 | 5.9 | 1258.9 | 1 |